Gianluca SBARDELLA | Publications
Gianluca SBARDELLA Publications
| 2024 | |
| Articolo in rivista | |
| The Lysine Acetyltransferase PCAF Functionally Interacts with Estrogen Receptor Alpha in the Hippocampus of Gonadally Intact Male - but not Female - Rats to Enhance Short-term Memory THE JOURNAL OF NEUROSCIENCE. Vol. 44. Pag.e1574232024-e1574232024 ISSN:0270-6474. | |
| Mitchnick, Krista A.; Nicholson, Kate; Wideman, Cassidy; Jardine, Kristen; Jamieson-Williams, Rhiannon; Creighton, Samantha D.; Lacoursiere, Allison; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Maclusky, Neil J.; Choleris, Elena; Winters, Boyer D. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1523/jneurosci.1574-23.2024 Codice identificativo ISI: WOS:001310415900004 Codice identificativo SCOPUS: 2-s2.0-85203269705 | |
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| 2024 | |
| Articolo in rivista | |
| Prodrug Approach to Exploit (S) Alanine as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors CHEMMEDCHEM. Vol. 19. Pag.e202400139(1)-e202400139(18) ISSN:1860-7187. | |
| Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Chini, Maria Giovanna; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202400139 Codice identificativo ISI: WOS:001253900000001 Codice identificativo SCOPUS: 2-s2.0-85196860902 | |
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| 2024 | |
| Articolo in rivista | |
| Successes and challenges in the development of BD1-selective BET inhibitors: a patent review EXPERT OPINION ON THERAPEUTIC PATENTS. Pag.1-17 ISSN:1354-3776. | |
| Viviano, Monica; Cipriano, Alessandra; Fabbrizi, Emanuele; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca; Mai, Antonello; Milite, Ciro; Rotili, Dante | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/13543776.2024.2327300 | |
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| 2024 | |
| Articolo in rivista | |
| DMSO‐Related Effects on Ligand‐Binding Properties of Lysine Methyltransferases G9a and SETD8 CHEMBIOCHEM. Vol. 25. Pag.e202300809-e202300809 ISSN:1439-4227. | |
| Feoli, Alessandra; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.202300809 Codice identificativo ISI: WOS:001148333600001 Codice identificativo SCOPUS: 2-s2.0-85183041993 | |
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| 2024 | |
| Contributo in volume (Capitolo o Saggio) | |
| Inhibiting Arginine Methylation. In Ho Man Chan, Cheryl Arrowsmith Epigenetic Drug Discovery Pag.343-382 Royal Society of Chemistry. | |
| Sbardella, Gianluca; Bedford, Mark T. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/9781837674916-00343 | |
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349978Chimica farmaceutica
| 2024 | |
| Monografia o trattato scientifico | |
| Chimica farmaceutica. Edises edizioni srl ISBN:9788836231522 | |
| Costantino, G.; Sbardella, G. | |
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| 2023 | |
| Articolo in rivista | |
| NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 66. Pag.11632-11655 ISSN:0022-2623. | |
| Cipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c00770 Codice identificativo ISI: WOS:001060994300001 Codice identificativo SCOPUS: 2-s2.0-85171309414 | |
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258840EFMC – Trends that Link Medicinal Chemistry and Chemical Biology to Translational Drug Discovery
| 2023 | |
| Articolo in rivista | |
| EFMC – Trends that Link Medicinal Chemistry and Chemical Biology to Translational Drug Discovery CHEMBIOCHEM. Pag.1-16 ISSN:1439-4227. | |
| Auberson, Yves P.; Arimondo, Paola B.; Duca, Maria; Essig, Sebastian; Grether, Uwe; Rufer, Arne C.; Sbardella, Gianluca; Schopfer, Ulrich; Torrens, Antoni; van der Stelt, Mario; Vauzeilles, Boris; Vázquez, Olalla; Zhang, Andrew X. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.202200690 Codice identificativo ISI: WOS:000940374200001 Codice identificativo SCOPUS: 2-s2.0-85149151879 | |
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| 2023 | |
| Articolo in rivista | |
| First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8 JOURNAL OF MEDICINAL CHEMISTRY. Vol. 66. Pag.6591-6616 ISSN:0022-2623. | |
| Fiorentino, Francesco; Sementilli, Sara; Menna, Martina; Turrisi, Federica; Tomassi, Stefano; Pellegrini, Francesca Romana; Iuzzolino, Angela; D'Acunzo, Francesca; Feoli, Alessandra; Wapenaar, Hannah; Taraglio, Sophie; Fraschetti, Caterina; Del Bufalo, Donatella; Sbardella, Gianluca; Dekker, Frank J; Paiardini, Alessandro; Trisciuoglio, Daniela; Mai, Antonello; Rotili, Dante | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.2c01937 Codice identificativo ISI: WOS:000988858800001 Codice identificativo SCOPUS: 2-s2.0-85159627845 | |
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| 2023 | |
| Articolo in rivista | |
| The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation CHEMMEDCHEM. Pag.1-7 ISSN:1860-7179. | |
| Quancard, Jean; Vulpetti, Anna; Bach, Anders; Cox, Brian; Guéret, Stéphanie M; Hartung, Ingo V; Koolman, Hannes F; Laufer, Stefan; Messinger, Josef; Sbardella, Gianluca; Craft, Russell | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202300002 Codice identificativo ISI: WOS:000945582500001 Codice identificativo SCOPUS: 2-s2.0-85150212364 | |
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| 2023 | |
| Articolo in rivista | |
| Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor JOURNAL OF MEDICINAL CHEMISTRY. Pag.13665-13683 ISSN:0022-2623. | |
| Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.3c01030 Codice identificativo ISI: WOS:001045914800001 Codice identificativo SCOPUS: 2-s2.0-85168362422 | |
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| 2022 | |
| Articolo in rivista | |
| Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 237. Pag.114410-114440 ISSN:0223-5234. | |
| Menna, Martina; Fiorentino, Francesco; Marrocco, Biagina; Lucidi, Alessia; Tomassi, Stefano; Cilli, Domenica; Romanenghi, Mauro; Cassandri, Matteo; Pomella, Silvia; Pezzella, Michele; Del Bufalo, Donatella; Zeya Ansari, Mohammad Salik; Tomašević, Nevena; Mladenović, Milan; Viviano, Monica; Sbardella, Gianluca; Rota, Rossella; Trisciuoglio, Daniela; Minucci, Saverio; Mattevi, Andrea; Rotili, Dante; Mai, Antonello | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.114410 Codice identificativo ISI: WOS:000804176200002 Codice identificativo SCOPUS: 2-s2.0-85129352278 | |
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| 2022 | |
| Articolo in rivista | |
| Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice LEARNING & MEMORY. Vol. 29. Pag.71-76 ISSN:1549-5485. | |
| Creighton, Samantha D.; Jardine, Kristen H.; Desimone, Alexa; Zmetana, Megan; Castellano, Sabrina; Milite, Ciro; Sbardella, Gianluca; Winters, Boyer D. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1101/lm.053536.121 Codice identificativo ISI: WOS:000757289600001 Codice identificativo SCOPUS: 2-s2.0-85124680497 | |
