Publications

Gianluca SBARDELLA Publications


2025
Articolo in rivista
New pyridobenothiazolone derivatives display nanomolar pan‐serotype anti‐DENV activity
CHEMMEDCHEM. Pag.1-47
ISSN:1860-7179.
Felicetti, Tommaso; Gwee, Chin Piaw; Chan, Kitti Wing Ki; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Watanabe, Satoru; Mazlan, Muhammad Danial Bin Mohd; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Sbardella, Gianluca; Vasudevan, Subhash G.; Manfroni, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1002/cmdc.202500163
Codice identificativo ISI: WOS:001471484800001
Codice identificativo SCOPUS: 2-s2.0-105003262433
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2025
Articolo in rivista
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit to Lead
CHEMMEDCHEM. Pag.1-8
ISSN:1860-7179.
Quancard, Jean; Bach, Anders; Borsari, Chiara; Craft, Russell; Gnamm, Christian; Guéret, Stéphanie M.; Hartung, Ingo V.; Koolman, Hannes F.; Laufer, Stefan; Lepri, Susan; Messinger, Josef; Ritter, Kurt; Sbardella, Gianluca; Unzue Lopez, Andrea; Willwacher, Marina K.; Cox, Brian; Young, Robert J.
Versione online
Digital Object Identifier (DOI): 10.1002/cmdc.202400931
Codice identificativo ISI: WOS:001422091900001
Codice identificativo SCOPUS: 2-s2.0-86000008260
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2025
Articolo in rivista
An Amazing 30-Year Journey around the DABO Family: A Medicinal Chemistry Lesson on a Versatile Class of Non-nucleoside HIV-1 Reverse Transcriptase Inhibitors
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 68. Pag.5993-6026
ISSN:0022-2623.
Fabbrizi, Emanuele; Chernyshov, Vladimir V.; Fiorentino, Francesco; Sbardella, Gianluca; Ragno, Rino; Nawrozkij, Maxim; Ivanov, Roman; Rotili, Dante; Mai, Antonello
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.4c02848
Codice identificativo ISI: WOS:001440408700001
Codice identificativo SCOPUS: 2-s2.0-86000539361
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2025
Articolo in rivista
In Quest of Chemical Probes for DNA Methylation Reader Proteins: Nucleoside and Dimer Analogues of 5‐Methylcytosine Interact with MBD2
ANGEWANDTE CHEMIE. INTERNATIONAL EDITION. Vol. 64. Pag.e202425599-e202425599
ISSN:1433-7851.
Contreras, Jean; Vichier-Guerre, Sophie; Dugué, Laurence; Bonhomme, Frédéric; Jallet, Corinne; Nguyen, Minh-Ha; Vitorge, Bruno; Feoli, Alessandra; Sbardella, Gianluca; Guijarro, J. Iñaki; Arimondo, Paola
Versione online
Digital Object Identifier (DOI): 10.1002/anie.202425599
Codice identificativo ISI: WOS:001483207600001
Codice identificativo SCOPUS: 2-s2.0-105004692795
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