PHARMACOLOGY AND PHARMACOTHERAPY

Rosalinda SORRENTINO PHARMACOLOGY AND PHARMACOTHERAPY

0760200020
DIPARTIMENTO DI FARMACIA
EQF7
PHARMACEUTICAL CHEMISTRY AND TECHNOLOGY
2020/2021

OBBLIGATORIO
YEAR OF COURSE 4
YEAR OF DIDACTIC SYSTEM 2016
PRIMO SEMESTRE
CFUHOURSACTIVITY
1FARMACOLOGIA GENERALE MODULO DI FARMACOLOGIA E FARMACOTERAPIA
540LESSONS
2FARMACOTERAPIA MODULO DI FARMACOLOGIA E FARMACOTERAPIA
540LESSONS
Objectives
THE COURSE HAS THE SCOPE TO PROVIDE KNOWLEDGE AND COMPREHENSION OF THE FUNDAMENTALS OF PHARMACOKINETICS AND PHARMACODYNAMICS TO BE APPLIED TO THE CLASS OF DRUGS THAT WILL BE STUDIED. THE INDIVIDUAL CLASSES OF DRUGS WILL BE RELATED TO THE BIOLOGY OF THE PATHOLOGY IN ORDER TO BE ABLE TO APPROACH THE THERAPEUTIC STRATEGY ACCORDING TO THE MECHANISM OF ACTION AND SIDE EFFECTS, AS WELL AS ADVERSE EVENTS, RELATED TO THE SPECIFIC CLINICALLY USED DRUGS. PARTICULAR ATTENTION WILL BE PAID ONTO NOVEL AND INNOVATIVE THERAPEUTIC STRATEGIES UNDER CLINICAL STUDIES IN ORDER TO EVALUATE BOTH ALTERNATIVE THERAPEUTIC AND INNOVATIVE APPROACHES IN FAVOUR OF AMELIORATION OF THE PHARMACOLOGICAL EFFICACY AND TO CIRCUMVENT NON-RESPONSIVENESS.
THE STUDENT WILL HAVE TO DEMONSTRATE THE ACQUIRED SKILLS BY EXPLAINING HOW TO MANAGE THE THERAPEUTIC APPROACH TO CURE THE PATHOLOGIES CONSIDERED DURING THE COURSE. IT IS OF PARTICULAR RELEVANCE THE USAGE OF AN APPROPRIATE SCIENTIFIC LANGUAGE TO EXPOSE THE ACQUIRED SKILLS.
Prerequisites
THE STUDENT SHOULD HAVE ACQUIRED KNOWLEDGE OF ANATOMY AND PHYSIOLOGY, BIOCHEMISTRY AND PATHOLOGY.
Contents
GENERAL PHARMACOLOGY: DEFINITION/S. DOSES. DOSE/EFFECT RESPONSE AND ITS ANALYSIS. DRUG/RECEPTOR INTERACTION AND ITS ANALYSIS. THERAPEUTIC INDEX. PLACEBO. HOMEOPATHY. PHASES OF THE STUDY OF NEW DRUGS. CONTROL AND DRUG INFORMATION.
PHARMACOKINETICS: ROUTES OF ADMINISTRATION. ABSORPTION. DISTRIBUTION. METABOLISM. EXCRETION. PHARMACOKINETIC INTERACTIONS.
PHARMACODYNAMICS: INTERACTION DRUG/RECEPTOR. AGONIST. PD2. ANTAGONIST. PA2. PARTIAL AGONIST/ANTAGONIST. TRANSDUCTION OF DRUG/RECEPTOR INTERACTION. IONOTROPIC RECEPTORS. METABOTROPIC RECEPTORS. VOLTAGE-GATED ION CHANNELS. INTRACELLULAR RECEPTORS. RECEPTORS FOR GROWTH FACTORS. INTRACELLULAR TRANSDUCTION MECHANISMS. CALCIUM HOMEOSTASIS. PHARMACODYNAMIC INTERACTIONS.

PHARMACOTHERAPY: NOMENCLATURE AND CLASSIFICATION OF DRUGS. PERIPHERAL NERVOUS SYSTEM AND ITS MEDIATORS. PARASYMPATHOMIMETICS. PARASYMPATHOLYTICS. SYMPATHOMIMETICS. SYMPATHOLYTICS. INHIBITORS OF ADRENERGIC NEURON. NEUROMUSCULAR BLOCKERS. DRUGS FOR GANGLIA. LOCAL ANESTHETICS. CENTRAL NERVOUS SYSTEM AND ITS MEDIATORS. GENERAL ANESTHETICS. SEDATIVES AND HYPNOTICS. CENTRAL NERVOUS SYSTEM STIMULANTS. ANXIOLYTICS. ANTI-PSYCHOTICS. ANTI-DEPRESSANTS. ANTI-EPILEPTIC. TREATMENT OF PARKINSON DISEASE. TREATMENT OF ALZHEIMER DISEASE. MUSCLE RELAXANTS. OPIOID ANALGESICS. AUTACOIDS: HISTAMINE, SEROTONIN, EICOSANOIDS, PAF, NITROGEN OXIDE. VASOACTIVE PEPTIDES: RENIN/ANGIOTENSIN SYSTEM, BRADYKININ, ENDOTHELIN. ANTI-HYPERTENSIVES. ANTI-ANGINAL. ANTI-ARRHYTHMICS. INOTROPES POSITIVE. ANTI-ANGIOEDEMA TREATMENT OF HYPERLIPIDEMIA. TREATMENT OF DIABETES. DIURETICS. ANTI-INFLAMMATORY. ANTI-GOUT. ANTI-ASTHMATICS. IMMUNOMODULATORS. ANTI-ACIDS AND ANTI-ULCER. ANTI-COAGULANTS. ANTI-THROMBOTIC. THROMBOLYSIS. DRUGS OF UTERINE MOTILITY. SEX HORMONES AND THEIR PHARMACOLOGICAL REGULATION.
Teaching Methods
THE COURSE INCLUDES 80 HOURS OF FRONTAL ASSISTED TEACHING (10 CFU).
ATTENDANCE IS MANDATORY. TO TAKE THE FINAL EXAM, THE STUDENT MUST HAVE ATTENDED AT LEAST 75% OF THE TEACHING HOURS. THE PRESENCE IS VERIFIED ELECTRONICALLY.
Verification of learning
THE ACQUIRED KNOWLEDGE WILL BE VERIFIED BY AN ORAL EXAM CERTIFIED ACCORDING TO THE EVALUATION 30 OUT OF 30. THE EXAM IS AN ORAL TEST WHICH CONSISTS OF AN INTERVIEW WITH QUESTIONS AND DISCUSSION ON THE CONTENTS OF THE TEACHING CLASS. THE ORAL EXAM AIMS TO VERIFY THE ACQUIRED KNOWLEDGE, ABILITY OF CONNECTIONS AMONG THE SUBJECTS AND THE USE OF AN APPROPRIATE TERMINOLOGY.
Texts
- GOODMAN & GILMAN, LE BASI FARMACOLOGICHE DELLA TERAPIA. (12A EDIZIONE). ZANICHELLI
- GOODMAN & GILMAN LE BASI FARMACOLOGICHE DELLA TERAPIA -IL MANUALE- II EDIZIONE ZANICHELLI
- ANNUNZIATO & DI RENZO, TRATTATO DI FARMACOLOGIA. IDELSON-GNOCCHI
More Information
YEAR OF COURSE: IV
SEMESTER: I
UFC: 10
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