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| 2022 | |
| Articolo in rivista | |
| Lysine methyltransferase inhibitors: where we are now. RSC CHEMICAL BIOLOGY. Vol. 3. Pag.359-406 ISSN:2633-0679. | |
| Feoli, Alessandra; Viviano, Monica; Cipriano, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/D1CB00196E Codice identificativo ISI: WOS:000739939100001 Codice identificativo SCOPUS: 2-s2.0-85129384483 | |
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| 2022 | |
| Articolo in rivista | |
| Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 65. Pag.11574-11606 ISSN:0022-2623. | |
| Iannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.2c00252 Codice identificativo ISI: WOS:000822512300001 Codice identificativo SCOPUS: 2-s2.0-85129915280 | |
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| 2022 | |
| Articolo in rivista | |
| Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain CHEMMEDCHEM. Vol. 17. Pag.1-14 ISSN:1860-7179. | |
| Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202200343 Codice identificativo ISI: WOS:000853917200001 Codice identificativo SCOPUS: 2-s2.0-85138079605 | |
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| 2021 | |
| Abstract in rivista | |
| Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: an in vitro study JOURNAL OF TRANSLATIONAL MEDICINE. Vol. 19. Pag.8-8 ISSN:1479-5876. | |
| Fattore, Luigi; Sbardella, Gianluca; Botti, Gerardo; Mancini, Rita; Ascierto, Paolo A.; Ciliberto, Gennaro | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1186/s12967-020-02685-2 Codice identificativo ISI: WOS:000632075000009 Codice identificativo SCOPUS: 2-s2.0-85103433769 | |
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| 2021 | |
| Articolo in rivista | |
| Development of a Microscale Thermophoresis-Based Method for Screening and Characterizing Inhibitors of the Methyl-Lysine Reader Protein MRG15 SLAS DISCOVERY. Vol. 26. Pag.77-87 ISSN:2472-5552. | |
| Feoli, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Castellano, Sabrina; Bartoschik, Tanja; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1177/2472555220949166 Codice identificativo ISI: WOS:000560777300001 Codice identificativo SCOPUS: 2-s2.0-85089488195 | |
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| 2021 | |
| Articolo in rivista | |
| The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Phenotypic Drug Discovery CHEMMEDCHEM. Vol. 16. Pag.1736-1739 ISSN:1860-7179. | |
| Quancard, J.; Bach, A.; Cox, B.; Craft, R.; Finsinger, D.; Gueret, S. M.; Hartung, I. V.; Laufer, S.; Messinger, J.; Sbardella, G.; Koolman, H. F. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202100041 Codice identificativo ISI: WOS:000637424900001 Codice identificativo SCOPUS: 2-s2.0-85103902097 | |
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| 2021 | |
| Articolo in rivista | |
| The Chemical Biology-Medicinal Chemistry Continuum: EFMC′s Vision CHEMBIOCHEM. Vol. 22. Pag.1-4 ISSN:1439-4227. | |
| Duca, M.; Gillingham, D.; Olsen, C. A.; Sbardella, G.; Skaanderup, P. R.; van der Stelt, M.; Vauzeilles, B.; Vazquez, O.; Auberson, Y. P. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.202100319 Codice identificativo ISI: WOS:000680922200001 Codice identificativo SCOPUS: 2-s2.0-85112596507 | |
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| 2020 | |
| Articolo in rivista | |
| Targeting epigenetic reader domains by chemical biology CURRENT OPINION IN CHEMICAL BIOLOGY. Vol. 57. Pag.82-94 ISSN:1367-5931. | |
| Cipriano, Alessandra; Sbardella, Gianluca; Ciulli, Alessio | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.cbpa.2020.05.006 Codice identificativo ISI: WOS:000568781700013 Codice identificativo SCOPUS: 2-s2.0-85088795636 | |
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| 2020 | |
| Articolo in rivista | |
| The European Federation for Medicinal Chemistry (EFMC) Best Practice Initiative: Validating Chemical Probes CHEMMEDCHEM. Vol. 15. Pag.1-4 ISSN:1860-7179. | |
| Quancard, J.; Cox, B.; Finsinger, D.; Gueret, S. M.; Hartung, I. V.; Koolman, H. F.; Messinger, J.; Sbardella, G.; Laufer, S. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202000597 Codice identificativo ISI: WOS:000565332200001 Codice identificativo SCOPUS: 2-s2.0-85090195703 | |
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| 2020 | |
| Articolo in rivista | |
| Reverse transcriptase inhibition potentiates target therapy in BRAF-mutant melanomas: effects on cell proliferation, apoptosis, DNA-damage, ROS induction and mitochondrial membrane depolarization CELL COMMUNICATION AND SIGNALING. Vol. 18. Pag.1-9 ISSN:1478-811X. | |
| Fattore, Luigi; Malpicci, Debora; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Botti, Gerardo; Ascierto, Paolo Antonio; Mancini, Rita; Ciliberto, Gennaro | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1186/s12964-020-00633-7 Codice identificativo ISI: WOS:000573044100001 Codice identificativo SCOPUS: 2-s2.0-85091051560 | |
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| 2020 | |
| Articolo in rivista | |
| Reverse transcriptase inhibitors promote the remodeling of nuclear architecture and induce autophagy in prostate cancer cells CANCER LETTERS. Vol. 478. Pag.133-145 ISSN:0304-3835. | |
| Bellisai, Cristina; Sciamanna, Ilaria; Rovella, Paola; Giovannini, Daniela; Baranzini, Mirko; Pugliese, Giusj Monia; Zeya Ansari, Mohammad Salik; Milite, Ciro; Sinibaldi-Vallebona, Paola; Cirilli, Roberto; Sbardella, Gianluca; Pichierri, Pietro; Trisciuoglio, Daniela; Lavia, Patrizia; Serafino, Annalucia; Spadafora, Corrado | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.canlet.2020.02.029 Codice identificativo ISI: WOS:000525868400013 Codice identificativo SCOPUS: 2-s2.0-85081900118 | |
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| 2020 | |
| Articolo in rivista | |
| Two novel SIRT1 activators, SCIC2 and SCIC2.1, enhance SIRT1-mediated effects in stress response and senescence EPIGENETICS. Vol. 15. Pag.664-683 ISSN:1559-2294. | |
| Scisciola, Lucia; Sarno, Federica; Carafa, Vincenzo; Cosconati, Sandro; Di Maro, Salvatore; Ciuffreda, Loreta; De Angelis, Antonella; Stiuso, Paola; Feoli, Alessandra; Sbardella, Gianluca; Altucci, Lucia; Nebbioso, Angela | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/15592294.2019.1704349 Codice identificativo ISI: WOS:000507445400001 Codice identificativo SCOPUS: 2-s2.0-85078601869 | |
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| 2020 | |
| Articolo in rivista | |
| Safety and efficacy of the Russian COVID-19 vaccine: more information needed THE LANCET. Vol. 10256. Pag.e53-e53 ISSN:0140-6736. | |
