Gianluigi LAURO | Publications
Gianluigi LAURO Publications
| 2024 | |
| Articolo in rivista | |
| A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Pag.1-24 ISSN:0022-2623. | |
| Vestuto, Vincenzo; Ciaglia, Tania; Musella, Simona; Di Sarno, Veronica; Smaldone, Gerardina; Di Matteo, Francesca; Scala, Maria Carmina; Napolitano, Valeria; Miranda, Maria Rosaria; Amodio, Giuseppina; Novi, Sara; Pepe, Giacomo; Basilicata, Manuela Giovanna; Gazzillo, Erica; Pace, Simona; Gomez-Monterrey, Isabel M.; Sala, Marina; Bifulco, Giuseppe; Tecce, Mario Felice; Campiglia, Pietro; Ostacolo, Carmine; Lauro, Gianluigi; Manfra, Michele; Bertamino, Alessia | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.4c00718 | |
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| 2024 | |
| Articolo in rivista | |
| Fatty Acid Synthase as Interacting Anticancer Target of the Terpenoid Myrianthic Acid Disclosed by MS-Based Proteomics Approaches INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. Vol. 25. Pag.5918-5938 ISSN:1422-0067. | |
| Capuano, A.; D'Urso, G.; Gazzillo, E.; Lauro, G.; Chini, M. G.; D'Auria, M. V.; Ferraro, M. G.; Iazzetti, F.; Irace, C.; Bifulco, G.; Casapullo, A. | |
| Digital Object Identifier (DOI): 10.3390/ijms25115918 Codice identificativo ISI: WOS:001245531000001 Codice identificativo SCOPUS: 2-s2.0-85195844052 | |
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| 2024 | |
| Articolo in rivista | |
| Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A MARINE DRUGS. Vol. 22. Pag.41-52 ISSN:1660-3397. | |
| Capuano, A.; D'Urso, G.; Aliberti, M.; Ruggiero, D.; Terracciano, S.; Festa, C.; Tosco, A.; Chini, M. G.; Lauro, G.; Bifulco, G.; Casapullo, A. | |
| Digital Object Identifier (DOI): 10.3390/md22010041 Codice identificativo ISI: WOS:001150851600001 Codice identificativo SCOPUS: 2-s2.0-85183127360 | |
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| 2024 | |
| Articolo in rivista | |
| NMR Metabolomics and Chemometrics of Commercial Varieties of Phaseolus vulgaris L. Seeds from Italy and In Vitro Antioxidant and Antifungal Activity PLANTS. Vol. 13. Pag.227-253 ISSN:2223-7747. | |
| Samukha, V.; Fantasma, F.; D'Urso, G.; Caprari, C.; De Felice, V.; Saviano, G.; Lauro, G.; Casapullo, A.; Chini, M. G.; Bifulco, G.; Iorizzi, M. | |
| Digital Object Identifier (DOI): 10.3390/plants13020227 Codice identificativo ISI: WOS:001153025200001 Codice identificativo SCOPUS: 2-s2.0-85183117074 | |
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| 2024 | |
| Articolo in rivista | |
| Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterization EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 266. Pag.1-23 ISSN:0223-5234. | |
| Ciaglia, Tania; Vestuto, Vincenzo; Di Sarno, Veronica; Musella, Simona; Smaldone, Gerardina; Di Matteo, Francesca; Napolitano, Valeria; Miranda, Maria Rosaria; Pepe, Giacomo; Basilicata, Manuela Giovanna; Novi, Sara; Capolupo, Ilaria; Bifulco, Giuseppe; Campiglia, Pietro; Gomez-Monterrey, Isabel; Snoeck, Robert; Andrei, Graciela; Manfra, Michele; Ostacolo, Carmine; Lauro, Gianluigi; Bertamino, Alessia | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2024.116128 Codice identificativo ISI: WOS:001166699700001 Codice identificativo SCOPUS: 2-s2.0-85182642774 | |
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| 2023 | |
| Articolo in rivista | |
| 2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 93. Pag.117444-117467 ISSN:1464-3391. | |
| De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2023.117444 Codice identificativo ISI: WOS:001064638100001 Codice identificativo SCOPUS: 2-s2.0-85168487978 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 247. Pag.115018-115018 ISSN:0223-5234. | |
| Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.115018 Codice identificativo ISI: WOS:000913013400001 Codice identificativo SCOPUS: 2-s2.0-85144788456 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors ACS MEDICINAL CHEMISTRY LETTERS. Vol. 14(1). Pag.26-34 ISSN:1948-5875. | |
| Potenza, Marianna; Giordano, Assunta; Chini, Maria G; Saviano, Anella; Kretzer, Christian; Raucci, Federica; Russo, Marina; Lauro, Gianluigi; Terracciano, Stefania; Bruno, Ines; Iorizzi, Maria; Hofstetter, Robert K; Pace, Simona; Maione, Francesco; Werz, Oliver; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1021/acsmedchemlett.2c00343 Codice identificativo SCOPUS: 2-s2.0-85143868000 | |
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263998Target identification by structure-based computational approaches: Recent advances and perspectives
| 2023 | |
| Articolo in rivista | |
