Stefania TERRACCIANO | Publications
Stefania TERRACCIANO Publications
| 2024 | |
| Articolo in rivista | |
| Chemoproteomics Reveals USP5 (Ubiquitin Carboxyl-Terminal Hydrolase 5) as Promising Target of the Marine Polyketide Gracilioether A MARINE DRUGS. Vol. 22. Pag.41-52 ISSN:1660-3397. | |
| Capuano, A.; D'Urso, G.; Aliberti, M.; Ruggiero, D.; Terracciano, S.; Festa, C.; Tosco, A.; Chini, M. G.; Lauro, G.; Bifulco, G.; Casapullo, A. | |
| Digital Object Identifier (DOI): 10.3390/md22010041 Codice identificativo ISI: WOS:001150851600001 Codice identificativo SCOPUS: 2-s2.0-85183127360 | |
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| 2023 | |
| Articolo in rivista | |
| A multidisciplinary functional proteomics-aided strategy as a tool for the profiling of a novel cytotoxic thiadiazolopyrimidone BIOORGANIC CHEMISTRY. Vol. 138. Pag.106620-106632 ISSN:0045-2068. | |
| Morretta, Elva; Ruggiero, Dafne; Belvedere, Raffaella; Petrella, Antonello; Bruno, Ines; Terracciano, Stefania; Monti, Maria Chiara | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2023.106620 Codice identificativo ISI: WOS:001011723900001 Codice identificativo SCOPUS: 2-s2.0-85159816112 | |
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| 2023 | |
| Articolo in rivista | |
| Exploring the chemical space of functionalized [1,2,4]triazolo[4,3-a]quinoxaline-based compounds targeting the bromodomain of BRD9 BIOORGANIC CHEMISTRY. Vol. 139. Pag.106677-106677 ISSN:0045-2068. | |
| Gazzillo, Erica; Pierri, Martina; Colarusso, Ester; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Bruno, Ines; Bifulco, Giuseppe; Terracciano, Stefania; Lauro, Gianluigi | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2023.106677 Codice identificativo ISI: WOS:001031583200001 Codice identificativo SCOPUS: 2-s2.0-85163217544 | |
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| 2023 | |
| Articolo in rivista | |
| 2-Substituted 1,5-benzothiazepine-based HDAC inhibitors exert anticancer activities on human solid and acute myeloid leukemia cell lines BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 93. Pag.117444-117467 ISSN:1464-3391. | |
| De Vita, Simona; Meninno, Sara; Capasso, Lucia; Colarusso, Ester; Chini, Maria Giovanna; Lauro, Gianluigi; Rinaldi, Romolo; De Cicco, Annalisa; Sian, Veronica; Terracciano, Stefania; Nebbioso, Angela; Lattanzi, Alessandra; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2023.117444 Codice identificativo ISI: WOS:001064638100001 Codice identificativo SCOPUS: 2-s2.0-85168487978 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based small molecules as selective BRD9 binders EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 247. Pag.115018-115018 ISSN:0223-5234. | |
| Colarusso, Ester; Ceccacci, Sara; Monti, Maria Chiara; Gazzillo, Erica; Giordano, Assunta; Chini, Maria Giovanna; Ferraro, Maria Grazia; Piccolo, Marialuisa; Ruggiero, Dafne; Irace, Carlo; Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Lauro, Gianluigi | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.115018 Codice identificativo ISI: WOS:000913013400001 Codice identificativo SCOPUS: 2-s2.0-85144788456 | |
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| 2022 | |
| Articolo in rivista | |
| Structural Refinement of 2,4-Thiazolidinedione Derivatives as New Anticancer Agents Able to Modulate the BAG3 Protein MOLECULES. Vol. 27. Pag.665-665 ISSN:1420-3049. | |
| Ruggiero, D.; Terracciano, S.; Lauro, G.; Pecoraro, M.; Franceschelli, S.; Bifulco, G.; Bruno, I. | |
| Digital Object Identifier (DOI): 10.3390/molecules27030665 Codice identificativo ISI: WOS:000814371500001 Codice identificativo SCOPUS: 2-s2.0-85123075067 | |
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| 2022 | |
| Articolo in rivista | |
| Identification of 2,4-Dinitro-Biphenyl-Based Compounds as MAPEG Inhibitors CHEMMEDCHEM. Pag.ecmdc.202200327-ecmdc.202200327 ISSN:1860-7179. | |