| Bucci, Enrico; Andreev, Konstantin; Björkman, Anders; Calogero, Raffaele Adolfo; Carafoli, Ernesto; Carninci, Piero; Castagnoli, Paola; Cossarizza, Andrea; Mussini, Cristina; Guerin, Philippe; Lipworth, Brian; Sbardella, Gianluca; Stocki, Teresa; Tuosto, Loretta; van Tulleken, Christoffer; Viola, Antonella | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/S0140-6736(20)31960-7 Codice identificativo ISI: WOS:000579146300001 Codice identificativo SCOPUS: 2-s2.0-85091778941 | |
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| 2020 | |
| Contributo in volume (Capitolo o Saggio) | |
| Methyl-Readers and Inhibitors. In A Ganesan, Christian A. Olsen, Maija Lahtela-Kakkonen, Dante Rotili, Sergio Valente, Nathaniel I. Martin, Takayoshi Suzuki, Akane Kawamura, Paola B. Arimondo, Natalia Tretyakova, Gianluca Sbardella, William Pomerantz, Raymond Pierce, Frank J Dekker, Lucia Altucci, Carlo M. Croce, Maria Berdasco Menendez Chemical Epigenetics Pag.339-399 Berlin, Heidelberg Springer, Berlin, Heidelberg. ISSN:1862-2461. | |
| Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1007/7355_2019_78 Codice identificativo SCOPUS: 2-s2.0-85083996113 | |
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| 2020 | |
| Contributo in volume (Capitolo o Saggio) | |
| Chemioterapici antiprotozoari. In Chimica farmaceutica. Con e-book Pag.860-880 Bologna Zanichelli Editore SpA. ISBN:9788808420268 | |
| Sbardella, Gianluca | |
| Versione online | |
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| 2019 | |
| Articolo in rivista | |
| Discovery of a novel chemotype of histone lysine methyltransferase EHMT1/2 (GLP/G9a) inhibitors: rational design, synthesis, biological evaluation and co-crystal structure JOURNAL OF MEDICINAL CHEMISTRY. Vol. 62. Pag.2666-2689 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Horton, John R; Rescigno, Donatella; Cipriano, Alessandra; Pisapia, Vincenzo; Viviano, Monica; Pepe, Giacomo; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Cheng, Xiaodong; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.8b02008 Codice identificativo ISI: WOS:000461537000030 Codice identificativo SCOPUS: 2-s2.0-85062555799 | |
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| 2019 | |
| Articolo in rivista | |
| Look for methods, not conclusions CELL DEATH & DISEASE. Vol. 10. Pag.931-932 ISSN:2041-4889. | |
| Bassi, Roberto; Bucci, Enrico M; Calogero, Raffaele A; Carninci, Piero; Ciliberto, Gennaro; Conte, Pellegrino; De Luca, Michele; Corbellini, Gilberto; Giordano, Antonio; Marchionni, Luigi; Massaro Giordano, Giacomina; Parini, Angelo; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/s41419-019-2179-8 Codice identificativo ISI: WOS:000502974500007 Codice identificativo SCOPUS: 2-s2.0-85076044631 | |
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| 2019 | |
| Articolo in rivista | |
| Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 163. Pag.722-735 ISSN:0223-5234. | |
| Stazi, Giulia; Battistelli, Cecilia; Piano, Valentina; Mazzone, Roberta; Marrocco, Biagina; Marchese, Sara; Louie, Sharon M.; Zwergel, Clemens; Antonini, Lorenzo; Patsilinakos, Alexandros; Ragno, Rino; Viviano, Monica; Sbardella, Gianluca; Ciogli, Alessia; Fabrizi, Giancarlo; Cirilli, Roberto; Strippoli, Raffaele; Marchetti, Alessandra; Tripodi, Marco; Nomura, Daniel K.; Mattevi, Andrea; Mai, Antonello; Valente, Sergio | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2018.11.050 Codice identificativo ISI: WOS:000458597300053 Codice identificativo SCOPUS: 2-s2.0-85058530369 | |
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| 2019 | |
| Contributo in volume (Capitolo o Saggio) | |
| Histone Acetyltransferases: Targets and Inhibitors. In W. Sippl, M. Jung Epigenetic Drug Discovery Pag.297-345 Weinheim Wiley-VCH. ISSN:1432-4636. | |
| Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/9783527809257.ch12 Codice identificativo ISI: WOS:000483635500014 | |
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| 2018 | |
| Articolo in rivista | |
| Combined HAT/EZH2 modulation leads to cancer-selective cell death ONCOTARGET. Vol. 9. Pag.25630-25646 ISSN:1949-2553. | |
| Petraglia, Francesca; Singh, Abhishek A.; Carafa, Vincenzo; Nebbioso, Angela; Conte, Mariarosaria; Scisciola, Lucia; Valente, Sergio; Baldi, Alfonso; Mandoli, Amit; Petrizzi, Valeria Belsito; Ingenito, Concetta; De Falco, Sandro; Cicatiello, Valeria; Apicella, Ivana; Janssen-Megens, Eva M.; Kim, Bowon; Yi, Guoqiang; Logie, Colin; Heath, Simon; Ruvo, Menotti; Wierenga, Albertus T. J.; Flicek, Paul; Yaspo, Marie Laure; Della Valle, Veronique; Bernard, Olivier; Tomassi, Stefano; Novellino, Ettore; Feoli, Alessandra; Sbardella, Gianluca; Gut, Ivo; Vellenga, Edo; Stunnenberg, Hendrik G.; Mai, Antonello; Martens, Joost H. A.; Altucci, Lucia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.18632/oncotarget.25428 Codice identificativo SCOPUS: 2-s2.0-85047400725 | |
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| 2018 | |
| Poster | |
| Design, synthesis and biological evaluation of new selective arginine methyltransferases (PRMTs) Inhibitors. In: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily2018 BOOK OF ABSTRACTS Pag.136-136 | |
| Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily2018 Palermo 17-20 Luglio 2018 | |
| Milite, C.; Feoli, A.; Rescigno, D.; Clarke, S.; Castellano, S.; Sbardella, G. | |
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| 2018 | |
| Poster | |
| Expanding the quinazoline ring to 3H-benzo[e][1,4]diazepine: development of new and selective G9a inhibitors. In: Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry MedChemSicily2018 BOOK OF ABSTRACTS Pag.135-135 | |
| Italian-Spanish-Portuguese Joint Meeting in Medicinal Chemistry - MedChemSicily2018 Palermo 17-20 Luglio 2018 | |
| Milite, C.; Feoli, A.; Rescigno, Donatella; Pisapia, Vincenzo; Cosconati, S.; Castellano, S.; Sbardella, G. | |
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| 2017 | |
| Articolo in rivista | |
| Exploiting the 4-Phenylquinazoline Scaffold for the Development of High Affinity Fluorescent Probes for the Translocator Protein (TSPO) JOURNAL OF MEDICINAL CHEMISTRY. Vol. 60. Pag.7897-7909 ISSN:0022-2623. | |
| Milite, Ciro; Barresi, Elisabetta; Da Pozzo, Eleonora; Costa, Barbara; Viviano, Monica; Porta, Amalia; Messere, Anna; Sbardella, Gianluca; Da Settimo, Federico; Novellino, Ettore; Cosconati, Sandro; Castellano, Sabrina; Taliani, Sabrina; Martini, Claudia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.7b01031 Codice identificativo ISI: WOS:000412150300017 Codice identificativo SCOPUS: 2-s2.0-85030253369 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Regulation of USP37 Expression by REST-associated G9a-dependent Histone Methylation MOLECULAR CANCER RESEARCH. Vol. 15. Pag.1073-1084 ISSN:1541-7786. | |
