Publications

Carmine OSTACOLO Publications


2025
Articolo in rivista
The fast-dissociating D2 antagonist antipsychotic JNJ-37822681 is a neuronal Kv7 channel opener: Potential repurposing for epilepsy treatment
BRITISH JOURNAL OF PHARMACOLOGY. Pag.1-22
ISSN:1476-5381.
Carotenuto, Lidia; Keminer, Oliver; Carleo, Giusy; Zaliani, Andrea; Leo, Antonio; Citraro, Rita; De Sarro, Giovambattista; Dirkx, Nina; Kaji, Marcus; Weckhuysen, Sarah; Reinshagen, Jeanette; Barrese, Vincenzo; Guida, Natascia; Ostacolo, Carmine; Miceli, Francesco; Gribbon, Philip; Taglialatela, Maurizio
Digital Object Identifier (DOI): 10.1111/bph.70119
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2025
Articolo in rivista
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibition
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 289. Pag.1-16
ISSN:0223-5234.
Lauro, Gianluigi; Aliberti, Michela; De Nisco, Mauro; Pedatella, Silvana; Pepe, Giacomo; Basilicata, Manuela Giovanna; Chini, Maria Giovanna; Fischer, Katrin; Hofstetter, Robert K.; Werz, Oliver; Ferraro, Maria Grazia; Piccolo, Marialuisa; Irace, Carlo; Saviano, Anella; Campiglia, Pietro; Bertamino, Alessia; Ostacolo, Carmine; Ciaglia, Tania; Manfra, Michele; Bifulco, Giuseppe
Versione online
Digital Object Identifier (DOI): 10.1016/j.ejmech.2025.117402
Codice identificativo SCOPUS: 2-s2.0-85218871040
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2025
Articolo in rivista
Untargeted Diversity-Oriented Synthesis for the Discovery of New Antitumor Agents: An Integrated Approach of Inverse Virtual Screening, Bioinformatics, and Omics for Target Deconvolution
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 68. Pag.16483-16517
ISSN:0022-2623.
Ciaglia, T.; Napolitano, V.; Miranda, M. R.; La Gioia, D.; Musella, S.; Schiano Moriello, A.; Merciai, F.; Di Sarno, V.; De Vita, S.; Colarusso, E.; Smaldone, G.; Di Matteo, F.; Sommella, E. M.; Kumar, P.; Allarà, M.; Ligresti, A.; Gomez-Monterrey, I. M.; Bifulco, G.; Lauro, G.; Campiglia, P.; Ostacolo, C.; Vestuto, V.; Bertamino, A.
Digital Object Identifier (DOI): 10.1021/acs.jmedchem.5c01344
Codice identificativo ISI: WOS:001535143300001
Codice identificativo SCOPUS: 2-s2.0-105013572710
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2025
Articolo in rivista
Novel para‐phenylenediamine‐based derivatives as Receptor Tyrosine Kinase‐like Orphan Receptor 1 (ROR1) Inhibitors: An in vitro preliminary characterization
CHEMMEDCHEM. Pag.1-20
ISSN:1860-7179.
Smaldone, Gerardina; Miranda, Maria Rosaria; Di Matteo, Francesca; Napolitano, Valeria; Aliberti, Michela; Musella, Simona; Di Sarno, Veronica; Lauro, Gianluigi; Bifulco, Giuseppe; Pepe, Giacomo; Aquino, Giovanna; Tecce, Mario Felice; Gomez-Monterrey, Isabel Maria; Campiglia, Pietro; Ostacolo, Carmine; Bertamino, Alessia; Vestuto, Vincenzo; Ciaglia, Tania
Digital Object Identifier (DOI): 10.1002/cmdc.202500247
Codice identificativo SCOPUS: 2-s2.0-105006916560
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