| Di Micco, Simone; Terracciano, Stefania; Pierri, Martina; Cantone, Vincenza; Liening, Stefanie; König, Stefanie; Garscha, Ulrike; Hofstetter, Robert Klaus; Koeberle, Andreas; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202200327 Codice identificativo ISI: WOS:000865844400001 Codice identificativo SCOPUS: 2-s2.0-85139716470 | |
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| 2022 | |
| Articolo in rivista | |
| Introducing structure-based three-dimensional pharmacophore models for accelerating the discovery of selective BRD9 binders BIOORGANIC CHEMISTRY. Vol. 118. Pag.105480-105480 ISSN:0045-2068. | |
| Pierri, M.; Gazzillo, E.; Chini, M. G.; Ferraro, M. G.; Piccolo, M.; Maione, F.; Irace, C.; Bifulco, G.; Bruno, I.; Terracciano, S.; Lauro, G. | |
| Digital Object Identifier (DOI): 10.1016/j.bioorg.2021.105480 Codice identificativo ISI: WOS:000821662200006 Codice identificativo SCOPUS: 2-s2.0-85119580843 | |
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| 2022 | |
| Articolo in rivista | |
| Repositioning of Quinazolinedione-Based Compounds on Soluble Epoxide Hydrolase (sEH) through 3D Structure-Based Pharmacophore Model-Driven Investigation MOLECULES. Vol. 27. Pag.3866-3866 ISSN:1420-3049. | |
| Gazzillo, Erica; Terracciano, Stefania; Ruggiero, Dafne; Potenza, Marianna; Chini, Maria Giovanna; Lauro, Gianluigi; Fischer, Katrin; Hofstetter, Robert Klaus; Giordano, Assunta; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.3390/molecules27123866 Codice identificativo ISI: WOS:000819099100001 Codice identificativo SCOPUS: 2-s2.0-85132592035 | |
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| 2021 | |
| Articolo in rivista | |
| Identification of 2-(thiophen-2-yl)acetic Acid-Based Lead Compound for mPGES-1 Inhibition FRONTIERS IN CHEMISTRY. Vol. 9. Pag.676631-676631 ISSN:2296-2646. | |
| Di Micco, S.; Terracciano, S.; Ruggiero, D.; Potenza, M.; Vaccaro, M. C.; Fischer, K.; Werz, O.; Bruno, I.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.3389/fchem.2021.676631 Codice identificativo ISI: WOS:000653652800001 Codice identificativo SCOPUS: 2-s2.0-85107041691 | |
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| 2020 | |
| Articolo in rivista | |
| A Combinatorial Virtual Screening Approach Driving the Synthesis of 2,4-Thiazolidinedione-Based Molecules as New Dual mPGES-1/5-LO Inhibitors CHEMMEDCHEM. Vol. 15. Pag.481-489 ISSN:1860-7179. | |
| Lauro, G.; Terracciano, S.; Cantone, V.; Ruggiero, D.; Fischer, K.; Pace, S.; Werz, O.; Bruno, I.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201900694 Codice identificativo ISI: WOS:000513689000001 Codice identificativo SCOPUS: 2-s2.0-85079711216 | |
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| 2020 | |
| Articolo in rivista | |
| Targeting mPGES-1 by a Combinatorial Approach: Identification of the Aminobenzothiazole Scaffold to Suppress PGE2Levels ACS MEDICINAL CHEMISTRY LETTERS. Vol. 11. Pag.783-789 ISSN:1948-5875. | |
| Chini, M. G.; Giordano, A.; Potenza, M.; Terracciano, S.; Fischer, K.; Vaccaro, M. C.; Colarusso, E.; Bruno, I.; Riccio, R.; Koeberle, A.; Werz, O.; Bifulco, G. | |
| Digital Object Identifier (DOI): 10.1021/acsmedchemlett.9b00618 Codice identificativo ISI: WOS:000535281200027 Codice identificativo SCOPUS: 2-s2.0-85087688875 | |
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| 2020 | |
| Articolo in rivista | |
| From Natural Compounds to Bioactive Molecules through NMR and In Silico Methodologies EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. Vol. 2020. Pag.6297-6317 ISSN:1434-193X. | |
| DE VITA, Simona; Terracciano, Stefania; Bruno, Ines; Giovanna Chini, Maria | |
| Digital Object Identifier (DOI): 10.1002/ejoc.202000469 Codice identificativo ISI: WOS:000553080700001 Codice identificativo SCOPUS: 2-s2.0-85088595349 | |
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| 2020 | |
| Articolo in rivista | |