| Target identification by structure-based computational approaches: Recent advances and perspectives BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. Vol. 83. Pag.129171-129171 ISSN:1464-3405. | |
| De Vita, Simona; Chini, Maria Giovanna; Bifulco, Giuseppe; Lauro, Gianluigi | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2023.129171 Codice identificativo ISI: WOS:000944919600001 Codice identificativo SCOPUS: 2-s2.0-85147876194 | |
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| 2023 | |
| Articolo in rivista | |
| Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 BIOORGANIC CHEMISTRY. Vol. 139. Pag.106677-106677 ISSN:0045-2068. | |
| Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2023.106677 Codice identificativo ISI: WOS:001031583200001 Codice identificativo SCOPUS: 2-s2.0-85163217544 | |
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| 2022 | |
| Articolo in rivista | |
| Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation MOLECULES. Vol. 27. Pag.3866-3866 ISSN:1420-3049. | |
| Gazzillo, Erica; Terracciano, Stefania; Ruggiero, Dafne; Potenza, Marianna; Chini, Maria Giovanna; Lauro, Gianluigi; Fischer, Katrin; Hofstetter, Robert Klaus; Giordano, Assunta; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.3390/molecules27123866 Codice identificativo ISI: WOS:000819099100001 Codice identificativo SCOPUS: 2-s2.0-85132592035 | |
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| 2022 | |
| Articolo in rivista | |
| New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 238. Pag.1-19 ISSN:0223-5234. | |
| Di Sarno, Veronica; Giovannelli, Pia; Medina-Peris, Alicia; Ciaglia, Tania; Di Donato, Marzia; Musella, Simona; Lauro, Gianluigi; Vestuto, Vincenzo; Smaldone, Gerardina; Di Matteo, Francesca; Bifulco, Giuseppe; Castoria, Gabriella; Migliaccio, Antimo; Fernandez-Carvajal, Asia; Campiglia, Pietro; Gomez-Monterrey, Isabel; Ostacolo, Carmine; Bertamino, Alessia | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.114435 Codice identificativo ISI: WOS:000806807500007 Codice identificativo SCOPUS: 2-s2.0-85130565120 | |
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| 2022 | |
| Articolo in rivista | |
| In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway BIOMOLECULES. Vol. 12. Pag.99-99 ISSN:2218-273X. | |
| Saviano, A.; De Vita, S.; Chini, M. G.; Marigliano, N.; Lauro, G.; Casillo, G. M.; Raucci, F.; Iorizzi, M.; Hofstetter, R. K.; Fischer, K.; Koeberle, A.; Werz, O.; Maione, F.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.3390/biom12010099 Codice identificativo ISI: WOS:000747842600001 Codice identificativo SCOPUS: 2-s2.0-85122248050 | |
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| 2022 | |
| Articolo in rivista | |
| Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein MOLECULES. Vol. 27. Pag.665-665 ISSN:1420-3049. | |
| Ruggiero, D.; Terracciano, S.; Lauro, G.; Pecoraro, M.; Franceschelli, S.; Bifulco, G.; Bruno, I. | |
| Digital Object Identifier (DOI): 10.3390/molecules27030665 Codice identificativo ISI: WOS:000814371500001 Codice identificativo SCOPUS: 2-s2.0-85123075067 | |
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| 2022 | |
| Articolo in rivista | |
| Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders BIOORGANIC CHEMISTRY. Vol. 118. Pag.105480-105480 ISSN:0045-2068. | |
| Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G. | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2021.105480 Codice identificativo ISI: WOS:000821662200006 Codice identificativo SCOPUS: 2-s2.0-85119580843 | |
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| 2022 | |
| Articolo in rivista | |
| Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies FRONTIERS IN PLANT SCIENCE. Vol. 13. Pag.805660-805660 ISSN:1664-462X. | |
| Masullo, M.; Lauro, G.; Cerulli, A.; Bifulco, G.; Piacente, S. | |
| Digital Object Identifier (DOI): 10.3389/fpls.2022.805660 Codice identificativo ISI: WOS:000761603900001 Codice identificativo SCOPUS: 2-s2.0-85125374215 | |
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| 2022 | |
| Articolo in rivista | |
| Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches PLANTS. Vol. 11. Pag.1671-1691 ISSN:2223-7747. | |
| De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria | |
| Versione online | |
| Digital Object Identifier (DOI): 10.3390/plants11131671 Codice identificativo ISI: WOS:000825696400001 Codice identificativo SCOPUS: 2-s2.0-85132770397 | |
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| 2022 | |
| Articolo in rivista | |
