Giuseppe BIFULCO | Publications
Giuseppe BIFULCO Publications
2011 | |
Articolo in rivista | |
Structure-Based Discovery of Inhibitors of Microsomal Prostaglandin E2 Synthase-1, 5-Lipoxygenase and 5-Lipoxygenase-Activating Protein: Promising Hits for the Development of New Anti-inflammatory Agents JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54 (6). Pag.1565-1575 ISSN:1520-4804. | |
R. De Simone; M. G. Chini; I. Bruno; R. Riccio; D. Mueller; O. Werz; G. Bifulco | |
Digital Object Identifier (DOI): 10.1021/jm101238d Codice identificativo ISI: WOS:000288400700003 Codice identificativo SCOPUS: 2-s2.0-79952788439 | |
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2011 | |
Articolo in rivista | |
Solomonsterols A and B from Theonella swinhoei. The First Example of C-24 and C-23 Sulfated Sterols from a Marine Source Endowed with a PXR Agonistic Activity JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54 (1). Pag.401-405 ISSN:1520-4804. | |
C. Festa; S. De Marino; M.V. D'Auria; G. Bifulco; B. Renga; S. Fiorucci; S. Petek; A.Zampella | |
Digital Object Identifier (DOI): 10.1021/jm100968b Codice identificativo ISI: WOS:000285818000036 Codice identificativo SCOPUS: 2-s2.0-78651112693 | |
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2011 | |
Articolo in rivista | |
The Binding Mode of Cladocoran A to the Human Group IIA Phospholipase A2. CHEMBIOCHEM. Vol. 12(17). Pag.2686-2691 ISSN:1439-4227. | |
M. C. Monti; M. G. Chini; L. Margarucci; R. Riccio; G. Bifulco; A. Casapullo | |
Digital Object Identifier (DOI): 10.1002/cbic.201100478 Codice identificativo ISI: WOS:000297160500025 Codice identificativo SCOPUS: 2-s2.0-81555196339 | |
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34427Structural basis for the potential antitumour activity of DNA-interacting benzo[kl]xanthene lignans
2011 | |
Articolo in rivista | |
Structural basis for the potential antitumour activity of DNA-interacting benzo[kl]xanthene lignans ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 9. Pag.701-710 ISSN:1477-0520. | |
S. Di Micco; F. Mazué; C. Daquino; C. Spatafora; D. Delmas; N. Latruffe; C. Tringali; R. Riccio; G. Bifulco | |
Digital Object Identifier (DOI): 10.1039/c0ob00480d Codice identificativo ISI: WOS:000286431500014 Codice identificativo SCOPUS: 2-s2.0-79251517428 | |
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2011 | |
Articolo in rivista | |
Towards new ligands of nuclear receptors. Discovery of malaitasterol A, an unique bis-secosterol from marine sponge Theonella swinhoei ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 9(13). Pag.4856-4862 ISSN:1477-0520. | |
S. De Marino; V. Sepe; M.V. D'Auria; G. Bifulco; B. Renga; S. Petek; S. Fiorucci; A. Zampella | |
Digital Object Identifier (DOI): 10.1039/C1OB05378G Codice identificativo ISI: WOS:000291654800026 Codice identificativo SCOPUS: 2-s2.0-79959759587 | |
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2011 | |
Articolo in rivista | |
Theonellasterols and Conicasterols from Theonella swinhoei. Novel Marine Natural Ligands for Human Nuclear Receptors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54(8). Pag.3065-3075 ISSN:1520-4804. | |
S. De Marino; R. Ummarino; M.V. D’Auria; M.G. Chini; G. Bifulco; B. Renga; C. D’Amore; S. Fiorucci; C. Debitus; A. Zampella | |
Digital Object Identifier (DOI): 10.1021/jm200169t Codice identificativo ISI: WOS:000289697800039 Codice identificativo SCOPUS: 2-s2.0-79955443595 | |
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2011 | |
Articolo in rivista | |
Inverse Virtual Screening of Antitumor Targets: Pilot Study on a Small Database of Natural Bioactive Compounds JOURNAL OF NATURAL PRODUCTS. Vol. 74 (6). Pag.1401-1407 ISSN:0163-3864. | |
G. Lauro; A. Romano; R. Riccio; G. Bifulco | |
Digital Object Identifier (DOI): 10.1021/np100935s Codice identificativo ISI: WOS:000291920600008 Codice identificativo SCOPUS: 2-s2.0-79959699687 | |
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2011 | |
Articolo in rivista | |
Solomonamides A and B, New Anti-inflammatory Peptides from Theonella swinhoei ORGANIC LETTERS. Vol. 13 (6). Pag.1532-1535 ISSN:1523-7060. | |
C. Festa; S. De Marino; V. Sepe; M.V. D'Auria; G. Bifulco; C. Débitus; M. Bucci; V. Vellecco; A.Zampella | |
Digital Object Identifier (DOI): 10.1021/ol200221n Codice identificativo ISI: WOS:000288148800069 Codice identificativo SCOPUS: 2-s2.0-79952615584 | |
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2011 | |
Articolo in rivista | |
Discovery of Sulfated Sterols from Marine Invertebrates as a New Class of Marine Natural Antagonists of Farnesoid-X-Receptor JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54(5). Pag.1314-1320 ISSN:1520-4804. | |
V. Sepe; G. Bifulco; B. Renga; C. D'Amore; S. Fiorucci; A. Zampella | |
Digital Object Identifier (DOI): 10.1021/jm101336m Codice identificativo ISI: WOS:000287833300019 Codice identificativo SCOPUS: 2-s2.0-79952274483 | |
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2011 | |
Articolo in rivista | |
The bile acid receptor GPBAR-1 (TGR5) modulates integrity of intestinal barrier and immune response to experimental Colitis. PLOS ONE. Vol. 6(10). Pag.e25637-e25637 ISSN:1932-6203. | |
S. Cipriani; A. Mencarelli; M.G. Chini; E. Distrutti; B. Renga; G. Bifulco; F. Baldelli; A. Donini; S. Fiorucci | |
Digital Object Identifier (DOI): 10.1371/journal.pone.0025637 Codice identificativo ISI: WOS:000296521400005 Codice identificativo SCOPUS: 2-s2.0-80055090450 | |
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2011 | |
Articolo in rivista | |
Farnesoid X Receptor Agonist for the Treatment of Liver and Metabolic Disorders: Focus on 6-ethyl-CDCA MINI-REVIEWS IN MEDICINAL CHEMISTRY. Vol. 11(9). Pag.753-762 ISSN:1389-5575. | |
S. Fiorucci; S. Cipriani; A. Mencarelli; F. Baldelli; G. Bifulco; A. Zampella | |
Digital Object Identifier (DOI): 10.2174/138955711796355258 Codice identificativo ISI: WOS:000294409300003 Codice identificativo SCOPUS: 2-s2.0-79960617989 | |
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2011 | |
Articolo in rivista | |
Perthamides C-F, potent human antipsoriatic cyclopeptides TETRAHEDRON. Vol. 67. Pag.7780-7786 ISSN:0040-4020. | |
C. Festa; S. De Marino; V. Sepe; MV. D'Auria; G.Bifulco; R. Andres; MC Terencio; M. Paya;C. Debitus; A. Zampella | |
Digital Object Identifier (DOI): 10.1016/j.tet.2011.07.077 Codice identificativo ISI: WOS:000295393700017 Codice identificativo SCOPUS: 2-s2.0-80052391994 | |
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