| Discovery of noscapine derivatives as potential β-tubulin inhibitors BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 30. Pag.127489-127489 ISSN:0960-894X. | |
| Nemati, F.; Salehi, P.; Bararjanian, M.; Hadian, N.; Mohebbi, M.; Lauro, G.; Ruggiero, D.; Terracciano, S.; Bifulco, G.; Bruno, I. | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2020.127489 Codice identificativo ISI: WOS:000576786000002 Codice identificativo SCOPUS: 2-s2.0-85089348593 | |
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| 2019 | |
| Articolo in rivista | |
| Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition ACS MEDICINAL CHEMISTRY LETTERS. Vol. 10. Pag.601-605 ISSN:1948-5875. | |
| Giordano, Assunta; Forte, Giovanni; Terracciano, Stefania; Russo, Alessandra; Sala, Marina; Scala, Maria C.; Johansson, Catrine; Oppermann, Udo; Riccio, Raffaele; Bruno, Ines; Di Micco, Simone | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acsmedchemlett.8b00589 Codice identificativo ISI: WOS:000464767700036 Codice identificativo SCOPUS: 2-s2.0-85064335016 | |
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| 2019 | |
| Articolo in rivista | |
| Protein Preparation Automatic Protocol for High-Throughput Inverse Virtual Screening: Accelerating the Target Identification by Computational Methods JOURNAL OF CHEMICAL INFORMATION AND MODELING. Pag.4678-4690 ISSN:1549-9596. | |
| De Vita, S.; Lauro, G.; Ruggiero, D.; Terracciano, S.; Riccio, R.; Bifulco, G. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jcim.9b00428 Codice identificativo ISI: WOS:000500038700018 Codice identificativo SCOPUS: 2-s2.0-85074665461 | |
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146707Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors
| 2018 | |
| Articolo in rivista | |
| Identification by Inverse Virtual Screening of magnolol-based scaffold as new tankyrase-2 inhibitors BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 26. Pag.3953-3957 ISSN:0968-0896. | |
| DI MICCO, Simone; Luana, Pulvirenti; Bruno, Ines; Terracciano, Stefania; Russo, Alessandra; Vaccaro, Mariacarmela; Ruggiero, Dafne; Vera, Muccilli; Nunzio, Cardullo; Corrado, Tringali; Riccio, Raffaele; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2018.06.019 Codice identificativo ISI: WOS:000440942100012 Codice identificativo SCOPUS: 2-s2.0-85048836726 | |
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| 2018 | |
| Articolo in rivista | |
| Glucopyranosylbianthrones from the Algerian Asphodelus tenuifolius: Structural Insights and Biological Evaluation on Melanoma Cancer Cells JOURNAL OF NATURAL PRODUCTS. Vol. 81. Pag.1786-1794 ISSN:0163-3864. | |
| Ayoub, Khalfaoui; Chini, MARIA GIOVANNA; Mohamed, Bouheroum; Soumia, Belaabed; Lauro, Gianluigi; Terracciano, Stefania; Vaccaro, Mariacarmela; Bruno, Ines; Samir, Benayache; Ines, Mancini; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.8b00234 Codice identificativo ISI: WOS:000443103700011 Codice identificativo SCOPUS: 2-s2.0-85052588349 | |
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| 2018 | |
| Articolo in rivista | |
| Discovery of new potent molecular entities able to inhibit mPGES-1 EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 143. Pag.1419-1427 ISSN:0223-5234. | |
| Di Micco, Simone; Terracciano, Stefania; Cantone, Vincenza; Fischer, Katrin; Koeberle, Andreas; Foglia, Antonio; Riccio, Raffaele; Werz, Oliver; Bruno, Ines; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2017.10.039 Codice identificativo ISI: WOS:000423641400021 Codice identificativo SCOPUS: 2-s2.0-85033582141 | |
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| 2018 | |
| Articolo in rivista | |
| Discovery of new molecular entities able to strongly interfere with Hsp90 C-terminal domain SCIENTIFIC REPORTS. Vol. 8. Pag.1709-1709 ISSN:2045-2322. | |