| 6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 2022. Pag.e202200868-e202200868 ISSN:1434-193X. | |
| Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G | |
| Digital Object Identifier (DOI): 10.1002/ejoc.202200868 Codice identificativo ISI: WOS:000854579600001 Codice identificativo SCOPUS: 2-s2.0-85138949165 | |
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| 2022 | |
| Articolo in rivista | |
| Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies PHYTOCHEMISTRY. Vol. 205. Pag.113471-113471 ISSN:0031-9422. | |
| Kılınc, Hilal; Masullo, Milena; Lauro, Gianluigi; D'Urso, Gilda; Alankus, Ozgen; Bifulco, Giuseppe; Piacente, Sonia | |
| Digital Object Identifier (DOI): 10.1016/j.phytochem.2022.113471 Codice identificativo ISI: WOS:000880850100004 Codice identificativo SCOPUS: 2-s2.0-85140583901 | |
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| 2022 | |
| Articolo in rivista | |
| Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor MOLECULAR INFORMATICS. Pag.2200140-2200140 ISSN:1868-1743. | |
| Di Micco, Simone; Lauro, Gianluigi; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1002/minf.202200140 Codice identificativo ISI: WOS:000861445400001 Codice identificativo SCOPUS: 2-s2.0-85138952002 | |
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| 2022 | |
| Articolo in rivista | |
| Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS. Vol. 5. Pag.100046-100046 ISSN:2772-4174. | |
| Colarusso, Ester; Potenza, Marianna; Lauro, Gianluigi; Giovanna Chini, Maria; Sepe, Valentina; Zampella, Angela; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.ejmcr.2022.100046 Codice identificativo ISI: WOS:001108747600004 Codice identificativo SCOPUS: 2-s2.0-85132583529 | |
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| 2021 | |
| Articolo in rivista | |
| The plant diterpene epoxysiderol targets Hsp70 in cancer cells, affecting its ATPase activity and reducing its translocation to plasma membrane INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES. Vol. 189. Pag.262-270 ISSN:0141-8130. | |
| Fiengo, L.; Lauro, G.; Bellone, M. L.; Bifulco, G.; Dal Piaz, F.; De Tommasi, N. | |
| Digital Object Identifier (DOI): 10.1016/j.ijbiomac.2021.08.138 Codice identificativo ISI: WOS:000702836800001 Codice identificativo SCOPUS: 2-s2.0-85113361329 | |
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| 2021 | |
| Articolo in rivista | |
| Identification of a dual acting SARS-CoV-2 proteases inhibitor through in silico design and step-by-step biological characterization EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 226. Pag.113863-113863 ISSN:0223-5234. | |
| Di Sarno, V.; Lauro, G.; Musella, S.; Ciaglia, T.; Vestuto, V.; Sala, M.; Scala, M. C.; Smaldone, G.; Di Matteo, F.; Novi, S.; Tecce, M. F.; Moltedo, O.; Bifulco, G.; Campiglia, P.; Gomez-Monterrey, I. M.; Snoeck, R.; Andrei, G.; Ostacolo, C.; Bertamino, A. | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2021.113863 Codice identificativo ISI: WOS:000703119000042 Codice identificativo SCOPUS: 2-s2.0-85115784362 | |
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| 2021 | |
| Articolo in rivista | |
| Giffonins, Antioxidant Diarylheptanoids from Corylus avellana, and Their Ability to Prevent Oxidative Changes in Human Plasma Proteins JOURNAL OF NATURAL PRODUCTS. Vol. 84. Pag.646-653 ISSN:0163-3864. | |
| Masullo, M.; Lauro, G.; Cerulli, A.; Kontek, B.; Olas, B.; Bifulco, G.; Piacente, S.; Pizza, C. | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.0c01251 Codice identificativo ISI: WOS:000635469000010 Codice identificativo SCOPUS: 2-s2.0-85102048391 | |
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| 2021 | |
| Articolo in rivista | |
| Biological Profile of Two Gentiana lutea L. Metabolites UsingComputational Approaches and In Vitro Tests BIOMOLECULES. Vol. 11. Pag.1-20 ISSN:2218-273X. | |
| DE VITA, Simona; Giovanna Chini, Maria; Saviano, Gabriella; Finamore, Claudia; Festa, Carmen; Lauro, Gianluigi; De Marino, Simona; Russo, Roberto; Avagliano, Carmen; Casapullo, Agostino; Calignano, Antonio; Bifulco, Giuseppe; Iorizzi, Maria | |
| Digital Object Identifier (DOI): 10.3390/biom11101490 Codice identificativo ISI: WOS:000715414700001 Codice identificativo SCOPUS: 2-s2.0-85116782513 | |
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| 2021 | |
| Articolo in rivista | |
| Addressing the Target Identification and Accelerating the Repositioning of Anti-Inflammatory/Anti-Cancer Organic Compounds by Computational Approaches EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 2021. Pag.2966-2981 ISSN:1434-193X. | |
