Publications

Maria Chiara MONTI Publications


2023
Articolo in rivista
Targeting USP-7 by a Novel Fluorinated 5-Pyrazolyl-Urea Derivative
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. Vol. 24. Pag.9200-9212
ISSN:1422-0067.
Morretta, Elva; Brullo, Chiara; Belvedere, Raffaella; Petrella, Antonello; Spallarossa, Andrea; Monti, Maria Chiara
Digital Object Identifier (DOI): 10.3390/ijms24119200
Codice identificativo ISI: WOS:001005902200001
Codice identificativo SCOPUS: 2-s2.0-85161663715
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2023
Articolo in rivista
A multidisciplinary functional proteomics-aided strategy as a tool for the profiling of a novel cytotoxic thiadiazolopyrimidone
BIOORGANIC CHEMISTRY. Vol. 138. Pag.106620-106632
ISSN:0045-2068.
Morretta, Elva; Ruggiero, Dafne; Belvedere, Raffaella; Petrella, Antonello; Bruno, Ines; Terracciano, Stefania; Monti, Maria Chiara
Versione online
Digital Object Identifier (DOI): 10.1016/j.bioorg.2023.106620
Codice identificativo ISI: WOS:001011723900001
Codice identificativo SCOPUS: 2-s2.0-85159816112
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2023
Articolo in rivista
Discovery of BAR502, as potent steroidal antagonist of leukemia inhibitory factor receptor for the treatment of pancreatic adenocarcinoma
FRONTIERS IN ONCOLOGY. Vol. 13. Pag.1140730-1140746
ISSN:2234-943X.
Di Giorgio, Cristina; Bellini, Rachele; Lupia, Antonio; Massa, Carmen; Bordoni, Martina; Marchianò, Silvia; Rosselli, Rosalinda; Sepe, Valentina; Rapacciuolo, Pasquale; Moraca, Federica; Morretta, Elva; Ricci, Patrizia; Urbani, Ginevra; Monti, Maria Chiara; Biagioli, Michele; Distrutti, Eleonora; Catalanotti, Bruno; Zampella, Angela; Fiorucci, Stefano
Digital Object Identifier (DOI): 10.3389/fonc.2023.1140730
Codice identificativo ISI: WOS:000956766300001
Codice identificativo SCOPUS: 2-s2.0-85150864923
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2023
Articolo in rivista
Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor
JOURNAL OF MEDICINAL CHEMISTRY. Pag.1-19
ISSN:0022-2623.
Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c01030
Codice identificativo ISI: WOS:001045914800001
Codice identificativo SCOPUS: 2-s2.0-85168362422
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2023
Articolo in rivista
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 247. Pag.115018-115018
ISSN:0223-5234.
Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi
Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.115018
Codice identificativo ISI: WOS:000913013400001
Codice identificativo SCOPUS: 2-s2.0-85144788456
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2023
Articolo in rivista
Curcumin Has Beneficial Effects on Lysosomal Alpha-Galactosidase: Potential Implications for the Cure of Fabry Disease
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. Vol. 24. Pag.1095-1109
ISSN:1422-0067.
Monticelli, Maria; Hay Mele, Bruno; Allocca, Mariateresa; Liguori, Ludovica; Lukas, Jan; Monti, Maria Chiara; Morretta, Elva; Cubellis, Maria Vittoria; Andreotti, Giuseppina
Digital Object Identifier (DOI): 10.3390/ijms24021095
Codice identificativo ISI: WOS:000918253800001
Codice identificativo SCOPUS: 2-s2.0-85146812544
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2023
Articolo in rivista
Combinatorial therapy with BAR502 and UDCA resets FXR and GPBAR1 signaling and reverses liver histopathology in a model of NASH
SCIENTIFIC REPORTS. Vol. 13. Pag.1602-1617
ISSN:2045-2322.
Marchiano, S.; Biagioli, M.; Morretta, E.; Di Giorgio, C.; Roselli, R.; Bordoni, M.; Bellini, R.; Urbani, G.; Massa, C.; Monti, M. C.; Zampella, A.; Distrutti, E.; Fiorucci, S.
Versione online
Digital Object Identifier (DOI): 10.1038/s41598-023-28647-4
Codice identificativo ISI: WOS:000923285800038
Codice identificativo SCOPUS: 2-s2.0-85146959582
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