| Terracciano, Stefania; Russo, Alessandra; Chini, Maria G.; Vaccaro, Maria C.; Potenza, Marianna; Vassallo, Antonio; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/s41598-017-14902-y Codice identificativo ISI: WOS:000423428300037 Codice identificativo SCOPUS: 2-s2.0-85041134440 | |
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| 2018 | |
| Articolo in rivista | |
| Discovery and synthesis of the first selective BAG domain modulator of BAG3 as an attractive candidate for the development of a new class of chemotherapeutics CHEMICAL COMMUNICATIONS. Vol. 54. Pag.7613-7616 ISSN:1359-7345. | |
| Terracciano, Stefania; Lauro, Gianluigi; Russo, Alessandra; Vaccaro, Maria Carmela; Vassallo, Antonio; De Marco, Margot; Ranieri, Bianca; Rosati, Alessandra; Turco, Maria Caterina; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c8cc03399d Codice identificativo ISI: WOS:000442118800009 Codice identificativo SCOPUS: 2-s2.0-85049623511 | |
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119360Cyclic Peptoids as Mycotoxin Mimics: An Exploration of Their Structural and Biological Properties
| 2017 | |
| Articolo in rivista | |
| Cyclic Peptoids as Mycotoxin Mimics: An Exploration of Their Structural and Biological Properties JOURNAL OF ORGANIC CHEMISTRY. Vol. 82. Pag.8848-8863 ISSN:0022-3263. | |
| D'Amato, Assunta; Volpe, Raffaele; Vaccaro, Maria Carmela; Terracciano, Stefania; Bruno, Ines; Tosolini, Massimo; Tedesco, Consiglia; Pierri, Giovanni; Tecilla, Paolo; Costabile, Chiara; DELLA SALA, Giorgio; Izzo, Irene; DE RICCARDIS, Francesco | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.joc.7b00965 Codice identificativo ISI: WOS:000410004800006 Codice identificativo SCOPUS: 2-s2.0-85028765857 | |
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| 2017 | |
| Articolo in rivista | |
| Identification of novel microsomal prostaglandin E2 synthase-1 (mPGES-1) lead inhibitors from Fragment Virtual Screening EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 125. Pag.278-287 ISSN:0223-5234. | |
| Lauro, Gianluigi; Manfra, Michele; Pedatella, Silvana; Fischer, Katrin; Cantone, Vincenza; Terracciano, Stefania; Bertamino, Alessia; Ostacolo, Carmine; Gomez Monterrey, Isabel; De Nisco, Mauro; Riccio, Raffaele; Novellino, Ettore; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2016.09.042 Codice identificativo ISI: WOS:000390496600020 Codice identificativo SCOPUS: 2-s2.0-84988579046 | |
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| 2016 | |
| Articolo in rivista | |
| Correction: Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors CHEMICAL COMMUNICATIONS. Vol. 52. Pag.13515-13515 ISSN:1364-548X. | |
| Terracciano, Stefania; Chini, Maria Giovanna; Vaccaro, Mariacarmela; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Digital Object Identifier (DOI): 10.1039/c6cc90506d Codice identificativo ISI: WOS:000388202900021 Codice identificativo SCOPUS: 2-s2.0-84994802440 | |
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| 2016 | |
| Articolo in rivista | |
| New dihydropyrimidin-2(1H)-one based Hsp90 C-terminal inhibitors RSC ADVANCES. Vol. 6. Pag.82330-82340 ISSN:2046-2069. | |
| Terracciano, Stefania; Foglia, Antonio; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Russo, Alessandra; DAL PIAZ, Fabrizio; Saturnino, C.; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c6ra17235k Codice identificativo ISI: WOS:000382776000109 Codice identificativo SCOPUS: 2-s2.0-84984802054 | |
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| 2016 | |
| Articolo in rivista | |
| Identification of the key structural elements of a dihydropyrimidinone core driving toward more potent Hsp90 C-terminal inhibitors CHEMICAL COMMUNICATIONS. Vol. 52. Pag.12857-12860 ISSN:1359-7345. | |
| Terracciano, Stefania; Chini, MARIA GIOVANNA; Vaccaro, M. C.; Strocchia, Maria; Foglia, Antonio; Vassallo, Antonio; Saturnino, Carmela; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c6cc06379a Codice identificativo ISI: WOS:000387025600015 Codice identificativo SCOPUS: 2-s2.0-84992740815 | |