| Chini, M. G.; Lauro, G.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1002/ejoc.202100245 Codice identificativo ISI: WOS:000674294200007 Codice identificativo SCOPUS: 2-s2.0-85110563481 | |
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| 2021 | |
| Articolo in rivista | |
| Insights into the ligand binding to bromodomain‐containing protein 9 (BRD9): A guide to the selection of potential binders by computational methods MOLECULES. Vol. 26. Pag.7192-7192 ISSN:1420-3049. | |
| De Vita, S.; Chini, M. G.; Bifulco, G.; Lauro, G. | |
| Digital Object Identifier (DOI): 10.3390/molecules26237192 Codice identificativo ISI: WOS:000734504900001 Codice identificativo SCOPUS: 2-s2.0-85120604348 | |
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| 2021 | |
| Articolo in rivista | |
| Inverse Virtual Screening for the rapid re-evaluation of the presumed biological safe profile of natural products. The case of steviol from Stevia rebaudiana glycosides on farnesoid X receptor (FXR) BIOORGANIC CHEMISTRY. Vol. 111. Pag.104897-104897 ISSN:0045-2068. | |
| Potenza, M.; Cavalluzzi, M. M.; Milani, G.; Lauro, G.; Carino, A.; Roselli, R.; Fiorucci, S.; Zampella, A.; Pierri, C. L.; Lentini, G.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2021.104897 Codice identificativo ISI: WOS:000656969600004 Codice identificativo SCOPUS: 2-s2.0-85104596103 | |
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| 2020 | |
| Articolo in rivista | |
| A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors CHEMMEDCHEM. Vol. 15. Pag.481-489 ISSN:1860-7179. | |
| Lauro, G.; Terracciano, S.; Cantone, V.; Ruggiero, D.; Fischer, K.; Pace, S.; Werz, O.; Bruno, I.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201900694 Codice identificativo ISI: WOS:000513689000001 Codice identificativo SCOPUS: 2-s2.0-85079711216 | |
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| 2020 | |
| Articolo in rivista | |
| Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their in Vitro Characterization and in Vivo Analgesic Activities JOURNAL OF MEDICINAL CHEMISTRY. Vol. 63. Pag.9672-9694 ISSN:0022-2623. | |
| Bertamino, A.; Ostacolo, C.; Medina, A.; Di Sarno, V.; Lauro, G.; Ciaglia, T.; Vestuto, V.; Pepe, G.; Basilicata, M. G.; Musella, S.; Smaldone, G.; Cristiano, C.; Gonzalez-Rodriguez, S.; Fernandez-Carvajal, A.; Bifulco, G.; Campiglia, P.; Gomez-Monterrey, I.; Russo, R. | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.0c00816 Codice identificativo ISI: WOS:000571493400046 Codice identificativo SCOPUS: 2-s2.0-85090870415 | |
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| 2020 | |
| Articolo in rivista | |
| Discovery of noscapine derivatives as potential β-tubulin inhibitors BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 30. Pag.127489-127489 ISSN:0960-894X. | |
| Nemati, F.; Salehi, P.; Bararjanian, M.; Hadian, N.; Mohebbi, M.; Lauro, G.; Ruggiero, D.; Terracciano, S.; Bifulco, G.; Bruno, I. | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2020.127489 Codice identificativo ISI: WOS:000576786000002 Codice identificativo SCOPUS: 2-s2.0-85089348593 | |
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| 2020 | |
| Articolo in rivista | |
| Elucidating the Relative and Absolute Configuration of Organic Compounds by Quantum Mechanical Approaches EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Pag.3929-3941 ISSN:1434-193X. | |
| Lauro, G.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1002/ejoc.201901878 Codice identificativo ISI: WOS:000548287400001 Codice identificativo SCOPUS: 2-s2.0-85081953588 | |
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| 2020 | |
| Articolo in rivista | |
| Accelerating the repurposing of FDA-approved drugs against coronavirus disease-19 (COVID-19) RSC ADVANCES. Vol. 10. Pag.40867-40875 ISSN:2046-2069. | |
| De Vita, S.; Chini, M. G.; Lauro, G.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1039/d0ra09010g Codice identificativo ISI: WOS:000588975500024 Codice identificativo SCOPUS: 2-s2.0-85096334679 | |
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| 2020 | |
| Articolo in rivista | |
| Discovery of a Secalonic Acid Derivative from Aspergillus aculeatus, an Endophyte of Rosa damascena Mill., Triggers Apoptosis in MDA-MB-231 Triple Negative Breast Cancer Cells ACS OMEGA. Vol. 5. Pag.24296-24310 ISSN:2470-1343. | |
| Farooq, S.; Qayum, A.; Nalli, Y.; Lauro, G.; Chini, M. G.; Bifulco, G.; Chaubey, A.; Singh, S. K.; Riyaz-Ul-Hassan, S.; Ali, A. | |
| Digital Object Identifier (DOI): 10.1021/acsomega.0c02505 Codice identificativo ISI: WOS:000576748800017 Codice identificativo SCOPUS: 2-s2.0-85092585192 | |
