Ciro MILITE | Publications

151199Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure

	2019
	Articolo in rivista
	Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.2666-2689 ISSN:0022-2623.
	Milite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca
	Versione online
	Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b02008 Codice identificativo ISI: WOS:000461537000030 Codice identificativo SCOPUS: 2-s2.0-85062555799
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351938Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases

	2019
	Articolo in rivista
	Benzothiopyranoindole- and pyridothiopyranoindole-based antiproliferative agents targeting topoisomerases EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 165. Pag.46-58 ISSN:0223-5234.
	Salerno, S.; La Pietra, V.; Hyeraci, M.; Taliani, S.; Robello, M.; Barresi, E.; Milite, C.; Simorini, F.; García-Argáez, A. N.; Marinelli, L.; Novellino, E.; Da Settimo, F.; Marini, A. M.; Dalla Via, L.
	Digital Object Identifier (DOI): 10.1016/j.ejmech.2019.01.015 Codice identificativo ISI: WOS:000459358600005 Codice identificativo SCOPUS: 2-s2.0-85060048556
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234018Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies

	2019
	Articolo in rivista
	Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. Vol. 34. Pag.1697-1710 ISSN:1475-6366.
	Milite, C.; Amendola, G.; Nocentini, A.; Bua, S.; Cipriano, A.; Barresi, E.; Feoli, A.; Novellino, E.; Da Settimo, F.; Supuran, C. T.; Castellano, S.; Cosconati, S.; Taliani, S.
	Digital Object Identifier (DOI): 10.1080/14756366.2019.1666836 Codice identificativo SCOPUS: 2-s2.0-85072371558
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