ALESSANDRA CIPRIANO | Publications
ALESSANDRA CIPRIANO Publications
| 2024 | |
| Articolo in rivista | |
| Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors CHEMMEDCHEM. Vol. 19. Pag.e202400139(1)-e202400139(18) ISSN:1860-7187. | |
| Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Chini, Maria Giovanna; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202400139 Codice identificativo ISI: WOS:001253900000001 Codice identificativo SCOPUS: 2-s2.0-85196860902 | |
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| 2024 | |
| Articolo in rivista | |
| Successes and challenges in the development of BD1-selective BET inhibitors: a patent review EXPERT OPINION ON THERAPEUTIC PATENTS. Pag.1-17 ISSN:1354-3776. | |
| Viviano, Monica; Cipriano, Alessandra; Fabbrizi, Emanuele; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca; Mai, Antonello; Milite, Ciro; Rotili, Dante | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/13543776.2024.2327300 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor JOURNAL OF MEDICINAL CHEMISTRY. Pag.13665-13683 ISSN:0022-2623. | |
| Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c01030 Codice identificativo ISI: WOS:001045914800001 Codice identificativo SCOPUS: 2-s2.0-85168362422 | |
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| 2023 | |
| Articolo in rivista | |
| A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors ARCHIV DER PHARMAZIE. Pag.1-16 ISSN:0365-6233. | |
| Donati, Greta; Viviano, Monica; D'Amore, Vincenzo Maria; Cipriano, Alessandra; Diakogiannaki, Isidora; Amato, Jussara; Tomassi, Stefano; Brancaccio, Diego; Russomanno, Pasquale; Di Leva, Francesco Saverio; Arosio, Daniela; Seneci, Pierfausto; Taliani, Sabrina; Magiera-Mularz, Katarzyna; Musielak, Bogdan; Skalniak, Lukasz; Holak, Tad A; Castellano, Sabrina; La Pietra, Valeria; Marinelli, Luciana | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/ardp.202300583 Codice identificativo ISI: WOS:001126478300001 Codice identificativo SCOPUS: 2-s2.0-85179959564 | |
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| 2023 | |
| Articolo in rivista | |
| NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 66. Pag.11632-11655 ISSN:0022-2623. | |
| Cipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c00770 Codice identificativo ISI: WOS:001060994300001 Codice identificativo SCOPUS: 2-s2.0-85171309414 | |
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| 2022 | |
| Articolo in rivista | |
| Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 65. Pag.11574-11606 ISSN:0022-2623. | |
| Iannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.2c00252 Codice identificativo ISI: WOS:000822512300001 Codice identificativo SCOPUS: 2-s2.0-85129915280 | |
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| 2022 | |
| Articolo in rivista | |
| Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain CHEMMEDCHEM. Vol. 17. Pag.1-14 ISSN:1860-7179. | |
| Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202200343 Codice identificativo ISI: WOS:000853917200001 Codice identificativo SCOPUS: 2-s2.0-85138079605 | |
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| 2022 | |
| Articolo in rivista | |
| Lysine methyltransferase inhibitors: where we are now. RSC CHEMICAL BIOLOGY. Vol. 3. Pag.359-406 ISSN:2633-0679. | |
| Feoli, Alessandra; Viviano, Monica; Cipriano, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/D1CB00196E Codice identificativo ISI: WOS:000739939100001 Codice identificativo SCOPUS: 2-s2.0-85129384483 | |
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| 2020 | |
| Articolo in rivista | |
| Targeting epigenetic reader domains by chemical biology CURRENT OPINION IN CHEMICAL BIOLOGY. Vol. 57. Pag.82-94 ISSN:1367-5931. | |
| Cipriano, Alessandra; Sbardella, Gianluca; Ciulli, Alessio | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.cbpa.2020.05.006 Codice identificativo ISI: WOS:000568781700013 Codice identificativo SCOPUS: 2-s2.0-85088795636 | |
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| 2019 | |
| Articolo in rivista | |
| Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. Vol. 34. Pag.1697-1710 ISSN:1475-6366. | |
| Milite, C.; Amendola, G.; Nocentini, A.; Bua, S.; Cipriano, A.; Barresi, E.; Feoli, A.; Novellino, E.; Da Settimo, F.; Supuran, C. T.; Castellano, S.; Cosconati, S.; Taliani, S. | |
| Digital Object Identifier (DOI): 10.1080/14756366.2019.1666836 Codice identificativo SCOPUS: 2-s2.0-85072371558 | |
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| 2019 | |
| Articolo in rivista | |
| Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.2666-2689 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b02008 Codice identificativo ISI: WOS:000461537000030 Codice identificativo SCOPUS: 2-s2.0-85062555799 | |
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| 2017 | |
| Poster | |
| Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.52-52 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca | |
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