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Publications

Gianluigi LAURO Publications


2022
Articolo in rivista
Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation
MOLECULES. Vol. 27. Pag.3866-3866
ISSN:1420-3049.
Gazzillo, Erica; Terracciano, Stefania; Ruggiero, Dafne; Potenza, Marianna; Chini, Maria Giovanna; Lauro, Gianluigi; Fischer, Katrin; Hofstetter, Robert Klaus; Giordano, Assunta; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe
Digital Object Identifier (DOI): 10.3390/molecules27123866
Codice identificativo ISI: WOS:000819099100001
Codice identificativo SCOPUS: 2-s2.0-85132592035
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2022
Articolo in rivista
New TRPM8 blockers exert anticancer activity over castration-resistant prostate cancer models
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 238. Pag.1-19
ISSN:0223-5234.
Di Sarno, Veronica; Giovannelli, Pia; Medina-Peris, Alicia; Ciaglia, Tania; Di Donato, Marzia; Musella, Simona; Lauro, Gianluigi; Vestuto, Vincenzo; Smaldone, Gerardina; Di Matteo, Francesca; Bifulco, Giuseppe; Castoria, Gabriella; Migliaccio, Antimo; Fernandez-Carvajal, Asia; Campiglia, Pietro; Gomez-Monterrey, Isabel; Ostacolo, Carmine; Bertamino, Alessia
Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.114435
Codice identificativo ISI: WOS:000806807500007
Codice identificativo SCOPUS: 2-s2.0-85130565120
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2022
Articolo in rivista
Thiazolidin-4-one-based compounds interfere with the eicosanoid biosynthesis pathways by mPGES-1/sEH/5-LO multi-target inhibition
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS. Vol. 5. Pag.100046-100046
ISSN:2772-4174.
Colarusso, Ester; Potenza, Marianna; Lauro, Gianluigi; Giovanna Chini, Maria; Sepe, Valentina; Zampella, Angela; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Bifulco, Giuseppe
Digital Object Identifier (DOI): 10.1016/j.ejmcr.2022.100046
Codice identificativo ISI: WOS:001108747600004
Codice identificativo SCOPUS: 2-s2.0-85132583529
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2022
Articolo in rivista
Extensive Molecular Dynamics Simulations Disclosed the Stability of mPGES-1 Enzyme and the Structural Role of Glutathione (GSH) Cofactor
MOLECULAR INFORMATICS. Pag.2200140-2200140
ISSN:1868-1743.
Di Micco, Simone; Lauro, Gianluigi; Bifulco, Giuseppe
Digital Object Identifier (DOI): 10.1002/minf.202200140
Codice identificativo ISI: WOS:000861445400001
Codice identificativo SCOPUS: 2-s2.0-85138952002
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2022
Articolo in rivista
Scabiosa atropurpurea: A rich source of iridoids with α-glucosidase inhibitory activity evaluated by in vitro and in silico studies
PHYTOCHEMISTRY. Vol. 205. Pag.113471-113471
ISSN:0031-9422.
Kılınc, Hilal; Masullo, Milena; Lauro, Gianluigi; D'Urso, Gilda; Alankus, Ozgen; Bifulco, Giuseppe; Piacente, Sonia
Digital Object Identifier (DOI): 10.1016/j.phytochem.2022.113471
Codice identificativo ISI: WOS:000880850100004
Codice identificativo SCOPUS: 2-s2.0-85140583901
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2022
Articolo in rivista
In Silico, In Vitro, and In Vivo Analysis of Tanshinone IIA and Cryptotanshinone from Salvia miltiorrhiza as Modulators of Cyclooxygenase-2/mPGES-1/Endothelial Prostaglandin EP3 Pathway
BIOMOLECULES. Vol. 12. Pag.99-99
ISSN:2218-273X.
Saviano, A.; De Vita, S.; Chini, M. G.; Marigliano, N.; Lauro, G.; Casillo, G. M.; Raucci, F.; Iorizzi, M.; Hofstetter, R. K.; Fischer, K.; Koeberle, A.; Werz, O.; Maione, F.; Bifulco, G.
Digital Object Identifier (DOI): 10.3390/biom12010099
Codice identificativo ISI: WOS:000747842600001
Codice identificativo SCOPUS: 2-s2.0-85122248050
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2022
Articolo in rivista
Phytochemical Analysis of the Methanolic Extract and Essential Oil from Leaves of Industrial Hemp Futura 75 Cultivar: Isolation of a New Cannabinoid Derivative and Biological Profile Using Computational Approaches
PLANTS. Vol. 11. Pag.1671-1691
ISSN:2223-7747.
De Vita, Simona; Finamore, Claudia; Chini, Maria Giovanna; Saviano, Gabriella; De Felice, Vincenzo; De Marino, Simona; Lauro, Gianluigi; Casapullo, Agostino; Fantasma, Francesca; Trombetta, Federico; Bifulco, Giuseppe; Iorizzi, Maria
Versione online
Digital Object Identifier (DOI): 10.3390/plants11131671
Codice identificativo ISI: WOS:000825696400001
Codice identificativo SCOPUS: 2-s2.0-85132770397
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2022
Articolo in rivista
Corylus avellana: A Source of Diarylheptanoids With α-Glucosidase Inhibitory Activity Evaluated by in vitro and in silico Studies
FRONTIERS IN PLANT SCIENCE. Vol. 13. Pag.805660-805660
ISSN:1664-462X.
Masullo, M.; Lauro, G.; Cerulli, A.; Bifulco, G.; Piacente, S.
Digital Object Identifier (DOI): 10.3389/fpls.2022.805660
Codice identificativo ISI: WOS:000761603900001
Codice identificativo SCOPUS: 2-s2.0-85125374215
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2022
Articolo in rivista
Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders
BIOORGANIC CHEMISTRY. Vol. 118. Pag.105480-105480
ISSN:0045-2068.
Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G.
Digital Object Identifier (DOI): 10.1016/j.bioorg.2021.105480
Codice identificativo ISI: WOS:000821662200006
Codice identificativo SCOPUS: 2-s2.0-85119580843
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2022
Articolo in rivista
Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein
MOLECULES. Vol. 27. Pag.665-665
ISSN:1420-3049.
Ruggiero, D.; Terracciano, S.; Lauro, G.; Pecoraro, M.; Franceschelli, S.; Bifulco, G.; Bruno, I.
Digital Object Identifier (DOI): 10.3390/molecules27030665
Codice identificativo ISI: WOS:000814371500001
Codice identificativo SCOPUS: 2-s2.0-85123075067
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2022
Articolo in rivista
6-Methylquinazolin-4(3H)-one Based Compounds as BRD9 Epigenetic Reader Binders: A Rational Combination of in silico Studies and Chemical Synthesis
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 2022. Pag.e202200868-e202200868
ISSN:1434-193X.
Colarusso, E; Gazzillo, E; Boccia, E; Giordano, A; Chini, Mg; Bifulco, G; Lauro, G
Digital Object Identifier (DOI): 10.1002/ejoc.202200868
Codice identificativo ISI: WOS:000854579600001
Codice identificativo SCOPUS: 2-s2.0-85138949165
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