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| 2020 | |
| Articolo in rivista | |
| DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data JOURNAL OF ORGANIC CHEMISTRY. Vol. 85. Pag.3297-3306 ISSN:0022-3263. | |
| Lauro, G.; Das, P.; Riccio, R.; Reddy, D. S.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1021/acs.joc.9b03129 Codice identificativo ISI: WOS:000518875700038 Codice identificativo SCOPUS: 2-s2.0-85081944844 | |
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| 2019 | |
| Articolo in rivista | |
| Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods JOURNAL OF CHEMICAL INFORMATION AND MODELING. Pag.4678-4690 ISSN:1549-9596. | |
| De Vita, S.; Lauro, G.; Ruggiero, D.; Terracciano, S.; Riccio, R.; Bifulco, G. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jcim.9b00428 Codice identificativo ISI: WOS:000500038700018 Codice identificativo SCOPUS: 2-s2.0-85074665461 | |
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| 2019 | |
| Articolo in rivista | |
| Immunomodulatory Biscembranoids and Assignment of Their Relative and Absolute Configurations: Data Set Modulation in the Density Functional Theory/Nuclear Magnetic Resonance Approach JOURNAL OF NATURAL PRODUCTS. Vol. 82. Pag.1264-1273 ISSN:0163-3864. | |
| Sun, P.; Cai, F. -Y.; Lauro, G.; Tang, H.; Su, L.; Wang, H. -L.; Li, H. H.; Mandi, A.; Kurtan, T.; Riccio, R.; Bifulco, G.; Zhang, W. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.8b01037 Codice identificativo ISI: WOS:000469410200025 Codice identificativo SCOPUS: 2-s2.0-85066113210 | |
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| 2019 | |
| Articolo in rivista | |
| Isolation, Synthesis And Structure Determination Of Cannabidiol Derivatives And Their Cytotoxic Activities NATURAL PRODUCT RESEARCH. Pag.1-10 ISSN:1478-6419. | |
| Nalli, Y.; Jan, S.; Lauro, G.; Ur Rasool, J.; Lone, W. I.; Sarkar, A. R.; Banday, J.; Bifulco, G.; Laatsch, H.; Syed, S. H.; Ali, A. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/14786419.2019.1638381 Codice identificativo ISI: WOS:000474843200001 Codice identificativo SCOPUS: 2-s2.0-85068694978 | |
| Show it in Product Database (IRIS) |
| 2019 | |
| Articolo in rivista | |
| Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 167. Pag.61-75 ISSN:0223-5234. | |
| Ostacolo, Carmine; Di Sarno, Veronica; Lauro, Gianluigi; Pepe, Giacomo; Musella, Simona; Ciaglia, Tania; Vestuto, Vincenzo; Autore, Giuseppina; Bifulco, Giuseppe; Marzocco, Stefania; Campiglia, Pietro; Gomez-Monterrey, Isabel M; Bertamino, Alessia | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2019.01.066 Codice identificativo ISI: WOS:000461728400005 Codice identificativo SCOPUS: 2-s2.0-85061236063 | |
| Show it in Product Database (IRIS) |
| 2018 | |
| Articolo in rivista | |
| Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics CHEMICAL COMMUNICATIONS. Vol. 54. Pag.7613-7616 ISSN:1359-7345. | |
| Terracciano, Stefania; Lauro, Gianluigi; Russo, Alessandra; Vaccaro, Maria Carmela; Vassallo, Antonio; De Marco, Margot; Ranieri, Bianca; Rosati, Alessandra; Turco, Maria Caterina; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c8cc03399d Codice identificativo ISI: WOS:000442118800009 Codice identificativo SCOPUS: 2-s2.0-85049623511 | |
| Show it in Product Database (IRIS) |
| 2018 | |
| Articolo in rivista | |
| Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells JOURNAL OF NATURAL PRODUCTS. Vol. 81. Pag.1786-1794 ISSN:0163-3864. | |
| Ayoub, Khalfaoui; Chini, MARIA GIOVANNA; Mohamed, Bouheroum; Soumia, Belaabed; Lauro, Gianluigi; Terracciano, Stefania; Vaccaro, Mariacarmela; Bruno, Ines; Samir, Benayache; Ines, Mancini; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.8b00234 Codice identificativo ISI: WOS:000443103700011 Codice identificativo SCOPUS: 2-s2.0-85052588349 | |
| Show it in Product Database (IRIS) |
| 2018 | |
| Articolo in rivista | |
| Discovery of 3-hydroxy-3-pyrrolin-2-one-based mPGES-1 inhibitors using a multi-step virtual screening protocol MEDCHEMCOMM. Vol. 9. Pag.2028-2036 ISSN:2040-2503. | |
| Lauro, G.; Cantone, V.; Potenza, M.; Fischer, K.; Koeberle, A.; Werz, O.; Riccio, R.; Bifulco, G. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c8md00497h Codice identificativo ISI: WOS:000453225200005 Codice identificativo SCOPUS: 2-s2.0-85058623321 | |
| Show it in Product Database (IRIS) |
| 2018 | |
| Articolo in rivista | |
| Total synthesis of the potent anti-inflammatory natural product solomonamide A along with structural revision and biological activity evaluation ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 16. Pag.9138-9142 ISSN:1477-0520. | |
