MONICA VIVIANO | Publications
MONICA VIVIANO Publications
| 2024 | |
| Articolo in rivista | |
| Successes and challenges in the development of BD1-selective BET inhibitors: a patent review EXPERT OPINION ON THERAPEUTIC PATENTS. Pag.1-17 ISSN:1354-3776. | |
| Viviano, Monica; Cipriano, Alessandra; Fabbrizi, Emanuele; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca; Mai, Antonello; Milite, Ciro; Rotili, Dante | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/13543776.2024.2327300 | |
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| 2024 | |
| Articolo in rivista | |
| Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors CHEMMEDCHEM. Vol. 19. Pag.e202400139(1)-e202400139(18) ISSN:1860-7187. | |
| Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Chini, Maria Giovanna; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202400139 Codice identificativo ISI: WOS:001253900000001 Codice identificativo SCOPUS: 2-s2.0-85196860902 | |
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| 2023 | |
| Articolo in rivista | |
| Indol-3-ylglyoxylamide as Privileged Scaffold in Medicinal Chemistry PHARMACEUTICALS. Vol. 16. Pag.1-43 ISSN:1424-8247. | |
| Barresi, Elisabetta; Robello, Marco; Baglini, Emma; Poggetti, Valeria; Viviano, Monica; Salerno, Silvia; Da Settimo, Federico; Taliani, Sabrina | |
| Digital Object Identifier (DOI): 10.3390/ph16070997 Codice identificativo ISI: WOS:001036636100001 Codice identificativo SCOPUS: 2-s2.0-85166252937 | |
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| 2023 | |
| Articolo in rivista | |
| NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 66. Pag.11632-11655 ISSN:0022-2623. | |
| Cipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c00770 Codice identificativo ISI: WOS:001060994300001 Codice identificativo SCOPUS: 2-s2.0-85171309414 | |
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| 2023 | |
| Articolo in rivista | |
| A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors ARCHIV DER PHARMAZIE. Pag.1-16 ISSN:0365-6233. | |
| Donati, Greta; Viviano, Monica; D'Amore, Vincenzo Maria; Cipriano, Alessandra; Diakogiannaki, Isidora; Amato, Jussara; Tomassi, Stefano; Brancaccio, Diego; Russomanno, Pasquale; Di Leva, Francesco Saverio; Arosio, Daniela; Seneci, Pierfausto; Taliani, Sabrina; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Skalniak, Lukasz; Holak, Tad A; Castellano, Sabrina; La Pietra, Valeria; Marinelli, Luciana | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/ardp.202300583 Codice identificativo ISI: WOS:001126478300001 Codice identificativo SCOPUS: 2-s2.0-85179959564 | |
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| 2023 | |
| Articolo in rivista | |
| Solubilizer Tag Effect on PD-L1/Inhibitor Binding Properties for m-Terphenyl Derivatives ACS MEDICINAL CHEMISTRY LETTERS. Vol. 15. Pag.36-44 ISSN:1948-5875. | |
| Surmiak, Ewa; Ząber, Julia; Plewka, Jacek; Wojtanowicz, Grzegorz; Kocik-Krol, Justyna; Kruc, Oskar; Muszak, Damian; Rodríguez, Ismael; Musielak, Bogdan; Viviano, Monica; Castellano, Sabrina; Skalniak, Lukasz; Magiera-Mularz, Katarzyna; Holak, Tad A.; Kalinowska-Tłuścik, Justyna | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acsmedchemlett.3c00306 Codice identificativo ISI: WOS:001141732600001 Codice identificativo SCOPUS: 2-s2.0-85181143388 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor JOURNAL OF MEDICINAL CHEMISTRY. Pag.13665-13683 ISSN:0022-2623. | |
| Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c01030 Codice identificativo ISI: WOS:001045914800001 Codice identificativo SCOPUS: 2-s2.0-85168362422 | |
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| 2022 | |
| Articolo in rivista | |
| Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain CHEMMEDCHEM. Vol. 17. Pag.1-14 ISSN:1860-7179. | |
| Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202200343 Codice identificativo ISI: WOS:000853917200001 Codice identificativo SCOPUS: 2-s2.0-85138079605 | |
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| 2022 | |
| Articolo in rivista | |
| Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 237. Pag.114410-114440 ISSN:0223-5234. | |
