Sabrina CASTELLANO | Pubblicazioni
Sabrina CASTELLANO Pubblicazioni
| 2015 | |
| Abstract in Atti di convegno | |
| Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.37-37 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Li, Haitao; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Abstract in rivista | |
| Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) CHEMMEDCHEM. Vol. 10. Pag.2-2 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201490050 | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Abstract in rivista | |
| ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery CHEM INFORM. Vol. 46. Pag.no-no ISSN:0931-7597. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201520216 | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Articolo in rivista | |
| CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli PHYSIOLOGICAL RESEARCH. Vol. 64. Pag.769-782 ISSN:1802-9973. | |
| Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E. | |
| Versione online | |
| Codice identificativo ISI: WOS:000367154800019 Codice identificativo SCOPUS: 2-s2.0-84983200500 | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF CHEMMEDCHEM. Vol. 10. Pag.144-157 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201402371 Codice identificativo ISI: WOS:000346766700014 Codice identificativo SCOPUS: 2-s2.0-84919779703 | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Articolo in rivista | |
| A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 58. Pag.2779-2798 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm5019687 Codice identificativo ISI: WOS:000351971800013 Codice identificativo SCOPUS: 2-s2.0-84925957014 | |
| Visualizza sul Database dei Prodotti (IRIS) |
62075A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
| 2015 | |
| Articolo in rivista | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery RSC ADVANCES. Vol. 5. Pag.1268-1273 ISSN:2046-2069. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/C4RA13392G Codice identificativo ISI: WOS:000346079900051 Codice identificativo SCOPUS: 2-s2.0-84916613613 | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.248-248 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Discovery of new chemical probes for the MRG15 chromo domain.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.249-249 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.250-250 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.243-243 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.244-244 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.241-241 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.247-247 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
| 2015 | |
| Poster | |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.245-245 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Visualizza sul Database dei Prodotti (IRIS) |
149068A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
| 2015 | |
| Poster | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.239-239 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
| Visualizza sul Database dei Prodotti (IRIS) |