| Dobson, Tara; Hatcher, Rashieda J; Swaminathan, Jyothismathi; Das, Chandra M; Shaik, Shavali; Tao, Rong Hua; Milite, Ciro; Castellano, Sabrina; Taylor, Pete; Sbardella, Gianluca; Gopalakrishnan, Vidya | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1158/1541-7786.MCR-16-0424 Codice identificativo ISI: WOS:000406681200011 Codice identificativo SCOPUS: 2-s2.0-85026641347 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Developing Spindlin1 small-molecule inhibitors by using protein microarrays NATURE CHEMICAL BIOLOGY. Vol. 13. Pag.750-756 ISSN:1552-4450. | |
| Bae, Narkhyun; Viviano, Monica; Su, Xiaonan; Lv, Jie; Cheng, Donghang; Sagum, Cari; Castellano, Sabrina; Bai, Xue; Johnson, Claire; Khalil, Mahmoud Ibrahim; Shen, Jianjun; Chen, Kaifu; Li, Haitao; Sbardella, Gianluca; Bedford, Mark T. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/nchembio.2377 Codice identificativo ISI: WOS:000403673700011 Codice identificativo SCOPUS: 2-s2.0-85021067771 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Inhibition of Wnt/β-Catenin pathway and Histone acetyltransferase activity by Rimonabant: a therapeutic target for colon cancer SCIENTIFIC REPORTS. Vol. 7. Pag.1-14 ISSN:2045-2322. | |
| Proto, MARIA CHIARA; Fiore, Donatella; Piscopo, Chiara; Franceschelli, Silvia; Bizzarro, Valentina; Laezza, Chiara; Lauro, Gianluigi; Feoli, Alessandra; Tosco, Alessandra; Bifulco, Giuseppe; Sbardella, Gianluca; Bifulco, Maurizio; Gazzerro, Patrizia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/s41598-017-11688-x Codice identificativo ISI: WOS:000410859400010 Codice identificativo SCOPUS: 2-s2.0-85029517928 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| A transcriptional coregulator, SPIN-DOC, attenuates the coactivator activity of Spindlin1 THE JOURNAL OF BIOLOGICAL CHEMISTRY. Vol. 292. Pag.20808-20817 ISSN:0021-9258. | |
| Bae, Narkhyun; Gao, Min; Li, Xu; Premkumar, Tolkappiyan; Sbardella, Gianluca; Chen, Junjie; Bedford, Mark T. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1074/JBC.M117.814913 Codice identificativo ISI: WOS:000418453400001 Codice identificativo SCOPUS: 2-s2.0-85039439820 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Articolo in rivista | |
| Transition state mimics are valuable mechanistic probes for structural studies with the arginine methyltransferase CARM1 PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA. Vol. 114. Pag.3625-3630 ISSN:0027-8424. | |
| van Haren, Matthijs J.; Marechal, Nils; Troffer Charlier, Nathalie; Cianciulli, Agostino; Sbardella, Gianluca; Cavarelli, Jean; Martin, Nathaniel I. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1073/pnas.1618401114 Codice identificativo ISI: WOS:000398159000042 Codice identificativo SCOPUS: 2-s2.0-85016997146 | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Contributo in Atti di convegno | |
| Sympathy for the methyl: a library-on-library screening approach to identify small-molecule ligands of methyl-lysine reader proteins. In: Epigenetic Chemical Probes Pag.5-5 | |
| Epigenetic Chemical Probes Belgrade, Republic of Serbia 16th January 2017 | |
| Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Poster | |
| Design, synthesis and biological evaluation of novel G9a inhibitors with improved brain permeability from a scaffold hopping approach. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.67-67 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Poster | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.62-62 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Poster | |
| Design, synthesis and in vitro evaluation of bivalent chemical probes for bromo and extra-terminal domain (BET) proteins. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.52-52 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Cipriano, Alessandra; Milite, Ciro; Panagis, Filippakopoulos; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Poster | |
| Identification of new KDM4 inhibitors through a HTS and hit refinement strategy. In: Atti del XXVI Congresso Nazionale della Società Chimica Italiana Pag.49-49 | |
| XXVI Congresso Nazionale della Società Chimica Italiana Paestum (SA) 10-14 settembre 2017 | |
| Balzano, AMODIO LUCA; Sarno, Federica; Milite, Ciro; Franci, Gianluigi; Forné, Ignasi; Lucia, Altucci; Rino, Ragno; Fabrizio, Micheli; Axel, Imhof; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2017 | |
| Recensione in rivista | |
| Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian CHEMMEDCHEM. Vol. 12. Pag.1099-1100 ISSN:1860-7179. | |
| Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201600641 Codice identificativo SCOPUS: 2-s2.0-85021026372 | |
| Show it in Product Database (IRIS) |
106150Cell-Permeable modulators of Histone Acetyltransferases for the regulation of behavioral plasticity
| 2016 | |
| Abstract in Atti di convegno | |
| Cell-Permeable modulators of Histone Acetyltransferases for the regulation of behavioral plasticity. In: 3rd Freiburg Epigenetic Spring Meeting: Chemical Biology of Epigenetics Pag.1-2 | |
| 3rd Freiburg Epigenetic Spring Meeting: Chemical Biology of Epigenetics Freiburg Institute for Advanced Studies Albert-Ludwigs-Universität Freiburg, Germany 10-13 April 2016 | |
| Sbardella, Gianluca | |
| Versione online | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Abstract in Atti di convegno | |
| A “library-on-library” screening approach to identify small-molecule ligands of methyl-lysine reader proteins. In: 2nd Annual Epigenetics Discovery Congress Pag.1-7 | |
| 2nd Annual Epigenetics Discovery Congress London Heathrow Marriott Hotel Bath Road, Heathrow Airport Hayes UB3 5AN, London, United Kingdom 8-9 September 2016 | |
| Sbardella, Gianluca | |
| Versione online | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Abstract in Atti di convegno | |
| Identification of new inhibitors of PRMTs by a multi-substrate-adduct approach. In: XXIV NMMC & 10th NPCF - September 11th-14th 2016, Perugia (Italy) - Book of Abstract Pag.77-77 | |
| XXIV NMMC & 10th NPCF Perugia (Italy) 11-14 Settembre 2016 | |
| Milite, Ciro; Rescigno, Donatella; Feoli, Alessandra; Nunziata, Antonietta; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Abstract in rivista | |
| ChemInform Abstract: Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors CHEM INFORM. Vol. 47. Pag.1-1 ISSN:0931-7597. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201642266 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| The emerging role of lysine methyltransferase SETD8 in human diseases CLINICAL EPIGENETICS. Vol. 8. Pag.1-15 ISSN:1868-7083. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Cianciulli, Agostino; Balzano, AMODIO LUCA; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1186/s13148-016-0268-4 Codice identificativo ISI: WOS:000384471400001 Codice identificativo SCOPUS: 2-s2.0-84994805952 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| Arginine demethylation of G3BP1 promotes stress granule assembly THE JOURNAL OF BIOLOGICAL CHEMISTRY. Vol. 291. Pag.22671-22685 ISSN:0021-9258. | |