| Menna, Martina; Fiorentino, Francesco; Marrocco, Biagina; Lucidi, Alessia; Tomassi, Stefano; Cilli, Domenica; Romanenghi, Mauro; Cassandri, Matteo; Pomella, Silvia; Pezzella, Michele; Del Bufalo, Donatella; Zeya Ansari, Mohammad Salik; Tomašević, Nevena; Mladenović, Milan; Viviano, Monica; Sbardella, Gianluca; Rota, Rossella; Trisciuoglio, Daniela; Minucci, Saverio; Mattevi, Andrea; Rotili, Dante; Mai, Antonello | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.114410 Codice identificativo ISI: WOS:000804176200002 Codice identificativo SCOPUS: 2-s2.0-85129352278 | |
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| 2022 | |
| Articolo in rivista | |
| Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 65. Pag.11574-11606 ISSN:0022-2623. | |
| Iannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.2c00252 Codice identificativo ISI: WOS:000822512300001 Codice identificativo SCOPUS: 2-s2.0-85129915280 | |
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| 2022 | |
| Articolo in rivista | |
| Lysine methyltransferase inhibitors: where we are now. RSC CHEMICAL BIOLOGY. Vol. 3. Pag.359-406 ISSN:2633-0679. | |
| Feoli, Alessandra; Viviano, Monica; Cipriano, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/D1CB00196E Codice identificativo ISI: WOS:000739939100001 Codice identificativo SCOPUS: 2-s2.0-85129384483 | |
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| 2022 | |
| Articolo in rivista | |
| Essential Principles and Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging CURRENT MEDICINAL CHEMISTRY. Vol. 29. Pag.4862-4890 ISSN:0929-8673. | |
| Viviano, Monica; Barresi, Elisabetta; Siméon, Fabrice G.; Costa, Barbara; Taliani, Sabrina; Da Settimo, Federico; Pike, Victor W.; Castellano, Sabrina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.2174/0929867329666220329204054 Codice identificativo ISI: WOS:000842480000006 Codice identificativo SCOPUS: 2-s2.0-85134206342 | |
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| 2022 | |
| Articolo in rivista | |
| Microwave-Assisted Aminoalkylation of Phenols via Mustard Carbonate Analogues SYNTHESIS. Pag.1-9 ISSN:0039-7881. | |
| Viviano, M.; Trapasso, G.; Annatelli, M.; Milite, C.; Castellano, S.; Arico, F. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1055/a-1742-3723 Codice identificativo ISI: WOS:000796080700010 Codice identificativo SCOPUS: 2-s2.0-85124520145 | |
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| 2021 | |
| Articolo in rivista | |
| Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 SLAS DISCOVERY. Vol. 26. Pag.77-87 ISSN:2472-5552. | |
| Feoli, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Castellano, Sabrina; Bartoschik, Tanja; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1177/2472555220949166 Codice identificativo ISI: WOS:000560777300001 Codice identificativo SCOPUS: 2-s2.0-85089488195 | |
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| 2021 | |
| Articolo in rivista | |
| Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 220. Pag.1-11 ISSN:0223-5234. | |
| Salerno, Silvia; Amendola, Giorgio; Angeli, Andrea; Baglini, Emma; Barresi, Elisabetta; Marini, Anna Maria; Ravichandran, Rahul; Viviano, Monica; Castellano, Sabrina; Novellino, Ettore; Da Settimo, Federico; Supuran, Claudiu T.; Cosconati, Sandro; Taliani, Sabrina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2021.113490 Codice identificativo ISI: WOS:000659148800033 Codice identificativo SCOPUS: 2-s2.0-85107137276 | |
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| 2021 | |
| Articolo in rivista | |
| Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. Vol. 36. Pag.1874-1883 ISSN:1475-6366. | |
| Baglini, Emma; Ravichandran, Rahul; Berrino, Eanuela; Salerno, Silvia; Barresi, Elisabetta; Marini, Anna Maria; Viviano, Monica; Castellano, Sabrina; Da Settimo, Federico; Supuran, Claudiu T.; Cosconati, Sandro; Taliani, Sabrina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/14756366.2021.1956913 Codice identificativo ISI: WOS:000680671600001 Codice identificativo SCOPUS: 2-s2.0-85111987663 | |
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| 2019 | |
| Articolo in rivista | |
| Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.2666-2689 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b02008 Codice identificativo ISI: WOS:000461537000030 Codice identificativo SCOPUS: 2-s2.0-85062555799 | |
