Patents

Research Patents

Enantioselective synthesis of isoindolinones

DESCRIZIONE

The present invention relates the asymmetrical synthesis of heterocyclic compounds of pharmaceutical interest. In particular a series of enantioselective methods is described, allowing the synthesis and transformations of isoindolinones of Formula (I), into high yields and enantiomeric excesses >90%

NEED

Asymmetrical synthesis of heterocyclic compounds of pharmaceutical interest

VANTAGGI

Efficient route to biological active isoindolinones

PRINCIPALI APPLICAZIONI

Process

TRL 4

- Tecnologia convalidata in laboratorio

PAROLE CHIAVE

asymmetric synthesis, isoindolinones, active compounds

 

 

Status
Italian Patent
Deposit no. 102015902348105 - 5 May 2015
Licence no. 102015902348105 - 31 August 2017
Expiration: 5 May 2015
European Patent
16728101.3 - 18 October 2017
Licence no. 3292102 - 8 September 2021
Expiration: 3 May 2036

Convalide Nazionali:

Italia, Francia, Germania, Regno Unito.

International Patent
PCT/IB2016/052507 - 3 May 2016
Publication no. WO2016/178140 - 10 November 2016
InventorMASSA Antonio, De Capraris Paolo, Di Mola Antonio

Category

C - CHEMISTRY; METALLURGY
C07 - ORGANIC CHEMISTRY

Allegati

Patents