| Jachak, G. R.; Athawale, P. R.; Agarwal, H.; Barthwal, M. K.; Lauro, G.; Bifulco, G.; Srinivasa Reddy, D. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c8ob02713g Codice identificativo ISI: WOS:000452321100006 Codice identificativo SCOPUS: 2-s2.0-85058177071 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Ring-Fused Cyclic Aminals from Tetrahydro-β-carboline-Based Dipeptide Compounds JOURNAL OF ORGANIC CHEMISTRY. Vol. 82. Pag.12014-12027 ISSN:0022-3263. | |
| Bertamino, Alessia; Lauro, Gianluigi; Ostacolo, Carmine; DI SARNO, Veronica; Musella, Simona; Ciaglia, Tania; Campiglia, Pietro; Bifulco, Giuseppe; Gomez-Monterrey, Isabel M. | |
| Digital Object Identifier (DOI): 10.1021/acs.joc.7b01656 Codice identificativo ISI: WOS:000417342300005 Codice identificativo SCOPUS: 2-s2.0-85036577381 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Tulongicin, an Antibacterial Tri-Indole Alkaloid from a Deep-Water Topsentia sp. Sponge JOURNAL OF NATURAL PRODUCTS. Vol. 80. Pag.2556-2560 ISSN:0163-3864. | |
| Liu, Hong-Bing; Lauro, Gianluigi; O'Connor, Robert D; Lohith, Katheryn; Kelly, Michelle; Colin, Patrick; Bifulco, Giuseppe; Bewley, Carole A. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.7b00452 Codice identificativo ISI: WOS:000411848300024 Codice identificativo SCOPUS: 2-s2.0-85029739350 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Cyclic Diarylheptanoids from Corylus avellana Green Leafy Covers: Determination of Their Absolute Configurations and Evaluation of Their Antioxidant and Antimicrobial Activities JOURNAL OF NATURAL PRODUCTS. Vol. 80. Pag.1703-1713 ISSN:0163-3864. | |
| Cerulli, Antonietta; Lauro, Gianluigi; Masullo, Milena; Cantone, Vincenza; Olas, Beata; Kontek, Bogdan; Nazzaro, Filomena; Bifulco, Giuseppe; Piacente, Sonia | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.6b00703 Codice identificativo ISI: WOS:000404322100001 Codice identificativo SCOPUS: 2-s2.0-85021162727 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Svetamycins A-G, Unusual Piperazic Acid-Containing Peptides from Streptomyces sp JOURNAL OF ORGANIC CHEMISTRY. Vol. 82. Pag.6032-6043 ISSN:0022-3263. | |
| Dardic, Denis; Lauro, Gianluigi; Bifulco, Giuseppe; Laboudie, Patricia; Sakhaii, Peyman; Bauer, Armin; Vilcinskas, Andreas; Hammann, Peter E; Plaza, Alberto | |
| Digital Object Identifier (DOI): 10.1021/acs.joc.7b00228 Codice identificativo ISI: WOS:000403854500004 Codice identificativo SCOPUS: 2-s2.0-85020879010 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Chemistry and Selective Tumor Cell Growth Inhibitory Activity of Polyketides from the South China Sea Sponge Plakortis sp MARINE DRUGS. Vol. 15 (5). Pag.129-129 ISSN:1660-3397. | |
| Li, Jiao; Li, Cui; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Li, Tie Jun; Tang, Hua; Zhuang, Chun Lin; Ma, Hao; Sun, Peng; Zhang, Wen | |
| Versione online | |
| Digital Object Identifier (DOI): 10.3390/md15050129 Codice identificativo ISI: WOS:000404235100005 Codice identificativo SCOPUS: 2-s2.0-85019550310 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer SCIENTIFIC REPORTS. Vol. 7. Pag.1-14 ISSN:2045-2322. | |
| Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/s41598-017-11688-x Codice identificativo ISI: WOS:000410859400010 Codice identificativo SCOPUS: 2-s2.0-85029517928 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 125. Pag.278-287 ISSN:0223-5234. | |
| Lauro, Gianluigi; Manfra, Michele; Pedatella, Silvana; Fischer, Katrin; Cantone, Vincenza; Terracciano, Stefania; Bertamino, Alessia; Ostacolo, Carmine; Gomez Monterrey, Isabel; De Nisco, Mauro; Riccio, Raffaele; Novellino, Ettore; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2016.09.042 Codice identificativo ISI: WOS:000390496600020 Codice identificativo SCOPUS: 2-s2.0-84988579046 | |
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101733Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride
| 2016 | |
| Articolo in rivista | |
| Bissubvilides A and B, Cembrane-capnosane heterodimers from the soft coral sarcophyton subviride JOURNAL OF NATURAL PRODUCTS. Vol. 79. Pag.2552-2558 ISSN:0163-3864. | |
| Sun, Peng; Yu, Qing; Li, Jiao; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Kurtán, Tibor; Mándi, Attila; Tang, Hua; Li, Tie Jun; Zhuang, Chun Lin; Gerwick, William H.; Zhang, Wen | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.6b00453 Codice identificativo ISI: WOS:000386745300017 Codice identificativo SCOPUS: 2-s2.0-84994031930 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme CHEMMEDCHEM. Vol. 11. Pag.612-619 ISSN:1860-7179. | |
