Pietro CAMPIGLIA | MEDICINAL CHEMISTRY I
Pietro CAMPIGLIA MEDICINAL CHEMISTRY I
cod. 0760100015
MEDICINAL CHEMISTRY I
0760100015 | |
DIPARTIMENTO DI FARMACIA | |
EQF7 | |
PHARMACY | |
2016/2017 |
OBBLIGATORIO | |
YEAR OF COURSE 3 | |
YEAR OF DIDACTIC SYSTEM 2010 | |
PRIMO SEMESTRE |
SSD | CFU | HOURS | ACTIVITY | |
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CHIM/08 | 10 | 80 | LESSONS |
Objectives | |
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KNOW THE MAIN CHEMOTHERAPEUTIC ANTIBIOTICS AND ANTICANCER DRUGS ANTIMICROBIAL, ANTIVIRAL DRUGS. OF EACH CLASS OF DRUGS, THE STUDENTS MUST KNOW THE ADME AND POSSIBLE INTERACTIONS BETWEEN DRUGS AND MEDICINES AND FOODS. |
Prerequisites | |
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ACQUISITION REQUIRED FOR THE FOLLOWING DISCIPLINES: ORGANIC CHEMISTRY AND BIOCHEMISTRY |
Contents | |
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DEFINITION OF DRUG; THE ACTIVE INGREDIENT AND PHARMACEUTICAL FORMS. DRUG DISCOVERY; THE MODERN TECHNOLOGIES IN DISCOVERY AND DRUG DEVELOPMENT. DRUGS FROM NATURAL AND SYNTHETIC ORIGIN. PHYSICO-CHEMICAL PROPERTIES OF DRUGS. PHARMACOKINETICS ; INTERACTIONS AMONG DRUGS AND AMONG DRUGS AND FOODS. BIOAVAILABILITY AND BIOEQUIVALENCE. PATENT. GENERIC DRUG. PHARMACODYNAMICS. AGONISTS, ANTAGONISTS, PARTIAL AGONISTS AND INVERSE AGONISTS. DRUG-METABOLIC INDUCTION AND INHIBITION. ENZYME INHIBITION. AIFA, EMEA, ORIGIN OF THE NAME OF THE DRUGS. INFLUENCE OF ISOMERISM ( OPTICAL , GEOMETRICAL AND CONFORMATIONAL) ON THE PHARMACOLOGICAL ACTIVITY. SPECIAL SECTION: ANTISEPTICS AND DISINFECTANTS. SULFA- DRUGS. ANTIBIOTICS . INHIBITOR VIRUS. MEDICAMENTS FOR TREATMENT OF AIDS. DRUGS USED FOR INFECTIONS WITH HEPATITIS B AND C. ANTICANCER DRUGS. ANTIFUNGALS; ANTIPROTOZOAN, PESTICIDES. EPIGENETIC DRUGS. |
Teaching Methods | |
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LECTURES, INTERACTIVE TEACHING WITH STUDENT PARTICIPATION |
Verification of learning | |
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TALKS IN ITINERE AND SELF-ASSESSMENT |
Texts | |
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ANY BOOK AS LONG AS THEY CONFORM TO THE PROGRAM |
More Information | |
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DURING THE COURSE, WILL BE CARRIED OUT IN THE FORM OF SEMINARS, TOPICS ON INNOVATIVE MEDICINES |
BETA VERSION Data source ESSE3 [Ultima Sincronizzazione: 2019-03-11]