Carmine OSTACOLO | Publications
Carmine OSTACOLO Publications
2025 | |
Articolo in rivista | |
The fast-dissociating D2 antagonist antipsychotic JNJ-37822681 is a neuronal Kv7 channel opener: Potential repurposing for epilepsy treatment BRITISH JOURNAL OF PHARMACOLOGY. Pag.1-22 ISSN:1476-5381. | |
Carotenuto, Lidia; Keminer, Oliver; Carleo, Giusy; Zaliani, Andrea; Leo, Antonio; Citraro, Rita; De Sarro, Giovambattista; Dirkx, Nina; Kaji, Marcus; Weckhuysen, Sarah; Reinshagen, Jeanette; Barrese, Vincenzo; Guida, Natascia; Ostacolo, Carmine; Miceli, Francesco; Gribbon, Philip; Taglialatela, Maurizio | |
Digital Object Identifier (DOI): 10.1111/bph.70119 | |
Show it in Product Database (IRIS) |
2025 | |
Articolo in rivista | |
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization CHEMMEDCHEM. Pag.1-20 ISSN:1860-7179. | |
Smaldone, Gerardina; Miranda, Maria Rosaria; Di Matteo, Francesca; Napolitano, Valeria; Aliberti, Michela; Musella, Simona; Di Sarno, Veronica; Lauro, Gianluigi; Bifulco, Giuseppe; Pepe, Giacomo; Aquino, Giovanna; Tecce, Mario Felice; Gomez-Monterrey, Isabel Maria; Campiglia, Pietro; Ostacolo, Carmine; Bertamino, Alessia; Vestuto, Vincenzo; Ciaglia, Tania | |
Digital Object Identifier (DOI): 10.1002/cmdc.202500247 Codice identificativo SCOPUS: 2-s2.0-105006916560 | |
Show it in Product Database (IRIS) |
2025 | |
Articolo in rivista | |
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 289. Pag.1-16 ISSN:0223-5234. | |
Lauro, Gianluigi; Aliberti, Michela; De Nisco, Mauro; Pedatella, Silvana; Pepe, Giacomo; Basilicata, Manuela Giovanna; Chini, Maria Giovanna; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Saviano, Anella; Campiglia, Pietro; Bertamino, Alessia; Ostacolo, Carmine; Ciaglia, Tania; Manfra, Michele; Bifulco, Giuseppe | |
Versione online | |
Digital Object Identifier (DOI): 10.1016/j.ejmech.2025.117402 Codice identificativo SCOPUS: 2-s2.0-85218871040 | |
Show it in Product Database (IRIS) |
2025 | |
Articolo in rivista | |
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution JOURNAL OF MEDICINAL CHEMISTRY. Vol. 68. Pag.16483-16517 ISSN:0022-2623. | |
Ciaglia, T.; Napolitano, V.; Miranda, M. R.; La Gioia, D.; Musella, S.; Schiano Moriello, A.; Merciai, F.; Di Sarno, V.; De Vita, S.; Colarusso, E.; Smaldone, G.; Di Matteo, F.; Sommella, E. M.; Kumar, P.; Allarà, M.; Ligresti, A.; Gomez-Monterrey, I. M.; Bifulco, G.; Lauro, G.; Campiglia, P.; Ostacolo, C.; Vestuto, V.; Bertamino, A. | |
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.5c01344 Codice identificativo ISI: WOS:001535143300001 Codice identificativo SCOPUS: 2-s2.0-105013572710 | |
Show it in Product Database (IRIS) |
2025 | |
Poster | |
In silico-assisted design of selective KCNT1 blocker: toward new epilepsy therapies. In: 8th RSC-BMCS/ SCI Symposium on Ion Channels as Therapeutic Targets Pag.1-1 | |
Turcio, Rita; Iraci, Nunzio; Carotenuto, Lidia; Ambrosino, Paolo; Pepe, Giacomo; Virginia Soldovieri, Maria; Campiglia, Pietro; Miceli, Francesco; Bertamino, Alessia; Taglialatela, Maurizio; Ostacolo, Carmine | |
Show it in Product Database (IRIS) |