| Lauro, Gianluigi; Tortorella, Paolo; Bertamino, Alessia; Ostacolo, Carmine; Koeberle, Andreas; Fischer, Katrin; Bruno, Ines; Terracciano, Stefania; Gomez Monterrey, Isabel Maria; Tauro, Marilena; Loiodice, Fulvio; Novellino, Ettore; Riccio, Raffaele; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201500598 Codice identificativo ISI: WOS:000372990700007 Codice identificativo SCOPUS: 2-s2.0-84959387319 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| Anti-inflammatory trends of new benzimidazole derivatives FUTURE MEDICINAL CHEMISTRY. Vol. 8. Pag.1953-1967 ISSN:1756-8919. | |
| Bukhari, Syed Nasir Abbas; Lauro, Gianluigi; Jantan, Ibrahim; Chee, Chin Fei; Amjad, Muhammad Wahab; Bifulco, Giuseppe; Sher, Hassan; Abdullah, Iskandar; Rahman, Noorsaadah Abd | |
| Versione online | |
| Digital Object Identifier (DOI): 10.4155/fmc-2016-0062 Codice identificativo ISI: WOS:000386339000007 Codice identificativo SCOPUS: 2-s2.0-84989851874 | |
| Show it in Product Database (IRIS) |
68732Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors
| 2015 | |
| Articolo in rivista | |
| Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors ACS MEDICINAL CHEMISTRY LETTERS. Vol. 6. Pag.187-91-191 ISSN:1948-5875. | |
| Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/ml500433j Codice identificativo ISI: WOS:000349652000015 Codice identificativo SCOPUS: 2-s2.0-84922936636 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Giffonins J-P, Highly Hydroxylated Cyclized Diarylheptanoids from the Leaves of Corylus avellana Cultivar "Tonda di Giffoni" JOURNAL OF NATURAL PRODUCTS. Vol. 78 (12). Pag.2975-2982 ISSN:0163-3864. | |
| Masullo, Milena; Cantone, Vincenza; Cerulli, Antonietta; Lauro, Gianluigi; Messano, Francesco; Russo, Gian Luigi; Pizza, Cosimo; Bifulco, Giuseppe; Piacente, Sonia | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.5b00695 Codice identificativo ISI: WOS:000367562600014 Codice identificativo SCOPUS: 2-s2.0-84953308429 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain JOURNAL OF MEDICINAL CHEMISTRY. Vol. 58. Pag.2718-2736 ISSN:0022-2623. | |
| Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm501893k Codice identificativo ISI: WOS:000351971800009 Codice identificativo SCOPUS: 2-s2.0-84925938831 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs. In: Atti del Convegno Pag.196-196 | |
| XXXVI Convegno Nazionale della Divisione di Chimica Organica della Società Chimica Italiana Bologna 13-17 settembre 2015 | |
| Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs. In: Atti del Congresso Federico Bella and Domenico Spinelli Pag.126-126 | |
| SIGMA-ALDRICH Young Chemists Symposium Rimini dal 27 al 29 ottobre 2015 | |
| Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| Pharmacological evaluation and docking studies of α,β-unsaturated carbonyl based synthetic compounds as inhibitors of secretory phospholipase A2, cyclooxygenases, lipoxygenase and proinflammatory cytokines BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 22. Pag.4151-4161 ISSN:0968-0896. | |
| Syed Nasir Abbas, Bukhari; Lauro, Gianluigi; Ibrahim, Jantan; Bifulco, Giuseppe; Muhammad Wahab, Amjad | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2014.05.052 Codice identificativo ISI: WOS:000339859700039 Codice identificativo SCOPUS: 2-s2.0-84905113460 | |
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| 2014 | |
| Articolo in rivista | |
| Reranking docking poses using molecular simulations and approximate free energy methods JOURNAL OF CHEMICAL INFORMATION AND MODELING. Vol. 54. Pag.2185-2189 ISSN:1549-9596. | |
| Lauro, G.; Ferruz, N.; Fulle, S.; Harvey, M. J.; Finn, P. W.; De Fabritiis, G. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/ci500309a Codice identificativo ISI: WOS:000340861900001 Codice identificativo SCOPUS: 2-s2.0-84906545263 | |
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60470New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei
| 2014 | |
| Articolo in rivista | |
| New Steroids with a Rearranged Skeleton as (h)P300 Inhibitors from the SpongeTheonella swinhoei ORGANIC LETTERS. Vol. 16. Pag.2224-2227 ISSN:1523-7060. | |
| Jun, Gong; Peng, Sun; Nan, Jiang; Riccio, Raffaele; Lauro, Gianluigi; Bifulco, Giuseppe; Tie Jun, Li; William H., Gerwick; Wen, Zhang | |
| Digital Object Identifier (DOI): 10.1021/ol5007345 Codice identificativo ISI: WOS:000334823600039 Codice identificativo SCOPUS: 2-s2.0-84898931634 | |
| Show it in Product Database (IRIS) |
