Publications

Gianluca SBARDELLA Publications


2017
Articolo in rivista
A transcriptional coregulator, SPIN-DOC, attenuates the coactivator activity of Spindlin1
THE JOURNAL OF BIOLOGICAL CHEMISTRY. Vol. 292. Pag.20808-20817
ISSN:0021-9258.
Bae, Narkhyun; Gao, Min; Li, Xu; Premkumar, Tolkappiyan; Sbardella, Gianluca; Chen, Junjie; Bedford, Mark T.
Versione online
Digital Object Identifier (DOI): 10.1074/JBC.M117.814913
Codice identificativo ISI: WOS:000418453400001
Codice identificativo SCOPUS: 2-s2.0-85039439820
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2017
Articolo in rivista
Developing Spindlin1 small-molecule inhibitors by using protein microarrays
NATURE CHEMICAL BIOLOGY. Vol. 13. Pag.750-756
ISSN:1552-4450.
Bae, Narkhyun; Viviano, Monica; Su, Xiaonan; Lv, Jie; Cheng, Donghang; Sagum, Cari; Castellano, Sabrina; Bai, Xue; Johnson, Claire; Khalil, Mahmoud Ibrahim; Shen, Jianjun; Chen, Kaifu; Li, Haitao; Sbardella, Gianluca; Bedford, Mark T.
Versione online
Digital Object Identifier (DOI): 10.1038/nchembio.2377
Codice identificativo ISI: WOS:000403673700011
Codice identificativo SCOPUS: 2-s2.0-85021067771
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2017
Articolo in rivista
Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO)
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 60. Pag.7897-7909
ISSN:0022-2623.
Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.7b01031
Codice identificativo ISI: WOS:000412150300017
Codice identificativo SCOPUS: 2-s2.0-85030253369
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2017
Articolo in rivista
Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation
MOLECULAR CANCER RESEARCH. Vol. 15. Pag.1073-1084
ISSN:1541-7786.
Dobson, Tara; Hatcher, Rashieda J; Swaminathan, Jyothismathi; Das, Chandra M; Shaik, Shavali; Tao, Rong Hua; Milite, Ciro; Castellano, Sabrina; Taylor, Pete; Sbardella, Gianluca; Gopalakrishnan, Vidya
Versione online
Digital Object Identifier (DOI): 10.1158/1541-7786.MCR-16-0424
Codice identificativo ISI: WOS:000406681200011
Codice identificativo SCOPUS: 2-s2.0-85026641347
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2017
Articolo in rivista
Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer
SCIENTIFIC REPORTS. Vol. 7. Pag.1-14
ISSN:2045-2322.
Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia
Versione online
Digital Object Identifier (DOI): 10.1038/s41598-017-11688-x
Codice identificativo ISI: WOS:000410859400010
Codice identificativo SCOPUS: 2-s2.0-85029517928
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2017
Articolo in rivista
Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA. Vol. 114. Pag.3625-3630
ISSN:0027-8424.
van Haren, Matthijs J.; Marechal, Nils; Troffer Charlier, Nathalie; Cianciulli, Agostino; Sbardella, Gianluca; Cavarelli, Jean; Martin, Nathaniel I.
Versione online
Digital Object Identifier (DOI): 10.1073/pnas.1618401114
Codice identificativo ISI: WOS:000398159000042
Codice identificativo SCOPUS: 2-s2.0-85016997146
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