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Publications

Giuseppe BIFULCO Publications


2023
Articolo in rivista
2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines
BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 93. Pag.117444-117467
ISSN:1464-3391.
De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1016/j.bmc.2023.117444
Codice identificativo ISI: WOS:001064638100001
Codice identificativo SCOPUS: 2-s2.0-85168487978
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2023
Articolo in rivista
Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9
BIOORGANIC CHEMISTRY. Vol. 139. Pag.106677-106677
ISSN:0045-2068.
Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi
Digital Object Identifier (DOI): 10.1016/j.bioorg.2023.106677
Codice identificativo ISI: WOS:001031583200001
Codice identificativo SCOPUS: 2-s2.0-85163217544
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2023
Articolo in rivista
Target identification by structure-based computational approaches: Recent advances and perspectives
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. Vol. 83. Pag.129171-129171
ISSN:1464-3405.
De Vita, Simona; Chini, Maria Giovanna; Bifulco, Giuseppe; Lauro, Gianluigi
Digital Object Identifier (DOI): 10.1016/j.bmcl.2023.129171
Codice identificativo ISI: WOS:000944919600001
Codice identificativo SCOPUS: 2-s2.0-85147876194
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2023
Articolo in rivista
Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 247. Pag.115018-115018
ISSN:0223-5234.
Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi
Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.115018
Codice identificativo ISI: WOS:000913013400001
Codice identificativo SCOPUS: 2-s2.0-85144788456
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2023
Articolo in rivista
Identification of 2-Aminoacyl-1,3,4-thiadiazoles as Prostaglandin E2 and Leukotriene Biosynthesis Inhibitors
ACS MEDICINAL CHEMISTRY LETTERS. Vol. 14(1). Pag.26-34
ISSN:1948-5875.
Potenza, Marianna; Giordano, Assunta; Chini, Maria G; Saviano, Anella; Kretzer, Christian; Raucci, Federica; Russo, Marina; Lauro, Gianluigi; Terracciano, Stefania; Bruno, Ines; Iorizzi, Maria; Hofstetter, Robert K; Pace, Simona; Maione, Francesco; Werz, Oliver; Bifulco, Giuseppe
Digital Object Identifier (DOI): 10.1021/acsmedchemlett.2c00343
Codice identificativo SCOPUS: 2-s2.0-85143868000
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2023
Articolo in rivista
Design, Synthesis, and Pharmacological Characterization of a Potent Soluble Epoxide Hydrolase Inhibitor for the Treatment of Acute Pancreatitis
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 66. Pag.9201-9222
ISSN:0022-2623.
Musella, Simona; D'Avino, Danilo; Peltner, Lukas Klaus; Di Sarno, Veronica; Cerqua, Ida; Merciai, Fabrizio; Vestuto, Vincenzo; Ciaglia, Tania; Smaldone, Gerardina; Di Matteo, Francesca; Di Micco, Simone; Napolitano, Valeria; Bifulco, Giuseppe; Pepe, Giacomo; Sommella, Eduardo Maria; Basilicata, Manuela Giovanna; Aquino, Giovanna; Gomez-Monterrey, Isabel M; Campiglia, Pietro; Ostacolo, Carmine; Roviezzo, Fiorentina; Werz, Oliver; Rossi, Antonietta; Bertamino, Alessia
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c00831
Codice identificativo ISI: WOS:001011703200001
Codice identificativo SCOPUS: 2-s2.0-85164388377
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