61925Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum
| 2014 | |
| Articolo in rivista | |
| Hyalachelins A–C, Unusual Siderophores Isolated from the Terrestrial MyxobacteriumHyalangium minutum ORGANIC LETTERS. Vol. 16. Pag.4130-4133 ISSN:1523-7060. | |
| Suvd, Nadmid; Alberto, Plaza; Lauro, Gianluigi; Ronald, Garcia; Bifulco, Giuseppe; Rolf, Müller | |
| Digital Object Identifier (DOI): 10.1021/ol501826a Codice identificativo ISI: WOS:000340517200019 Codice identificativo SCOPUS: 2-s2.0-84906213082 | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 80. Pag.407-415 ISSN:0223-5234. | |
| Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2014.04.061 Codice identificativo ISI: WOS:000337985400037 Codice identificativo SCOPUS: 2-s2.0-84899871048 | |
| Show it in Product Database (IRIS) |
61926Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase
| 2014 | |
| Articolo in rivista | |
| Structural Evidence ofN6-Isopentenyladenosine As a New Ligand of Farnesyl Pyrophosphate Synthase JOURNAL OF MEDICINAL CHEMISTRY. Vol. 57. Pag.7798-7803 ISSN:0022-2623. | |
| Scrima, Mario; Lauro, Gianluigi; Grimaldi, Manuela; Sara Di, Marino; Tosco, Alessandra; Picardi, Paola; Gazzerro, Patrizia; Riccio, Raffaele; Ettore, Novellino; Bifulco, Maurizio; Bifulco, Giuseppe; D'Ursi, Anna Maria | |
| Digital Object Identifier (DOI): 10.1021/jm500869x Codice identificativo ISI: WOS:000342396200023 Codice identificativo SCOPUS: 2-s2.0-84907457173 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Articolo in rivista | |
| Chemical proteomics reveals HSP70 1A as a target for the anticancer diterpene oridonin in Jurkat cells JOURNAL OF PROTEOMICS. Vol. 82. Pag.14-26 ISSN:1874-3919. | |
| DAL PIAZ, Fabrizio; Cotugno, Roberta; Lepore, Laura; Vassallo, Antonio; Malafronte, Nicola; Lauro, Gianluigi; Bifulco, Giuseppe; Belisario, MARIA ANTONIETTA; DE TOMMASI, Nunziatina | |
| Digital Object Identifier (DOI): 10.1016/j.jprot.2013.01.030 Codice identificativo ISI: WOS:000319643300002 Codice identificativo SCOPUS: 2-s2.0-84875598212 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Articolo in rivista | |
| Oxygenated polyketides from plakinastrella mamillaris as a new chemotype of PXR agonists MARINE DRUGS. Vol. 11. Pag.2314-2327 ISSN:1660-3397. | |
| Festa, Carmen; D'Amore, Claudio; Renga, Barbara; Lauro, Gianluigi; De Marino, Simona; D'Auria, Maria Valeria; Bifulco, Giuseppe; Zampella, Angela; Fiorucci, Stefano | |
| Versione online | |
| Digital Object Identifier (DOI): 10.3390/md11072314 Codice identificativo ISI: WOS:000328621500005 Codice identificativo SCOPUS: 2-s2.0-84880909903 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Inverse Virtual Screening allows the discovery of the biological activity of natural compounds BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 20. Pag.3596-3602 ISSN:0968-0896. | |
| Lauro, Gianluigi; Masullo, Milena; Piacente, Sonia; Riccio, Raffaele; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2012.03.072 Codice identificativo ISI: WOS:000303935800021 Codice identificativo SCOPUS: 2-s2.0-84861189353 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.8303-8317 ISSN:0022-2623. | |
| Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela | |
| Digital Object Identifier (DOI): 10.1021/jm300911g Codice identificativo ISI: WOS:000309643500010 Codice identificativo SCOPUS: 2-s2.0-84867352661 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 10. Pag.6350-6362 ISSN:1477-0520. | |
| Valentina, Sepe; Raffaella, Ummarino; Maria Valeria, Dauria; Lauro, Gianluigi; Bifulco, Giuseppe; Claudio, D'Amore; Barbara, Renga; Stefano, Fiorucci; Angela, Zampella | |
| Digital Object Identifier (DOI): 10.1039/c2ob25800e Codice identificativo ISI: WOS:000306480100014 Codice identificativo SCOPUS: 2-s2.0-84863908159 | |
| Show it in Product Database (IRIS) |
43470Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor
| 2012 | |
| Articolo in rivista | |
| Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.735-742 ISSN:0022-2623. | |
| Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A. | |
| Digital Object Identifier (DOI): 10.1021/jm201238p Codice identificativo ISI: WOS:000299453300017 Codice identificativo SCOPUS: 2-s2.0-84856367249 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds JOURNAL OF NATURAL PRODUCTS. Vol. 74 (6). Pag.1401-1407 ISSN:0163-3864. | |
| Lauro, Gianluigi; A., Romano; Riccio, Raffaele; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1021/np100935s Codice identificativo ISI: WOS:000291920600008 Codice identificativo SCOPUS: 2-s2.0-79959699687 | |
| Show it in Product Database (IRIS) |
