Gianluca SBARDELLA | Publications
Gianluca SBARDELLA Publications
2017 | |
Articolo in rivista | |
A transcriptional coregulator, SPIN-DOC, attenuates the coactivator activity of Spindlin1 THE JOURNAL OF BIOLOGICAL CHEMISTRY. Vol. 292. Pag.20808-20817 ISSN:0021-9258. | |
Bae, Narkhyun; Gao, Min; Li, Xu; Premkumar, Tolkappiyan; Sbardella, Gianluca; Chen, Junjie; Bedford, Mark T. | |
Versione online | |
Digital Object Identifier (DOI): 10.1074/JBC.M117.814913 Codice identificativo ISI: WOS:000418453400001 Codice identificativo SCOPUS: 2-s2.0-85039439820 | |
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2017 | |
Articolo in rivista | |
Developing Spindlin1 small-molecule inhibitors by using protein microarrays NATURE CHEMICAL BIOLOGY. Vol. 13. Pag.750-756 ISSN:1552-4450. | |
Bae, Narkhyun; Viviano, Monica; Su, Xiaonan; Lv, Jie; Cheng, Donghang; Sagum, Cari; Castellano, Sabrina; Bai, Xue; Johnson, Claire; Khalil, Mahmoud Ibrahim; Shen, Jianjun; Chen, Kaifu; Li, Haitao; Sbardella, Gianluca; Bedford, Mark T. | |
Versione online | |
Digital Object Identifier (DOI): 10.1038/nchembio.2377 Codice identificativo ISI: WOS:000403673700011 Codice identificativo SCOPUS: 2-s2.0-85021067771 | |
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2017 | |
Articolo in rivista | |
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) JOURNAL OF MEDICINAL CHEMISTRY. Vol. 60. Pag.7897-7909 ISSN:0022-2623. | |
Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia | |
Versione online | |
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.7b01031 Codice identificativo ISI: WOS:000412150300017 Codice identificativo SCOPUS: 2-s2.0-85030253369 | |
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2017 | |
Articolo in rivista | |
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation MOLECULAR CANCER RESEARCH. Vol. 15. Pag.1073-1084 ISSN:1541-7786. | |
Dobson, Tara; Hatcher, Rashieda J; Swaminathan, Jyothismathi; Das, Chandra M; Shaik, Shavali; Tao, Rong Hua; Milite, Ciro; Castellano, Sabrina; Taylor, Pete; Sbardella, Gianluca; Gopalakrishnan, Vidya | |
Versione online | |
Digital Object Identifier (DOI): 10.1158/1541-7786.MCR-16-0424 Codice identificativo ISI: WOS:000406681200011 Codice identificativo SCOPUS: 2-s2.0-85026641347 | |
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2017 | |
Articolo in rivista | |
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer SCIENTIFIC REPORTS. Vol. 7. Pag.1-14 ISSN:2045-2322. | |
Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia | |
Versione online | |
Digital Object Identifier (DOI): 10.1038/s41598-017-11688-x Codice identificativo ISI: WOS:000410859400010 Codice identificativo SCOPUS: 2-s2.0-85029517928 | |
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2017 | |
Articolo in rivista | |
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA. Vol. 114. Pag.3625-3630 ISSN:0027-8424. | |
van Haren, Matthijs J.; Marechal, Nils; Troffer Charlier, Nathalie; Cianciulli, Agostino; Sbardella, Gianluca; Cavarelli, Jean; Martin, Nathaniel I. | |
Versione online | |
Digital Object Identifier (DOI): 10.1073/pnas.1618401114 Codice identificativo ISI: WOS:000398159000042 Codice identificativo SCOPUS: 2-s2.0-85016997146 | |
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