Publications

Giacomo PEPE Publications


2019
Articolo in rivista
Yield parameters and antioxidant compounds of tomato fruit: the role of plant defence inducers with or without Cucumber mosaic virus infection
JOURNAL OF THE SCIENCE OF FOOD AND AGRICULTURE. Vol. 99. Pag.5541-5549
ISSN:0022-5142.
Rendina, Nunzia; Nuzzaci, Maria; Sofo, Adriano; Campiglia, Pietro; Scopa, Antonio; Sommella, EDUARDO MARIA; Pepe, Giacomo; De Nisco, Mauro; Basilicata, MANUELA GIOVANNA; Manfra, Michele
Digital Object Identifier (DOI): 10.1002/jsfa.9818
Codice identificativo ISI: WOS:000473952600001
Codice identificativo SCOPUS: 2-s2.0-85068609845
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2019
Articolo in rivista
Design, Synthesis, and Biological Evaluation of New 1-(Aryl-1 H-pyrrolyl)(phenyl)methyl-1 H-imidazole Derivatives as Antiprotozoal Agents
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.1330-1347
ISSN:0022-2623.
Saccoliti, Francesco; Noemi Madia, Valentina; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Calvet, Claudia M.; Jennings, Gareth K.; Podust, Larissa M.; Pepe, Giacomo; Cirilli, Roberto; Faggi, Cristina; Di Marco, Annalise; Rosaria Battista, Maria; Summa, Vincenzo; Cost, Roberta; Di Santo, Iroberto
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b01464
Codice identificativo ISI: WOS:000459223600016
Codice identificativo SCOPUS: 2-s2.0-85061636363
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2019
Articolo in rivista
β -Lactoglobulin Heptapeptide Reduces Oxidative Stress in Intestinal Epithelial Cells and Angiotensin II-Induced Vasoconstriction on Mouse Mesenteric Arteries by Induction of Nuclear Factor Erythroid 2-Related Factor 2 (Nrf2) Translocation
OXIDATIVE MEDICINE AND CELLULAR LONGEVITY. Vol. 2019. Pag.1616239-1616251
ISSN:1942-0900.
Pepe, G.; Basilicata, M. G.; Carrizzo, A.; Adesso, S.; Ostacolo, C.; Sala, M.; Sommella, E.; Ruocco, M.; Cascioferro, S.; Ambrosio, M.; Pisanti, S.; Di Sarno, V.; Bertamino, A.; Marzocco, S.; Vecchione, C.; Campiglia, P.
Digital Object Identifier (DOI): 10.1155/2019/1616239
Codice identificativo ISI: WOS:000499163800003
Codice identificativo SCOPUS: 2-s2.0-85075669961
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2019
Articolo in rivista
Anti-inflammatory and antioxidant properties of dehydrated potato-derived bioactive compounds in intestinal cells
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. Vol. 20. Pag.6087-6101
ISSN:1661-6596.
Basilicata, M. G.; Pepe, G.; Rapa, S. F.; Merciai, F.; Ostacolo, C.; Manfra, M.; Sarno, V.; Autore, G.; de Vita, D.; Marzocco, S.; Campiglia, P.
Versione online
Digital Object Identifier (DOI): 10.3390/ijms20236087
Codice identificativo ISI: WOS:000504428300269
Codice identificativo SCOPUS: 2-s2.0-85076174100
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2019
Articolo in rivista
Identification of an indol-based multi-target kinase inhibitor through phenotype screening and target fishing using inverse virtual screening approach
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 167. Pag.61-75
ISSN:0223-5234.
Ostacolo, Carmine; Di Sarno, Veronica; Lauro, Gianluigi; Pepe, Giacomo; Musella, Simona; Ciaglia, Tania; Vestuto, Vincenzo; Autore, Giuseppina; Bifulco, Giuseppe; Marzocco, Stefania; Campiglia, Pietro; Gomez-Monterrey, Isabel M; Bertamino, Alessia
Digital Object Identifier (DOI): 10.1016/j.ejmech.2019.01.066
Codice identificativo ISI: WOS:000461728400005
Codice identificativo SCOPUS: 2-s2.0-85061236063
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2019
Articolo in rivista
An Efficient Approach to Aromatic Aminomethylation Using Dichloromethane as Methylene Source
FRONTIERS IN CHEMISTRY. Vol. 7. Pag.1-10
ISSN:2296-2646.
Ostacolo, Carmine; DI SARNO, Veronica; Musella, Simona; Ciaglia, Tania; Vestuto, Vincenzo; Pepe, Giacomo; Merciai, Fabrizio; Campiglia, Pietro; Monterrey Isabel M., Gomez; Bertamino, Alessia
Digital Object Identifier (DOI): 10.3389/fchem.2019.00568
Codice identificativo ISI: WOS:000480523500002
Codice identificativo SCOPUS: 2-s2.0-85072734877
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2019
Articolo in rivista
Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.2666-2689
ISSN:0022-2623.
Milite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca
Versione online
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b02008
Codice identificativo ISI: WOS:000461537000030
Codice identificativo SCOPUS: 2-s2.0-85062555799
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