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| 2019 | |
| Articolo in rivista | |
| Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 163. Pag.722-735 ISSN:0223-5234. | |
| Stazi, Giulia; Battistelli, Cecilia; Piano, Valentina; Mazzone, Roberta; Marrocco, Biagina; Marchese, Sara; Louie, Sharon M.; Zwergel, Clemens; Antonini, Lorenzo; Patsilinakos, Alexandros; Ragno, Rino; Viviano, Monica; Sbardella, Gianluca; Ciogli, Alessia; Fabrizi, Giancarlo; Cirilli, Roberto; Strippoli, Raffaele; Marchetti, Alessandra; Tripodi, Marco; Nomura, Daniel K.; Mattevi, Andrea; Mai, Antonello; Valente, Sergio | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2018.11.050 Codice identificativo ISI: WOS:000458597300053 Codice identificativo SCOPUS: 2-s2.0-85058530369 | |
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| 2017 | |
| Articolo in rivista | |
| Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) JOURNAL OF MEDICINAL CHEMISTRY. Vol. 60. Pag.7897-7909 ISSN:0022-2623. | |
| Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.7b01031 Codice identificativo ISI: WOS:000412150300017 Codice identificativo SCOPUS: 2-s2.0-85030253369 | |
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| 2017 | |
| Articolo in rivista | |
| Developing Spindlin1 small-molecule inhibitors by using protein microarrays NATURE CHEMICAL BIOLOGY. Vol. 13. Pag.750-756 ISSN:1552-4450. | |
| Bae, Narkhyun; Viviano, Monica; Su, Xiaonan; Lv, Jie; Cheng, Donghang; Sagum, Cari; Castellano, Sabrina; Bai, Xue; Johnson, Claire; Khalil, Mahmoud Ibrahim; Shen, Jianjun; Chen, Kaifu; Li, Haitao; Sbardella, Gianluca; Bedford, Mark T. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/nchembio.2377 Codice identificativo ISI: WOS:000403673700011 Codice identificativo SCOPUS: 2-s2.0-85021067771 | |
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| 2017 | |
| Poster | |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.67-67 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
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| 2016 | |
| Abstract in rivista | |
| ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors CHEM INFORM. Vol. 47. Pag.1-1 ISSN:0931-7597. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201642266 | |
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| 2016 | |
| Articolo in rivista | |
| The emerging role of lysine methyltransferase SETD8 in human diseases CLINICAL EPIGENETICS. Vol. 8. Pag.1-15 ISSN:1868-7083. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1186/s13148-016-0268-4 Codice identificativo ISI: WOS:000384471400001 Codice identificativo SCOPUS: 2-s2.0-84994805952 | |
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| 2016 | |
| Articolo in rivista | |
| Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors CHEMMEDCHEM. Vol. 11. Pag.1680-1685 ISSN:1860-7179. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201600272 Codice identificativo ISI: WOS:000383579700002 Codice identificativo SCOPUS: 2-s2.0-84983335802 | |
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149157DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
| 2016 | |
| Poster | |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH. In: XXIV NMMC & 10th NPCF - September 11th-14th 2016, Perugia (Italy) - Book of Abstract Pag.207-207 | |
| XXIV NMMC & 10th NPCF Perugia 11-14 Settembre 2016 | |
| Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
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| 2015 | |
| Abstract in Atti di convegno | |
| Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.37-37 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Li, Haitao; Sbardella, Gianluca | |
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| 2015 | |
| Abstract in rivista | |
| Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) CHEMMEDCHEM. Vol. 10. Pag.2-2 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201490050 | |
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| 2015 | |
| Abstract in rivista | |
| ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery CHEM INFORM. Vol. 46. Pag.no-no ISSN:0931-7597. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201520216 | |
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| 2015 | |
| Articolo in rivista | |
| Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF CHEMMEDCHEM. Vol. 10. Pag.144-157 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201402371 Codice identificativo ISI: WOS:000346766700014 Codice identificativo SCOPUS: 2-s2.0-84919779703 | |
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62075A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
| 2015 | |
| Articolo in rivista | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery RSC ADVANCES. Vol. 5. Pag.1268-1273 ISSN:2046-2069. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/C4RA13392G Codice identificativo ISI: WOS:000346079900051 Codice identificativo SCOPUS: 2-s2.0-84916613613 | |
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| 2015 | |
| Poster | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.250-250 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
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| 2015 | |
| Poster | |
| Discovery of new chemical probes for the MRG15 chromo domain.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.249-249 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.248-248 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
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| 2015 | |
| Poster | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.244-244 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
149068A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
| 2015 | |
| Poster | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.239-239 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
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| 2014 | |
| Articolo in rivista | |
| Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 57. Pag.2413-2428 ISSN:0022-2623. | |
| Castellano, Sabrina; Sabrina, Taliani; Viviano, Monica; Milite, Ciro; Eleonora Da, Pozzo; Barbara, Costa; Elisabetta, Barresi; Agostino, Bruno; Sandro, Cosconati; Luciana, Marinelli; Giovanni, Greco; Ettore, Novellino; Sbardella, Gianluca; Federico Da, Settimo; Claudia, Martini | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm401721h Codice identificativo ISI: WOS:000333578400017 Codice identificativo SCOPUS: 2-s2.0-84897411408 | |
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| 2012 | |
| Articolo in rivista | |
| Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.9875-9890 ISSN:0022-2623. | |
| Castellano, Sabrina; Spannhoff, Astrid; Milite, Ciro; DAL PIAZ, Fabrizio; Cheng, Donghang; Tosco, Alessandra; Viviano, Monica; Yamani, Abdellah; Cianciulli, Agostino; Sala, Marina; Cura, Vincent; Cavarelli, Jean; Novellino, Ettore; Mai, Antonello; Bedford, Mark T.; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm301097p Codice identificativo ISI: WOS:000311461500040 Codice identificativo SCOPUS: 2-s2.0-84869995779 | |
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| 2012 | |
| Articolo in rivista | |
| Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions RSC ADVANCES. Vol. 2. Pag.5229-5233 ISSN:2046-2069. | |
| Milite, Ciro; Viviano, Monica; Marisabella, Santoriello; Fabio, Arico`; Sbardella, Gianluca; Castellano, Sabrina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c2ra20275a Codice identificativo ISI: WOS:000304487000043 Codice identificativo SCOPUS: 2-s2.0-84893259222 | |
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| 2011 | |
| Articolo in rivista | |
| Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54. Pag.7663-7677 ISSN:0022-2623. | |
| Castellano, Sabrina; Dirk, Kuck; Viviano, Monica; Jakyung, Yoo; Fabian López, Vallejo; Paola, Conti; Lucia, Tamborini; Andrea, Pinto; José L., Medina Franco; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm2010404 Codice identificativo ISI: WOS:000296408100020 Codice identificativo SCOPUS: 2-s2.0-80455173681 | |
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| 2010 | |
| Articolo in rivista | |
| Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. JOURNAL OF ORGANIC CHEMISTRY. Vol. 75. Pag.7439-7442 ISSN:0022-3263. | |
| Castellano, Sabrina; Lucia, Tamborini; Viviano, Monica; Andrea, Pinto; Sbardella, Gianluca; Paola, Conti | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jo1014323 Codice identificativo ISI: WOS:000283531100051 Codice identificativo SCOPUS: 2-s2.0-78049513527 | |
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