Gianluca SBARDELLA | Publications
Gianluca SBARDELLA Publications
| 2015 | |
| Abstract in Atti di convegno | |
| Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.37-37 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Li, Haitao; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Abstract in rivista | |
| Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) CHEMMEDCHEM. Vol. 10. Pag.2-2 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201490050 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Abstract in rivista | |
| ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery CHEM INFORM. Vol. 46. Pag.no-no ISSN:0931-7597. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201520216 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli PHYSIOLOGICAL RESEARCH. Vol. 64. Pag.769-782 ISSN:1802-9973. | |
| Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E. | |
| Versione online | |
| Codice identificativo ISI: WOS:000367154800019 Codice identificativo SCOPUS: 2-s2.0-84983200500 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 58. Pag.2779-2798 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm5019687 Codice identificativo ISI: WOS:000351971800013 Codice identificativo SCOPUS: 2-s2.0-84925957014 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF CHEMMEDCHEM. Vol. 10. Pag.144-157 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201402371 Codice identificativo ISI: WOS:000346766700014 Codice identificativo SCOPUS: 2-s2.0-84919779703 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells FOLIA BIOLOGICA. Vol. 61. Pag.49-59 ISSN:0015-5500. | |
| Legartová, Soňa; Sbardella, Gianluca; Kozubek, Stanislav; Bártová, Eva | |
| Versione online | |
| Codice identificativo ISI: WOS:000355375900001 Codice identificativo SCOPUS: 2-s2.0-84930704221 | |
| Show it in Product Database (IRIS) |
62075A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
| 2015 | |
| Articolo in rivista | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery RSC ADVANCES. Vol. 5. Pag.1268-1273 ISSN:2046-2069. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/C4RA13392G Codice identificativo ISI: WOS:000346079900051 Codice identificativo SCOPUS: 2-s2.0-84916613613 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in Atti di convegno | |
| STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA. In: Abstracts from the 3rd Biennial Conference on Pediatric Neuro-Oncology Basic and Translational Research Oxford, UK Oxford University Press Vol.17, Pag.8-8 | |
| 3rd Biennial Conference on Pediatric Neuro-Oncology Basic and Translational Research San Diego, CA 7-9 maggio 2015 | |
| Hatcher, R.; Das, C.; Fangusaro, J.; Rajaram, V.; Lulla, R.; Goldman, S.; Khatua, S.; Sbardella, Gianluca; Gopalakrishnan, V. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1093/neuonc/nov061.29 Codice identificativo ISI: WOS:000361304800030 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in volume (Capitolo o Saggio) | |
| Chemioterapici antiprotozoari. In Alberto Gasco,Fulvio Gualtieri,Carlo Melchiorre Chimica farmaceutica Pag.832-852 Bologna Zanichelli Editore spa. ISBN:9788808187123 | |
| Sbardella, Gianluca | |
| Digital Object Identifier (DOI): 10.978.8808/187123 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in volume (Capitolo o Saggio) | |
| Agenti antimicotici, antimicobatterici e antiprotozoari. In Maria Laura Bolognesi, Paola Conti, Gabriele Costantino, Gloria Cristalli, Roberta Fruttero, Loretta Lazzarato, Giovanni Lentini, Marco Macchia, Antonio Macchiarulo, Antonello Mai, Clementina Manera, Gabriella Marucci, Filippo Minutolo, Marco Mor, Gianluca Sbardella, Rosaria Volpini Chimica Farmaceutica di Graham L. Patrick Pag.589-636 Napoli EdiSES. ISBN:9788879598453 | |
| Costantino, Gabriele; Mai, Antonello; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.248-248 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Discovery of new chemical probes for the MRG15 chromo domain.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.249-249 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.250-250 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.244-244 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.241-241 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
149068A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
| 2015 | |
| Poster | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.239-239 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.247-247 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.245-245 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.243-243 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