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| 2016 | |
| Articolo in rivista | |
| Structure-Based Design of Microsomal Prostaglandin E2 Synthase-1 (mPGES-1) Inhibitors using a Virtual Fragment Growing Optimization Scheme CHEMMEDCHEM. Vol. 11. Pag.612-619 ISSN:1860-7179. | |
| Lauro, Gianluigi; Tortorella, Paolo; Bertamino, Alessia; Ostacolo, Carmine; Koeberle, Andreas; Fischer, Katrin; Bruno, Ines; Terracciano, Stefania; Gomez Monterrey, Isabel Maria; Tauro, Marilena; Loiodice, Fulvio; Novellino, Ettore; Riccio, Raffaele; Werz, Oliver; Campiglia, Pietro; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201500598 Codice identificativo ISI: WOS:000372990700007 Codice identificativo SCOPUS: 2-s2.0-84959387319 | |
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| 2015 | |
| Articolo in rivista | |
| 9H-purine scaffold reveals induced-fit pocket plasticity of the BRD9 bromodomain JOURNAL OF MEDICINAL CHEMISTRY. Vol. 58. Pag.2718-2736 ISSN:0022-2623. | |
| Picaud, Sarah; Strocchia, Maria; Terracciano, Stefania; Lauro, Gianluigi; Mendez, Jacqui; Daniels, Danette L; Riccio, Raffaele; Bifulco, Giuseppe; Bruno, Ines; Filippakopoulos, Panagis | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm501893k Codice identificativo ISI: WOS:000351971800009 Codice identificativo SCOPUS: 2-s2.0-84925938831 | |
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74065Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold
| 2015 | |
| Articolo in rivista | |
| Targeting the Hsp90 C-terminal domain by the chemically accessible dihydropyrimidinone scaffold CHEMICAL COMMUNICATIONS. Vol. 51. Pag.3850-3853 ISSN:1359-7345. | |
| Strocchia, Maria; Terracciano, Stefania; Chini, MARIA GIOVANNA; Vassallo, Antonio; Vaccaro, Maria C.; DAL PIAZ, Fabrizio; Leone, Antonietta; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1039/C4CC10074C Codice identificativo ISI: WOS:000349990600033 Codice identificativo SCOPUS: 2-s2.0-84923164308 | |
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| 2015 | |
| Articolo in rivista | |
| Identification of Lead Compounds as Inhibitors of STAT3: Design, Synthesis and Bioactivity MOLECULAR INFORMATICS. Vol. 34. Pag.689-697 ISSN:1868-1743. | |
| Botta, Antonio; Sirignano, Esther; Popolo, Ada; Saturnino, Carmela; Terracciano, Stefania; Foglia, Antonio; Sinicropi, Maria Stefania; Longo, Pasquale; DI MICCO, Simone | |
| Digital Object Identifier (DOI): 10.1002/minf.201500043 Codice identificativo ISI: WOS:000365319900004 Codice identificativo SCOPUS: 2-s2.0-84944354193 | |
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68732Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors
| 2015 | |
| Articolo in rivista | |
| Structural Insights for the Optimization of Dihydropyrimidin-2(1H)-one Based mPGES-1 Inhibitors ACS MEDICINAL CHEMISTRY LETTERS. Vol. 6. Pag.187-91-191 ISSN:1948-5875. | |
| Terracciano, Stefania; Lauro, Gianluigi; Strocchia, Maria; Fischer, Katrin; Werz, Oliver; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/ml500433j Codice identificativo ISI: WOS:000349652000015 Codice identificativo SCOPUS: 2-s2.0-84922936636 | |
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| 2015 | |
| Articolo in rivista | |
| Hsp90 Activity Modulation by Plant Secondary Metabolites PLANTA MEDICA. Vol. 81. Pag.1223-1239 ISSN:0032-0943. | |
| DAL PIAZ, Fabrizio; Terracciano, Stefania; DE TOMMASI, Nunziatina; Braca, Alessandra | |
| Digital Object Identifier (DOI): 10.1055/s-0035-1546251 Codice identificativo ISI: WOS:000361681000001 Codice identificativo SCOPUS: 2-s2.0-84942068020 | |
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| 2015 | |
| Articolo in rivista | |
| Can Small Chemical Modifications of Natural Pan-inhibitors Modulate the Biological Selectivity? the Case of Curcumin Prenylated Derivatives Acting as HDAC or mPGES-1 Inhibitors JOURNAL OF NATURAL PRODUCTS. Vol. 78. Pag.2867-2879 ISSN:0163-3864. | |
