Research | Patents
Research Patents
Enantioselective synthesis of isoindolinones
DESCRIZIONE
The present invention relates the asymmetrical synthesis of heterocyclic compounds of pharmaceutical interest. In particular a series of enantioselective methods is described, allowing the synthesis and transformations of isoindolinones of Formula (I), into high yields and enantiomeric excesses >90%
NEED
Asymmetrical synthesis of heterocyclic compounds of pharmaceutical interest
VANTAGGI
Efficient route to biological active isoindolinones
PRINCIPALI APPLICAZIONI
Process
TRL 4
- Tecnologia convalidata in laboratorio
PAROLE CHIAVE
asymmetric synthesis, isoindolinones, active compounds
Status | Italian Patent Deposit no. 102015902348105 - 5 May 2015 Licence no. 102015902348105 - 31 August 2017 Expiration: 5 May 2015 European Patent 16728101.3 - 18 October 2017 Licence no. 3292102 - 8 September 2021 Expiration: 3 May 2036 Convalide Nazionali: Italia, Francia, Germania, Regno Unito. International Patent PCT/IB2016/052507 - 3 May 2016 Publication no. WO2016/178140 - 10 November 2016 | |
Inventor | MASSA Antonio, De Capraris Paolo, Di Mola Antonio |
Category
C - CHEMISTRY; METALLURGYC07 - ORGANIC CHEMISTRY