| Tsai, Wei Chih; Gayatri, Sitaram; Reineke, Lucas C; Sbardella, Gianluca; Bedford, Mark T; Lloyd, Richard E. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1074/jbc.M116.739573 Codice identificativo ISI: WOS:000386760600027 Codice identificativo SCOPUS: 2-s2.0-84992345066 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| The 23(rd) National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015) CHEMMEDCHEM. Vol. 11. Pag.1670-1675 ISSN:1860-7179. | |
| Campiglia, Pietro; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201600358 Codice identificativo ISI: WOS:000383579700001 Codice identificativo SCOPUS: 2-s2.0-84983354256 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Articolo in rivista | |
| Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors CHEMMEDCHEM. Vol. 11. Pag.1680-1685 ISSN:1860-7179. | |
| Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Rescigno, Donatella; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201600272 Codice identificativo ISI: WOS:000383579700002 Codice identificativo SCOPUS: 2-s2.0-84983335802 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Contributo in Atti di convegno | |
| MECHANISMS OF IMMUNE RESISTANCE IN PEDIATRIC POSTERIOR FOSSA TUMORS. In: Abstracts from the 17th International Symposium on Pediatric Neuro-Oncology (ISPNO) June 12 — 15, 2016 Liverpool, United Kingdom Oxford, UK Oxford University Press Vol.18, Pag.170-170 | |
| 17th International Symposium on Pediatric Neuro-Oncology (ISPNO) Liverpool, United Kingdom June 12 — 15, 2016 | |
| Brugmann, William; Laureano, Alvaro; Torchia, Jonathan; Hatcher, Rashieda; Kennis, Bridget; Khatua, Soumen; Zaky, Wafik; Sbardella, Gianluca; Moyes, Judy; Goldman, Stewart; Lulla, Rishi; Fangusaro, Jason; Sandberg, David; Silla, Lucia; Rajaram, Veena; Hawkins, Cynthia; Huang, Annie; Cooper, Laurence; Lee, Dean; Gopalakrishnan, Vidya | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1093/neuonc/now084.05 Codice identificativo ISI: WOS:000379749000681 | |
| Show it in Product Database (IRIS) |
| 2016 | |
| Poster | |
| IDENTIFICATION OF NEW KDM4 INHIBITORS THROUGH A HTS AND HIT REFINEMENT STRATEGY. In: XXIV NMMC & 10th NPCF - September 11th-14th 2016, Perugia (Italy) - Book of Abstract Pag.88-88 | |
| XXIV NMMC & 10th NPCF PA 11-14 Settembre 2016 | |
| Balzano, AMODIO LUCA; Sarno, Federica; Fasanino, Mariacristina; Milite, Ciro; Franci, Gianluigi; Altucci, Lucia; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
149157DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH
| 2016 | |
| Poster | |
| DESIGN, SYNTHESIS AND BIOLOGICAL EVALUATION OF NOVEL G9A INHIBITORS FROM A SCAFFOLD HOPPING APPROACH. In: XXIV NMMC & 10th NPCF - September 11th-14th 2016, Perugia (Italy) - Book of Abstract Pag.207-207 | |
| XXIV NMMC & 10th NPCF Perugia 11-14 Settembre 2016 | |
| Rescigno, Donatella; Milite, Ciro; Viviano, Monica; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Abstract in Atti di convegno | |
| Discovery of the first-in-class chemical probe for the Spindlin1 methyl-lysine reader domain. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.37-37 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Li, Haitao; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Abstract in rivista | |
| ChemInform Abstract: A Continuous-Flow Synthesis of 1,4-Benzodiazepin-5-ones, Privileged Scaffolds for Drug Discovery CHEM INFORM. Vol. 46. Pag.no-no ISSN:0931-7597. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201520216 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Abstract in rivista | |
| Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015) CHEMMEDCHEM. Vol. 10. Pag.2-2 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Mai, Antonello; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201490050 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| A novel cell-permeable, selective and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 58. Pag.2779-2798 ISSN:0022-2623. | |
| Milite, Ciro; Feoli, Alessandra; Kazuki, Sasaki; Valeria, La Pietra; Balzano, AMODIO LUCA; Luciana, Marinelli; Antonello, Mai; Ettore, Novellino; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm5019687 Codice identificativo ISI: WOS:000351971800013 Codice identificativo SCOPUS: 2-s2.0-84925957014 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Ellagic Acid-Changed Epigenome of Ribosomal Genes and Condensed RPA194-Positive Regions of Nucleoli in Tumour Cells FOLIA BIOLOGICA. Vol. 61. Pag.49-59 ISSN:0015-5500. | |
| Legartová, Soňa; Sbardella, Gianluca; Kozubek, Stanislav; Bártová, Eva | |
| Versione online | |
| Codice identificativo ISI: WOS:000355375900001 Codice identificativo SCOPUS: 2-s2.0-84930704221 | |
| Show it in Product Database (IRIS) |
62075A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery
| 2015 | |
| Articolo in rivista | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery RSC ADVANCES. Vol. 5. Pag.1268-1273 ISSN:2046-2069. | |
| Viviano, Monica; Milite, Ciro; Rescigno, Donatella; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/C4RA13392G Codice identificativo ISI: WOS:000346079900051 Codice identificativo SCOPUS: 2-s2.0-84916613613 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| CARM1 modulators affect epigenome of stem cells and change morphology of nucleoli PHYSIOLOGICAL RESEARCH. Vol. 64. Pag.769-782 ISSN:1802-9973. | |
| Franek, M; Legartová, S; Suchánková, J; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca; Kozubek, S; Bártová, E. | |
| Versione online | |
| Codice identificativo ISI: WOS:000367154800019 Codice identificativo SCOPUS: 2-s2.0-84983200500 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Articolo in rivista | |
| Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF CHEMMEDCHEM. Vol. 10. Pag.144-157 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Antonello, Mai; Ettore, Novellino; Tosco, Alessandra; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201402371 Codice identificativo ISI: WOS:000346766700014 Codice identificativo SCOPUS: 2-s2.0-84919779703 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in Atti di convegno | |
| STUDY OF EPIGENETIC DEREGULATION OF A NOVEL DEUBIQUITYLASE IN MEDULLOBLASTOMA. In: Abstracts from the 3rd Biennial Conference on Pediatric Neuro-Oncology Basic and Translational Research Oxford, UK Oxford University Press Vol.17, Pag.8-8 | |
| 3rd Biennial Conference on Pediatric Neuro-Oncology Basic and Translational Research San Diego, CA 7-9 maggio 2015 | |
| Hatcher, R.; Das, C.; Fangusaro, J.; Rajaram, V.; Lulla, R.; Goldman, S.; Khatua, S.; Sbardella, Gianluca; Gopalakrishnan, V. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1093/neuonc/nov061.29 Codice identificativo ISI: WOS:000361304800030 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in volume (Capitolo o Saggio) | |
| Chemioterapici antiprotozoari. In Alberto Gasco,Fulvio Gualtieri,Carlo Melchiorre Chimica farmaceutica Pag.832-852 Bologna Zanichelli Editore spa. ISBN:9788808187123 | |
| Sbardella, Gianluca | |
| Digital Object Identifier (DOI): 10.978.8808/187123 | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Contributo in volume (Capitolo o Saggio) | |
| Agenti antimicotici, antimicobatterici e antiprotozoari. In Maria Laura Bolognesi, Paola Conti, Gabriele Costantino, Gloria Cristalli, Roberta Fruttero, Loretta Lazzarato, Giovanni Lentini, Marco Macchia, Antonio Macchiarulo, Antonello Mai, Clementina Manera, Gabriella Marucci, Filippo Minutolo, Marco Mor, Gianluca Sbardella, Rosaria Volpini Chimica Farmaceutica di Graham L. Patrick Pag.589-636 Napoli EdiSES. ISBN:9788879598453 | |
| Costantino, Gabriele; Mai, Antonello; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Identification of novel small-molecule ligands of methyl-lysine binding protein PHF20. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.248-248 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Tosco, Alessandra; Mer, Georges; Bedford, Mark T.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Discovery of new chemical probes for the MRG15 chromo domain.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.249-249 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Bedford, Mark T.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Design, synthesis and biological evaluation of pyrrole derivatives as coactivator associated arginine methyltransferase 1 (CARM1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.247-247 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Cianciulli, Agostino; Milite, Ciro; Castellano, Sabrina; Chini, MARIA GIOVANNA; Bifulco, Giuseppe; Xu, Wei; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Synthesis and biological evaluation of delta2-isoxazoline derivatives as DNA methyltransferase 1 (DNMT1) inhibitors. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.250-250 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Viviano, Monica; Castellano, Sabrina; Conti, Paola; Tamborini, Lucia; Novellino, Ettore; Lyko, Frank; Medina-Franco, Josè; Jeltsch, Albert; Arimondo, Paola B.; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Development of a Non-Radioactive, No-Wash Biochemical Assay for High-Throughput Screening of Small Molecule Modulators of PHF20.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.245-245 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Castellano, Sabrina; Tosco, Alessandra; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Use of Microscale Thermophoresis (MST) for Studying binding interactions of PRSet-7/SETD8 with small molecule specific inhibitors EPI-9 and EPI-23.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.244-244 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Viviano, Monica; Imhof, Axel; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| Biomolecular and biophysical approaches to interrogate p300: a platform for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.243-243 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Feoli, Alessandra; Milite, Ciro; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2015 | |
| Poster | |
| From garcinol to barbituric acid derivatives: development of a novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.241-241 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Milite, Ciro; Feoli, Alessandra; La Pietra, Valeria; Marinelli, Luciana; Mai, Antonello; Sasaki, Kazuki; Novellino, Ettore; Tosco, Alessandra; Castellano, Sabrina; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
149068A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.
| 2015 | |
| Poster | |
| A continuous-flow synthesis of 1,4-benzodiazepin-5-ones, privileged scaffolds for drug discovery.. In: XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) - Abstract e-book Pag.239-239 | |
| XXIII National Meeting on Medicinal Chemistry (NMMC2015) and 9th Young Medicinal Chemists Symposium “Nuove Prospettive in Chimica Farmaceutica” (NPCF9) Campus di Fisciano - Università degli Studi di Salerno September 6-9 2015 | |
| Rescigno, Donatella; Viviano, Monica; Milite, Ciro; Sbardella, Gianluca; Castellano, Sabrina | |
| Show it in Product Database (IRIS) |
149066FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS.
| 2014 | |
| Abstract in Atti di convegno | |
| FROM GARCINOL TO BARBITURIC ACID DERIVATIVES: DEVELOPMENT OF NEW AND SELECTIVE P300 INHIBITORS.. In: VIII Edizione del Meeting "Nuove Prospettive in Chimica Farmaceutica”(NPCF8) - Book degli Abstracts Pag.35-35 | |
| VIII Edizione del Meeting "Nuove Prospettive in Chimica Farmaceutica”(NPCF8) Parma - Starhotel Du Parc 9 – 11 Giugno 2014 | |
| Milite, Ciro; Castellano, Sabrina; Feoli, Alessandra; La Pietra, Valeria; Cosconati, Sandro; Mai, Antonello; Sasaki, Kazuki; Yoshida, Minoru; Novellino, Ettore; Tosco, Alessandra; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| The Histone Acetylase Activator Pentadecylidenemalonate 1b Rescues Proliferation and Differentiation in Human Cardiac Mesenchymal Cells of Type 2 Diabetic Patients DIABETES. Vol. 63. Pag.2132-2147 ISSN:0012-1797. | |
| Vecellio, Matteo; Spallotta, Francesco; Nanni, Simona; Colussi, Claudia; Cencioni, Chiara; Derlet, Anja; Bassetti, Beatrice; Tilenni, Manuela; Carena, Maria Cristina; Farsetti, Antonella; Sbardella, Gianluca; Castellano, Sabrina; Mai, Antonello; Martelli, Fabio; Pompilio, Giulio; Capogrossi, Maurizio C.; Rossini, Alessandra; Dimmeler, Stefanie; Zeiher, Andreas; Gaetano, Carlo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.2337/db13-0731 Codice identificativo ISI: WOS:000336643900037 Codice identificativo SCOPUS: 2-s2.0-84899824083 | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells CHEMMEDCHEM. Vol. 9. Pag.542-548 ISSN:1860-7179. | |
| Alessia, Lenoci; Stefano, Tomassi; Mariarosaria, Conte; Rosaria, Benedetti; Veronica, Rodriguez; Simone, Carradori; Daniela, Secci; Castellano, Sabrina; Sbardella, Gianluca; Patrizia, Filetici; Ettore, Novellino; Lucia, Altucci; Dante, Rotili; Antonello, Mai | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.201300536 Codice identificativo ISI: WOS:000331795500010 Codice identificativo SCOPUS: 2-s2.0-84896698147 | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| Structure–Activity Relationship Refinement and Further Assessment of 4-phenylquinazoline-2-carboxamide Translocator Protein (TSPO) Ligands as Antiproliferative Agents in Human Glioblastoma Tumors. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 57. Pag.2413-2428 ISSN:0022-2623. | |
| Castellano, Sabrina; Sabrina, Taliani; Viviano, Monica; Milite, Ciro; Eleonora Da, Pozzo; Barbara, Costa; Elisabetta, Barresi; Agostino, Bruno; Sandro, Cosconati; Luciana, Marinelli; Giovanni, Greco; Ettore, Novellino; Sbardella, Gianluca; Federico Da, Settimo; Claudia, Martini | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm401721h Codice identificativo ISI: WOS:000333578400017 Codice identificativo SCOPUS: 2-s2.0-84897411408 | |
| Show it in Product Database (IRIS) |
| 2014 | |
| Articolo in rivista | |
| Synthesis and Evaluation of Translocator 18 kDa Protein (TSPO) Positron Emission Tomography (PET) Radioligands with Low Binding Sensitivity to Human Single Nucleotide Polymorphism rs6971 ACS CHEMICAL NEUROSCIENCE. Vol. 5. Pag.963-971 ISSN:1948-7193. | |
| Paolo Zanotti, Fregonara; Yi, Zhang; Kimberly J., Jenko; Robert L., Gladding; Sami S., Zoghbi; Masahiro, Fujita; Sbardella, Gianluca; Castellano, Sabrina; Sabrina, Taliani; Claudia, Martini; Robert B., Innis; Federico Da, Settimo; Victor W., Pike | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/cn500138n Codice identificativo ISI: WOS:000343276600012 Codice identificativo SCOPUS: 2-s2.0-84908022420 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Abstract in rivista | |
| Cover Picture: A TR-FRET-Based Functional Assay for Screening Activators of CARM1 (ChemBioChem 7/2013) CHEMBIOCHEM. Vol. 14. Pag.773-773 ISSN:1439-4227. | |
| Zeng, Hao; Wu, Jiacai; Bedford, Mark T.; Sbardella, Gianluca; Hoffmann, F. Michael; Bi, Kun; Xu, Wei | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.201390020 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Articolo in rivista | |
| A TR-FRET-Based Functional Assay for Screening Activators of CARM1 CHEMBIOCHEM. Vol. 14. Pag.827-835 ISSN:1439-7633. | |
| Hao, Zeng; Jiacai, Wu; Mark T., Bedford; Sbardella, Gianluca; F., Michael Hoffmann; Kun, Bi; Wei, Xu | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.201300029 Codice identificativo ISI: WOS:000318280500008 Codice identificativo SCOPUS: 2-s2.0-84877067824 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Articolo in rivista | |
| Antifungal activity of azole compounds CPA18 and CPA109 against azole-susceptible and -resistant strains of Candida albicans JOURNAL OF ANTIMICROBIAL CHEMOTHERAPY. Vol. 68. Pag.1111-1119 ISSN:0305-7453. | |
| Calabrese, ELENA CONCETTA; Castellano, Sabrina; M., Santoriello; C., Sgherri; M. F., Quartacci; L., Calucci; A. G. S., Warrilow; D. C., Lamb; S. L., Kelly; Milite, Ciro; Granata, Ilaria; Sbardella, Gianluca; G., Stefancich; Maresca, Bruno; Porta, Amalia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1093/jac/dks506 Codice identificativo ISI: WOS:000318105100021 Codice identificativo SCOPUS: 2-s2.0-84877133207 | |
| Show it in Product Database (IRIS) |
| 2013 | |
| Articolo in rivista | |
| Enhancement of lysine acetylation accelerates wound repair COMMUNICATIVE & INTEGRATIVE BIOLOGY. Vol. 6. Pag.e25466-1-e25466-3 ISSN:1942-0889. | |
| Francesco, Spallotta; Chiara, Cencioni; Stefania, Straino; Sbardella, Gianluca; Castellano, Sabrina; Maurizio C., Capogrossi; Fabio, Martelli; Carlo, Gaetano | |
| Versione online | |
| Digital Object Identifier (DOI): 10.4161/cib.25466 Codice identificativo SCOPUS: 2-s2.0-84884691965 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Straightforward, Metal-free, and Stereoselective Synthesis of 9-Oxo- and 10-Hydroxy-2(E)-decenoic acids, Important Components of Honeybee (Apis mellifera) secretions RSC ADVANCES. Vol. 2. Pag.5229-5233 ISSN:2046-2069. | |
| Milite, Ciro; Viviano, Monica; Marisabella, Santoriello; Fabio, Arico`; Sbardella, Gianluca; Castellano, Sabrina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/c2ra20275a Codice identificativo ISI: WOS:000304487000043 Codice identificativo SCOPUS: 2-s2.0-84893259222 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells BIOCHIMIE. Vol. 94. Pag.2308-2313 ISSN:0300-9084. | |
| Sergio, Valente; Ilaria, Lepore; Carmela, Dell’Aversana; Tardugno, Maria; Castellano, Sabrina; Sbardella, Gianluca; Stefano, Tomassi; Salvatore Di, Maro; Ettore, Novellino; Roberto Di, Santo; Roberta, Costi; Lucia, Altucci; Antonello, Mai | |
| Digital Object Identifier (DOI): 10.1016/j.biochi.2012.06.003 Codice identificativo ISI: WOS:000310929200011 Codice identificativo SCOPUS: 2-s2.0-84867395419 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| p300/CBP-Associated Factor Selectively Regulates the Extinction of Conditioned Fear THE JOURNAL OF NEUROSCIENCE. Vol. 32. Pag.11930-11941 ISSN:0270-6474. | |
| Wei, Wei; Coelho, Carlos M.; Li, Xiang; Marek, Roger; Yan, Shanzhi; Anderson, Shawn; Meyers, David; Mukherjee, Chandrani; Sbardella, Gianluca; Castellano, Sabrina; Milite, Ciro; Rotili, Dante; Mai, Antonello; Cole, Philip A.; Sah, Pankaj; Kobor, Michael S.; Bredy, Timothy W. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1523/JNEUROSCI.0178-12.2012 Codice identificativo ISI: WOS:000308213900003 Codice identificativo SCOPUS: 2-s2.0-84865472870 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| P300/CBP Associated Factor Regulates Nitroglycerin-Dependent Arterial Relaxation by N -Lysine Acetylation of Contractile Proteins ARTERIOSCLEROSIS, THROMBOSIS, AND VASCULAR BIOLOGY. Vol. 32. Pag.2435-2443 ISSN:1079-5642. | |
| Colussi, Claudia); Scopece, Alessandro; Vitale, Serena; Spallotta, Francesco; Mattiussi, Stefania; Rosati, Jessica; Illi, Barbara; Mai, Antonello; Castellano, Sabrina; Sbardella, Gianluca; Farsetti, Antonella; Capogrossi, Maurizio C.; Gaetano, Carlo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1161/ATVBAHA.112.254011 Codice identificativo ISI: WOS:000308811200013 Codice identificativo SCOPUS: 2-s2.0-84866630451 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Synthesis and Biological Evaluation of 4-Phenylquinazoline-2-carboxamides Designed as a Novel Class of Potent Ligands of the Translocator Protein JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.4506-4510 ISSN:0022-2623. | |
| Castellano, Sabrina; Sabrina, Taliani; Milite, Ciro; Isabella, Pugliesi; Eleonora Da, Pozzo; Elisa, Rizzetto; Sara, Bendinelli; Barbara, Costa; Sandro, Cosconati; Giovanni, Greco; Ettore, Novellino; Sbardella, Gianluca; Giorgio, Stefancich; Claudia, Martini; Federico Da, Settimo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm201703k Codice identificativo ISI: WOS:000303785900036 Codice identificativo SCOPUS: 2-s2.0-84861054375 | |
| Show it in Product Database (IRIS) |
| 2012 | |
| Articolo in rivista | |
| Identification of Small-Molecule Enhancers of Arginine Methylation Catalyzed by Coactivator-Associated Arginine Methyltransferase 1 JOURNAL OF MEDICINAL CHEMISTRY. Vol. 55. Pag.9875-9890 ISSN:0022-2623. | |
| Castellano, Sabrina; Spannhoff, Astrid; Milite, Ciro; DAL PIAZ, Fabrizio; Cheng, Donghang; Tosco, Alessandra; Viviano, Monica; Yamani, Abdellah; Cianciulli, Agostino; Sala, Marina; Cura, Vincent; Cavarelli, Jean; Novellino, Ettore; Mai, Antonello; Bedford, Mark T.; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm301097p Codice identificativo ISI: WOS:000311461500040 Codice identificativo SCOPUS: 2-s2.0-84869995779 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Abstract in Atti di convegno | |
| Abstract 11858: Epigenetic Reversion of Metabolic Memory Alterations in Human Cardiac Stromal Cells Isolated from Type-2 Diabetic Patients. In: Abstracts from American Heart Association Scientific Sessions 2011 Baltimore, MD; Stanford, CA (USA) Lippincott Williams & Wilkins;Highwire Press Vol.124, Pag.A11858-A11858 | |
| American Heart Association - Scientific Sessions 2011 Orange County Convention Center - Orlando, FL (USA) 12-16 Novembre 2011 | |
| M., Vecellio; G., Pompilio; F., Spallotta; C., Colussi; Sbardella, Gianluca; Castellano, Sabrina; A., Mai; M. C., Capogrossi; A., Rossini; C., Gaetano | |
| Versione online | |
| Codice identificativo ISI: WOS:000299738704023 | |
| Show it in Product Database (IRIS) |
79476ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators
| 2011 | |
| Abstract in rivista | |
| ChemInform Abstract: Chemical Biology of Histone Acetyltransferase Natural Compounds Modulators CHEM INFORM. Vol. 42. Pag.no-no ISSN:0931-7597. | |
| DAL PIAZ, Fabrizio; Vassallo, Antonio; Cuesta Rubio, Osmany; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.201136272 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54. Pag.7663-7677 ISSN:0022-2623. | |
| Castellano, Sabrina; Dirk, Kuck; Viviano, Monica; Jakyung, Yoo; Fabian López, Vallejo; Paola, Conti; Lucia, Tamborini; Andrea, Pinto; José L., Medina Franco; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm2010404 Codice identificativo ISI: WOS:000296408100020 Codice identificativo SCOPUS: 2-s2.0-80455173681 | |
| Show it in Product Database (IRIS) |
34306Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs)
| 2011 | |
| Articolo in rivista | |
| Modulation of the Activity of Histone Acetyltransferases by Long Chain Alkylidene-malonates (LoCAMs) BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 19. Pag.3690-3701 ISSN:1464-3391. | |
| Milite, Ciro; Castellano, Sabrina; Benedetti, Rosaria; Tosco, Alessandra; Ciliberti, Carmen; Vicidomini, Caterina; Boully, Ludovic; Franci, Gianluigi; Altucci, Lucia; Mai, Antonello; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2011.01.013 Codice identificativo ISI: WOS:000291477600010 Codice identificativo SCOPUS: 2-s2.0-79958265044 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA. Vol. 108. Pag.2795-2800 ISSN:0027-8424. | |
| Claudia, Colussi; Jessica, Rosati; Stefania, Straino; Francesco, Spallotta; Roberta, Berni; Donatella, Stilli; Stefano, Rossi; Ezio, Musso; Emilio, Macchi; Antonello, Mai; Sbardella, Gianluca; Castellano, Sabrina; Cristina, Chimenti; Andrea, Frustaci; Angela, Nebbioso; Lucia, Altucci; Maurizio C., Capogrossi; Carlo, Gaetano | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1073/pnas.1013124108 Codice identificativo ISI: WOS:000287377000035 Codice identificativo SCOPUS: 2-s2.0-79952613152 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54. Pag.5927-5936 ISSN:0022-2623. | |
| Sbardella, Gianluca; Mai, Antonello; Bartolini, Sara; Castellano, Sabrina; Cirilli, Roberto; Rotili, Dante; Milite, Ciro; Santoriello, Marisabella; Orlando, Serena; Sciamanna, Ilaria; Serafino, Annalucia; Lavia, Patrizia; Spadafora, Corrado | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm200734j Codice identificativo ISI: WOS:000294077300023 Codice identificativo SCOPUS: 2-s2.0-80051873043 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Chemical biology of Histone acetyltransferase natural compounds modulators. MOLECULAR DIVERSITY. Vol. 15. Pag.401-416 ISSN:1381-1991. | |
| DAL PIAZ, Fabrizio; Vassallo, Antonio; Osmany Cuesta, Rubio; Castellano, Sabrina; Sbardella, Gianluca; DE TOMMASI, Nunziatina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1007/s11030-010-9299-5 Codice identificativo ISI: WOS:000290042900010 Codice identificativo SCOPUS: 2-s2.0-80051572654 | |
| Show it in Product Database (IRIS) |
| 2011 | |
| Articolo in rivista | |
| Novel 3,5-Bis(bromohydroxybenzylidene)piperidin-4-ones as Coactivator-associated Arginine Methyltransferase 1 Inhibitors: Enzyme Selectivity and Cellular Activity. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 54. Pag.4928-4932 ISSN:0022-2623. | |
| Donghang, Cheng; Sergio, Valente; Castellano, Sabrina; Sbardella, Gianluca; Roberto Di, Santo; Roberta, Costi; Mark T., Bedford; Antonello, Mai | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm200453n Codice identificativo ISI: WOS:000292479600049 Codice identificativo SCOPUS: 2-s2.0-79960191524 | |
| Show it in Product Database (IRIS) |
34538Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees.
| 2011 | |
| Articolo in rivista | |
| Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees. EMBO REPORTS. Vol. 12. Pag.238-243 ISSN:1469-221X. | |
| Astrid, Spannhoff; Yong Kee, Kim; Noel J. M., Raynal; Vazganush, Gharibyan; Ming Bo, Su; Yue Yang, Zhou; Jia, Li; Castellano, Sabrina; Sbardella, Gianluca; Jean Pierre J., Issa; Mark T., Bedford | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1038/embor.2011.9 Codice identificativo ISI: WOS:000287961800016 Codice identificativo SCOPUS: 2-s2.0-79952280451 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Abstract in rivista | |
| ChemInform Abstract: A Simplified Synthesis of Ethyl 5-Chloro-4-fluoro-1H-indole-2-carboxylate and Ethyl 5-Chloro-6-fluoro-1H-indole-2-carboxylate CHEM INFORM. Vol. 33. Pag.no-no ISSN:0931-7597. | |
| Silvestri, Romano; De Martino, Gabriella; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.200252113 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Abstract in rivista | |
| ChemInform Abstract: N-[4-(1,1′-Biphenyl)methyl]-4-(4-thiomorpholinylmethyl)benzenamines as Non-oxazolidinone Analogues of Antimycobacterial U-100480 CHEM INFORM. Vol. 29. Pag.no-no ISSN:0931-7597. | |
| Artico, M.; Mai, A.; Sbardella, Gianluca; Massa, S.; Lampis, G.; Deidda, D.; Pompei, R. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.199840169 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Abstract in rivista | |
| ChemInform Abstract: A New Facile and Expeditious Synthesis of N-Hydroxy-N′-phenyloctanediamide, a Potent Inducer of Terminal Cytodifferentiation CHEM INFORM. Vol. 32. Pag.no-no ISSN:0931-7597. | |
| Mai, Antonello; Esposito, Monica; Sbardella, Gianluca; Massa, Silvio | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.200144085 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Abstract in rivista | |
| ChemInform Abstract: Nitroquinolones with Broad-Spectrum Antimycobacterial Activity in vitro CHEM INFORM. Vol. 30. Pag.no-no ISSN:0931-7597. | |
| Artico, Marino; