Publications

Giuseppe BIFULCO Publications


2018
Articolo in rivista
Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol
MEDCHEMCOMM. Vol. 9. Pag.2028-2036
ISSN:2040-2503.
Lauro, G.; Cantone, V.; Potenza, M.; Fischer, K.; Koeberle, A.; Werz, O.; Riccio, R.; Bifulco, G.
Versione online
Digital Object Identifier (DOI): 10.1039/c8md00497h
Codice identificativo ISI: WOS:000453225200005
Codice identificativo SCOPUS: 2-s2.0-85058623321
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2018
Articolo in rivista
Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation
ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 16. Pag.9138-9142
ISSN:1477-0520.
Jachak, G. R.; Athawale, P. R.; Agarwal, H.; Barthwal, M. K.; Lauro, G.; Bifulco, G.; Srinivasa Reddy, D.
Versione online
Digital Object Identifier (DOI): 10.1039/c8ob02713g
Codice identificativo ISI: WOS:000452321100006
Codice identificativo SCOPUS: 2-s2.0-85058177071
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2018
Articolo in rivista
Discovery of new potent molecular entities able to inhibit mPGES-1
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 143. Pag.1419-1427
ISSN:0223-5234.
Di Micco, Simone; Terracciano, Stefania; Cantone, Vincenza; Fischer, Katrin; Koeberle, Andreas; Foglia, Antonio; Riccio, Raffaele; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1016/j.ejmech.2017.10.039
Codice identificativo ISI: WOS:000423641400021
Codice identificativo SCOPUS: 2-s2.0-85033582141
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2018
Articolo in rivista
Down regulation of pro-inflammatory pathways by tanshinone IIA and cryptotanshinone in a non-genetic mouse model of Alzheimer's disease
PHARMACOLOGICAL RESEARCH. Vol. 129. Pag.482-490
ISSN:1043-6618.
Maione, Francesco; Piccolo, Marialuisa; DE VITA, Simona; Chini, Maria Giovanna; Cristiano, Claudia; De Caro, Carmen; Lippiello, Pellegrino; Miniaci, Maria Concetta; Santamaria, Rita; Irace, Carlo; De Feo, Vincenzo; Calignano, Antonio; Mascolo, Nicola; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1016/j.phrs.2017.11.018
Codice identificativo ISI: WOS:000428102600045
Codice identificativo SCOPUS: 2-s2.0-85034994652
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2018
Articolo in rivista
Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors
BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 26. Pag.3953-3957
ISSN:0968-0896.
DI MICCO, Simone; Pulvirenti, Luana; Bruno, Ines; Terracciano, Stefania; Russo, Alessandra; Vaccaro, Mariacarmela; Ruggiero, Dafne; Muccilli, Vera; Cardullo, Nunzio; Tringali, Corrado; Riccio, Raffaele; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1016/j.bmc.2018.06.019
Codice identificativo ISI: WOS:000440942100012
Codice identificativo SCOPUS: 2-s2.0-85048836726
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2018
Articolo in rivista
Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics
CHEMICAL COMMUNICATIONS. Vol. 54. Pag.7613-7616
ISSN:1359-7345.
Terracciano, Stefania; LAURO, GIANLUIGI; Russo, Alessandra; Vaccaro, Maria Carmela; VASSALLO, ANTONIO; De Marco, Margot; Ranieri, Bianca; Rosati, Alessandra; Turco, Maria Caterina; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Versione online
Digital Object Identifier (DOI): 10.1039/c8cc03399d
Codice identificativo ISI: WOS:000442118800009
Codice identificativo SCOPUS: 2-s2.0-85049623511
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2018
Articolo in rivista
Discovery of new erbB4 inhibitors: Repositioning an orphan chemical library by inverse virtual screening
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 152. Pag.253-263
ISSN:0223-5234.
Giordano, Assunta; Forte, Giovanni; Massimo, Luigia; Riccio, Raffaele; Bifulco, Giuseppe; Di Micco, Simone
Digital Object Identifier (DOI): 10.1016/j.ejmech.2018.04.018
Codice identificativo ISI: WOS:000435048900020
Codice identificativo SCOPUS: 2-s2.0-85046405635
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2018
Articolo in rivista
Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells
JOURNAL OF NATURAL PRODUCTS. Vol. 81. Pag.1786-1794
ISSN:0163-3864.
Khalfaoui, Ayoub; Chini, Maria G.; Bouheroum, Mohamed; Belaabed, Soumia; Lauro, Gianluigi; Terracciano, Stefania; Vaccaro, Mariacarmela; Bruno, Ines; Benayache, Samir; Mancini, Ines; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jnatprod.8b00234
Codice identificativo ISI: WOS:000443103700011
Codice identificativo SCOPUS: 2-s2.0-85052588349
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2018
Articolo in rivista
Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain
SCIENTIFIC REPORTS. Vol. 8. Pag.1709-1709
ISSN:2045-2322.
Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines
Versione online
Digital Object Identifier (DOI): 10.1038/s41598-017-14902-y
Codice identificativo ISI: WOS:000423428300037
Codice identificativo SCOPUS: 2-s2.0-85041134440
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