Publications

Giuseppe BIFULCO Publications


2012
Articolo in rivista
Discovery That Theonellasterol a Marine Sponge Sterol Is a Highly Selective FXR Antagonist That Protects against Liver Injury in Cholestasis
PLOS ONE. Vol. 7. Pag.1-12
ISSN:1932-6203.
Barbara Renga;Andrea Mencarelli;Claudio D'Amore;Sabrina Cipriani;Maria Valeria D'Auria;Valentina Sepe;Maria Giovanna Chini;Maria Chiara Monti;Giuseppe Bifulco;Angela Zampella;Stefano Fiorucci
Digital Object Identifier (DOI): 10.1371/journal.pone.0030443
Codice identificativo ISI: WOS:000301570600043
Codice identificativo SCOPUS: 2-s2.0-84856084764
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2012
Articolo in rivista
Natural iminosugar (+)-lentiginosine inhibits ATPase and chaperone activity of Hsp90
PLOS ONE. Vol. 7(8). Pag.e43316-e43316
ISSN:1932-6203.
Dal Piaz Fabrizio; Vassallo Antonio; Chini Maria Giovanna; Cordero Franca M.; Cardona Francesca; Pisano Claudio; Bifulco Giuseppe; De Tommasi Nunziatina; Brandi Alberto
Versione online
Digital Object Identifier (DOI): 10.1371/journal.pone.0043316
Codice identificativo ISI: WOS:000307733800059
Codice identificativo SCOPUS: 2-s2.0-84865197487
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2012
Articolo in rivista
Preliminary Structure-Activity Relationship on Theonellasterol, a New Chemotype of FXR Antagonist, from the Marine Sponge Theonella swinhoei
MARINE DRUGS. Vol. 10. Pag.2448-2466
ISSN:1660-3397.
Valentina Sepe;Raffaella Ummarino;Maria D'Auria;Orazio Taglialatela-Scafati;Simona Marino;Claudio D'Amore;Barbara Renga;Maria Chini;Giuseppe Bifulco;Yoichi Nakao;Nobuhiro Fusetani;Stefano Fiorucci;Angela Zampella
Digital Object Identifier (DOI): 10.3390/md10112448
Codice identificativo ISI: WOS:000311425800006
Codice identificativo SCOPUS: 2-s2.0-84870003556
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2012
Articolo in rivista
Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors
CHEMMEDCHEM. Vol. 7. Pag.694-702
ISSN:1860-7179.
Stefania Terracciano;Maria Giovanna Chini;Raffaele Riccio;Ines Bruno;Giuseppe Bifulco
Digital Object Identifier (DOI): 10.1002/cmdc.201100531
Codice identificativo ISI: WOS:000302073100017
Codice identificativo SCOPUS: 2-s2.0-84859181022
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2012
Articolo in rivista
Conicasterol E, a Small Heterodimer Partner Sparing Farnesoid X Receptor Modulator Endowed with a Pregnane X Receptor Agonistic Activity, from the Marine SpongeTheonella swinhoei
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.84-93
ISSN:0022-2623.
Valentina Sepe;Raffaella Ummarino;Maria Valeria D’Auria;Maria Giovanna Chini;Giuseppe Bifulco;Barbara Renga;Claudio D’Amore;Cécile Debitus;Stefano Fiorucci;Angela Zampella
Digital Object Identifier (DOI): 10.1021/jm201004p
Codice identificativo ISI: WOS:000298978800007
Codice identificativo SCOPUS: 2-s2.0-84855837566
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2012
Articolo in rivista
Inverse Virtual Screening allows the discovery of the biological activity of natural compounds
BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 20. Pag.3596-3602
ISSN:0968-0896.
Gianluigi Lauro;Milena Masullo;Sonia Piacente;Raffaele Riccio;Giuseppe Bifulco
Digital Object Identifier (DOI): 10.1016/j.bmc.2012.03.072
Codice identificativo ISI: WOS:000303935800021
Codice identificativo SCOPUS: 2-s2.0-84861189353
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2012
Articolo in rivista
Gracilioethers E-J, new oxygenated polyketides from the marine sponge Plakinastrella mamillaris
TETRAHEDRON. Vol. 68. Pag.10157-10163
ISSN:0040-4020.
Carmen Festa;Simona De Marino;Maria Valeria D'Auria;Eric Deharo;German Gonzalez;Chloe Deyssard;Sylvain Petek;Giuseppe Bifulco;Angela Zampella
Digital Object Identifier (DOI): 10.1016/j.tet.2012.09.106
Codice identificativo ISI: WOS:000310817700007
Codice identificativo SCOPUS: 2-s2.0-84867865059
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2012
Articolo in rivista
Marine sponge steroids as nuclear receptor ligands
TRENDS IN PHARMACOLOGICAL SCIENCES. Vol. 33, (11). Pag.591-601
ISSN:0165-6147.
Stefano Fiorucci;Eleonora Distrutti;Giuseppe Bifulco;Maria Valeria D’Auria;Angela Zampella
Digital Object Identifier (DOI): 10.1016/j.tips.2012.08.004
Codice identificativo ISI: WOS:000311176900006
Codice identificativo SCOPUS: 2-s2.0-84867894196
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2012
Articolo in rivista
Design and synthesis of a second series of triazole-based compounds as potent dual mPGES-1 and 5-lipoxygenase inhibitors
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54. Pag.311-323
ISSN:0223-5234.
Maria Giovanna Chini;Rosa De Simone;Ines Bruno;Raffaele Riccio;Friederike Dehm;Christina Weinigel;Dagmar Barz;Oliver Werz;Giuseppe Bifulco
Digital Object Identifier (DOI): 10.1016/j.ejmech.2012.05.014
Codice identificativo ISI: WOS:000307920600034
Codice identificativo SCOPUS: 2-s2.0-84864408638
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2012
Articolo in rivista
The Inactivation Mechanism of Human Group IIA Phospholipase A2by Scalaradial
CHEMBIOCHEM. Vol. 13. Pag.2259-2264
ISSN:1439-4227.
Luigi Margarucci;Maria Chiara Monti;Maria Giovanna Chini;Alessandra Tosco;Raffaele Riccio;Giuseppe Bifulco;Agostino Casapullo
Digital Object Identifier (DOI): 10.1002/cbic.201200453
Codice identificativo ISI: WOS:000309596000015
Codice identificativo SCOPUS: 2-s2.0-84867224490
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2012
Articolo in rivista
Plakilactones from the marine sponge Plakinastrella mamillaris. Discovery of a new class of marine ligands of peroxisome proliferator-activated receptor γ
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.8303-8317
ISSN:0022-2623.
Festa, Carmen; Lauro, Gianluigi; De Marino, Simon; D'Auria, Maria Valeria; Monti, Maria Chiara; Casapullo, Agostino; D'Amore, Claudio; Renga, Barbara; Mencarelli, Andrea; Petek, Sylvain; Bifulco, Giuseppe; Fiorucci, Stefano; Zampella, Angela
Digital Object Identifier (DOI): 10.1021/jm300911g
Codice identificativo ISI: WOS:000309643500010
Codice identificativo SCOPUS: 2-s2.0-84867352661
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2012
Articolo in rivista
Modification in the side chain of solomonsterol A: discovery of cholestan disulfate as a potent pregnane-X-receptor agonist
ORGANIC & BIOMOLECULAR CHEMISTRY. Vol. 10. Pag.6350-6362
ISSN:1477-0520.
Valentina Sepe;Raffaella Ummarino;Maria Valeria DAuria;Gianluigi Lauro;Giuseppe Bifulco;Claudio D'Amore;Barbara Renga;Stefano Fiorucci;Angela Zampella
Digital Object Identifier (DOI): 10.1039/c2ob25800e
Codice identificativo ISI: WOS:000306480100014
Codice identificativo SCOPUS: 2-s2.0-84863908159
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2012
Articolo in rivista
Synthesis of Enantiopure 7-Substituted Azepane-2-Carboxylic Acids as Templates for Conformationally Constrained Peptidomimetics
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 11. Pag.2133-2141
ISSN:1434-193X.
Cini Elena; Bifulco Giuseppe; Menchi Gloria; Rodriquez Manuela; Taddei Maurizio
Digital Object Identifier (DOI): 10.1002/ejoc.201101387
Codice identificativo ISI: WOS:000302621400007
Codice identificativo SCOPUS: 2-s2.0-84859232982
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2012
Articolo in rivista
4-Methylenesterols from Theonella swinhoei sponge are natural pregnane-X-receptor agonists and farnesoid-X-receptor antagonists that modulate innate immunity
STEROIDS. Vol. 77. Pag.484-495
ISSN:0039-128X.
Simona De Marino;Raffaella Ummarino;Maria Valeria D’Auria;Maria Giovanna Chini;Giuseppe Bifulco;Claudio D’Amore;Barbara Renga;Andrea Mencarelli;Sylvain Petek;Stefano Fiorucci;Angela Zampella
Digital Object Identifier (DOI): 10.1016/j.steroids.2012.01.006
Codice identificativo ISI: WOS:000303084000019
Codice identificativo SCOPUS: 2-s2.0-84858337325
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2012
Articolo in rivista
Structural characterization of tetranortriterpenes from Pseudrocedrela kotschyi and Trichilia emetica and study of their activity towards the chaperone Hsp90
PHYTOCHEMISTRY. Vol. 75. Pag.78-89
ISSN:0031-9422.
Fabrizio Dal Piaz;Nicola Malafronte;Adriana Romano;Dario Gallotta;Maria Antonietta Belisario;Giuseppe Bifulco;Maria Josefine Gualtieri;Rokia Sanogo;Nunziatina De Tommasi;Claudio Pisano
Digital Object Identifier (DOI): 10.1016/j.phytochem.2011.12.002
Codice identificativo ISI: WOS:000300868600009
Codice identificativo SCOPUS: 2-s2.0-84856227300
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2012
Articolo in rivista
Quantitative NMR-Derived Interproton Distances Combined with Quantum Mechanical Calculations of13C Chemical Shifts in the Stereochemical Determination of Conicasterol F, a Nuclear Receptor Ligand fromTheonella swinhoei
JOURNAL OF ORGANIC CHEMISTRY. Vol. 77. Pag.1489-1496
ISSN:0022-3263.
Maria Giovanna Chini;Catharine R. Jones;Angela Zampella;Maria Valeria D’Auria;Barbara Renga;Stefano Fiorucci;Craig P. Butts;Giuseppe Bifulco
Digital Object Identifier (DOI): 10.1021/jo2023763
Codice identificativo ISI: WOS:000300462700027
Codice identificativo SCOPUS: 2-s2.0-84856637775
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2012
Articolo in rivista
Aetheramides A and B, Potent HIV-Inhibitory Depsipeptides from a Myxobacterium of the New Genus “Aetherobacter”
ORGANIC LETTERS. Vol. 14. Pag.2854-2857
ISSN:1523-7060.
Alberto Plaza;Ronald Garcia;Giuseppe Bifulco;Javier Pablo Martinez;Stephan Hüttel;Florenz Sasse;Andreas Meyerhans;Marc Stadler;Rolf Müller
Digital Object Identifier (DOI): 10.1021/ol3011002
Codice identificativo ISI: WOS:000304682700051
Codice identificativo SCOPUS: 2-s2.0-84861838031
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2012
Articolo in rivista
Discovery and Synthesis of Namalide Reveals a New Anabaenopeptin Scaffold and Peptidase Inhibitor
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.735-742
ISSN:0022-2623.
Cheruku, Pradeep; Plaza, Alberto; Lauro, Gianluigi; Keffer, Jessica; Lloyd, John R.; Bifulco, Giuseppe; Bewley, Carole A.
Digital Object Identifier (DOI): 10.1021/jm201238p
Codice identificativo ISI: WOS:000299453300017
Codice identificativo SCOPUS: 2-s2.0-84856367249
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2012
Contributo in volume (Capitolo o Saggio)
Quantum Chemical Calculation of Chemical Shifts in the Stereochemical Determination of Organic Compounds: A Practical Approach.
In Handbook of Marine Natural Products Pag.571-599 New York, Heidelberg, London Springer.
ISBN:9789048138333; 9789048138340
Simone Di Micco; Maria Giovanna Chini; Raffaele Riccio; Giuseppe Bifulco
Versione online
Digital Object Identifier (DOI): 10.1007/978-90-481-3834-0_10
Codice identificativo SCOPUS: 2-s2.0-84891930570
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