| Iranshahi, Mehrdad; Chini, MARIA GIOVANNA; Masullo, Milena; Sahebkar, Amirhossein; Javidnia, Azita; Chitsazian Yazdi, Mahsa; Pergola, Carlo; Koeberle, Andreas; Werz, Oliver; Pizza, Cosimo; Terracciano, Stefania; Piacente, Sonia; Bifulco, Giuseppe | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jnatprod.5b00700 Codice identificativo ISI: WOS:000367562600001 Codice identificativo SCOPUS: 2-s2.0-84953253869 | |
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| 2015 | |
| Contributo in Atti di convegno | |
| 40 th "A. Corbella" International Summer School on Organic Synthesis - ISOS 2015. In: LX Pag.58-58 | |
| 40 th " International Summer School on Organic Synthesis" Gargnano (BS) 14-18 giugno | |
| Foglia, Antonio; Di Micco, Simone; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Oppermann, Udo; Bifulco, Giuseppe; Bruno, Ines | |
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| 2015 | |
| Poster | |
| Targeting Microsomal Prostaglanding E2 Synthase 1 for the Development of new potential Anti-Inflammatory Drugs. In: Atti del Convegno Pag.196-196 | |
| XXXVI Convegno Nazionale della Divisione di Chimica Organica della Società Chimica Italiana Bologna 13-17 settembre 2015 | |
| Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
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| 2015 | |
| Poster | |
| Inhibition of Microsomal Prostaglandin E2 Synthase 1: focused design of new anti-inflammatory and anti-cancer drugs. In: Atti del Congresso Federico Bella and Domenico Spinelli Pag.126-126 | |
| SIGMA-ALDRICH Young Chemists Symposium Rimini dal 27 al 29 ottobre 2015 | |
| Foglia, Antonio; Terracciano, Stefania; Lauro, Gianluigi; Saturnino, Carmela; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
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| 2014 | |
| Articolo in rivista | |
| Exploration of the dihydropyrimidine scaffold for the development of new potential anti-inflammatory agents blocking prostaglandin E2 synthase-1 enzyme (mPGES-1) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 80. Pag.407-415 ISSN:0223-5234. | |
| Lauro, Gianluigi; Strocchia, Maria; Terracciano, Stefania; Bruno, Ines; Katrin, Fischer; Carlo, Pergola; Oliver, Werz; Riccio, Raffaele; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2014.04.061 Codice identificativo ISI: WOS:000337985400037 Codice identificativo SCOPUS: 2-s2.0-84899871048 | |
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| 2014 | |
| Contributo in Atti di convegno | |
| Design,virtual Screening and Synthesis of Potential Microsomal Prostaglandine E2 Synthase-1 (mPGES-1)Inhibitors. In: Atti del Congresso Cosenza uni Pag.354-354 | |
| XXV Congresso della Società Chimica Italiana Cosenza 7-12 settembre 2014 | |
| Foglia, Antonio; Simone Di, Micco; Terracciano, Stefania; Saturnino, Carmela; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
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56563Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors
| 2013 | |
| Articolo in rivista | |
| Dimeric and trimeric triazole based molecules as a new class of Hsp90 molecular chaperone inhibitors EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 65. Pag.464-476 ISSN:0223-5234. | |
| Terracciano, Stefania; Chini, MARIA GIOVANNA; DAL PIAZ, Fabrizio; Antonio, Vassallo; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2013.05.016 Codice identificativo ISI: WOS:000322850100045 Codice identificativo SCOPUS: 2-s2.0-84884272072 | |
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| 2013 | |
| Articolo in rivista | |
| Structural basis for the design and synthesis of selective HDAC inhibitors BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 21. Pag.3795-3807 ISSN:0968-0896. | |
| DI MICCO, Simone; Chini, MARIA GIOVANNA; Terracciano, Stefania; Bruno, Ines; Riccio, Raffaele; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2013.04.036 Codice identificativo ISI: WOS:000320347100018 Codice identificativo SCOPUS: 2-s2.0-84878551168 | |
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| 2012 | |
| Articolo in rivista | |
| Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors CHEMMEDCHEM. Vol. 7. Pag.694-702 ISSN:1860-7179. | |
| Terracciano, Stefania; Chini, MARIA GIOVANNA; Riccio, Raffaele; Bruno, Ines; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201100531 Codice identificativo ISI: WOS:000302073100017 Codice identificativo SCOPUS: 2-s2.0-84859181022 | |
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| 2010 | |
| Articolo in rivista | |
| Synthesis and biological activity of cyclotetrapeptide analogues of the natural HDAC inhibitor FR235222 BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 18. Pag.3252-3260 ISSN:0968-0896. | |
| Terracciano, Stefania; DI MICCO, Simone; Bifulco, Giuseppe; Gallinari, P; Riccio, Raffaele; Bruno, Ines | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2010.03.022 Codice identificativo ISI: WOS:000277083400027 Codice identificativo SCOPUS: 2-s2.0-77951207678 | |
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30296Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors
| 2010 | |
| Articolo in rivista | |
| Synthesis of new mono and bis amides projected as potential histone deacetylase (HDAC) inhibitors TETRAHEDRON. Vol. 66(13). Pag.2520-2528 ISSN:0040-4020. | |
| Terracciano, Stefania; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; E., Damico; Marzocco, Stefania; Riccio, Raffaele; Bruno, Ines | |
| Digital Object Identifier (DOI): 10.1016/j.tet.2010.01.061 Codice identificativo ISI: WOS:000275927100038 Codice identificativo SCOPUS: 2-s2.0-77349125579 | |
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| 2010 | |
| Articolo in rivista | |
| Conformationally locked calixarene-based histone deacetylase inhibitors ORGANIC LETTERS. Vol. 12. Pag.5382-5385 ISSN:1523-7060. | |
| Chini, MARIA GIOVANNA; Terracciano, Stefania; Riccio, Raffaele; Bifulco, Giuseppe; Ciao, Roberta; Gaeta, Carmine; Troisi, Francesco; Neri, Placido | |
| Digital Object Identifier (DOI): 10.1021/ol102420b Codice identificativo ISI: WOS:000284555600007 Codice identificativo SCOPUS: 2-s2.0-78650317971 | |
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| 2008 | |
| Articolo in rivista | |
| Effects of FR235222, a novel HDAC inhibitor, in proliferation and apoptosis of human leukaemia cell lines: role of annexin A1 EUROPEAN JOURNAL OF CANCER. Vol. 44. Pag.740-749 ISSN:0959-8049. | |
| Petrella, Antonello; D'Acunto, Cw; Rodriquez, Manuela; Festa, M; Tosco, Alessandra; Bruno, Ines; Terracciano, Stefania; Taddei, M; Paloma, Lg; Parente, Luca | |
| Digital Object Identifier (DOI): 10.1016/j.ejca.2008.01.023 Codice identificativo ISI: WOS:000255225200022 Codice identificativo SCOPUS: 2-s2.0-40849151859 | |
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| 2008 | |
| Articolo in rivista | |
| Synthetic and pharmacological studies on new simplified analogues of the potent actin-targeting Jaspamide BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 16. Pag.6580-6588 ISSN:1464-3391. | |
| Terracciano, Stefania; Bruno, Ines; Elisabetta, D’Amico; Bifulco, Giuseppe; Angela, Zampella; Valentina, Sepe; Charles D., Smith; Riccio, Raffaele | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2008.05.019 Codice identificativo SCOPUS: 2-s2.0-44849104388 | |
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| 2008 | |
| Articolo in rivista | |
| Molecular modeling studies toward the structural optimization of new cyclopeptide-based HDAC inhibitors modeled on the natural product FR235222 BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 2008. Pag.8635-8642 ISSN:0968-0896. | |
| DI MICCO, S; Terracciano, Stefania; Bruno, Ines; Rodriquez, Manuela; Riccio, Raffaele; Taddei, M; Bifulco, Giuseppe | |
| Digital Object Identifier (DOI): 10.1016/J.BMC.2008.08.003 Codice identificativo ISI: WOS:000259173400036 Codice identificativo SCOPUS: 2-s2.0-51549109903 | |
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17557Design and Synthesis of cyclopeptide analogues of the potent Histone deacetylase inhibitor FR235222
| 2007 | |
| Articolo in rivista | |
| Design and Synthesis of cyclopeptide analogues of the potent Histone deacetylase inhibitor FR235222 CHEMMEDCHEM. Vol. 2. Pag.1511-1519 ISSN:1860-7179. | |
| LUIGI GOMEZ, Paloma; Bruno, Ines; Elena, Cini; Saadi, Khochbin; Rodriquez, Manuela; Maurizio, Taddei; Terracciano, Stefania; AND KARIN, Sadoul | |
| Digital Object Identifier (DOI): 10.1002/cmdc.200700095 Codice identificativo ISI: WOS:000250283300012 Codice identificativo SCOPUS: 2-s2.0-41849109752 | |
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| 2006 | |
| Articolo in rivista | |
| Chemistry and biology of anti-inflammatory marine natural products: molecules interfering with cyclooxygenase, NF-κB and other unidentified targets CURRENT MEDICINAL CHEMISTRY. Vol. 13. Pag.1947-1969 ISSN:0929-8673. | |
| Terracciano, Stefania; Aquino, Maurizio; Rodriquez, Manuela; Monti, Maria Chiara; Casapullo, Agostino; Riccio, Raffaele; Gomez Paloma, Luigi | |
| Digital Object Identifier (DOI): 10.2174/092986706777585095 Codice identificativo ISI: WOS:000238674400008 Codice identificativo SCOPUS: 2-s2.0-33745761029 | |
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| 2006 | |
| Articolo in rivista | |
| Total Synthesis, NMR Solution Structure, and Binding Model of the Potent Histone Deacetylase Inhibitor FR235222 ANGEWANDTE CHEMIE. INTERNATIONAL EDITION. Vol. 45. Pag.423-427 ISSN:1433-7851. | |
| Rodriquez, Manuela; Terracciano, Stefania; E., Cini; G., Settembrini; Bruno, Ines; Bifulco, Giuseppe; M., Taddei; L., GOMEZ PALOMA | |
| Digital Object Identifier (DOI): 10.1002/anie.200501995 Codice identificativo ISI: WOS:000234604400013 Codice identificativo SCOPUS: 2-s2.0-30444433547 | |
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| 2005 | |
| Articolo in rivista | |
| Chemistry and Biology of Anti-Inflammatory Marine Natural Products.Phospholipase A2 Inhibitors CURRENT ORGANIC CHEMISTRY. Vol. 9. Pag.1419-1427 ISSN:1385-2728. | |
| Luigi Gomez, Paloma; Monti, Maria Chiara; Terracciano, Stefania; Casapullo, Agostino; Riccio, Raffaele | |
| Digital Object Identifier (DOI): 10.2174/1385272054880205 Codice identificativo ISI: WOS:000231377600004 Codice identificativo SCOPUS: 2-s2.0-23844478640 | |
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| 2005 | |
| Articolo in rivista | |
| Synthesis, solution structure, and bioactivity of six new simplified analogues of the natural cyclodepsipeptide jaspamide BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 13(17). Pag.5225-5239 ISSN:0968-0896. | |
| Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; E., Avallone; C. D., Smith; L., GOMEZ PALOMA; Riccio, Raffaele | |
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| 2005 | |
| Contributo in volume (Capitolo o Saggio) | |
| Critical Surveys Covering the Year 2004:Total Synthesis of Natural Products. In VARI Seminars in Organic Synthesis Pag.289-324 | |
| Bruno, Ines; P., Dambruoso; Terracciano, Stefania; Bifulco, Giuseppe | |
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| 2004 | |
| Articolo in rivista | |
| Synthesis, Conformational Analysis, and Cytotoxicity of New Analogues of the Natural Cyclodepsipeptide Jaspamide JOURNAL OF NATURAL PRODUCTS. Vol. 67(8). Pag.1325-1331 ISSN:0163-3864. | |
| Terracciano, Stefania; Bruno, Ines; Bifulco, Giuseppe; Copper Jean, E.; Smith Charles, D.; GOMEZ PALOMA, Luigi; Riccio, Raffaele | |
| Digital Object Identifier (DOI): 10.1021/np049955b Codice identificativo ISI: WOS:000223600200021 Codice identificativo SCOPUS: 2-s2.0-4344619554 | |
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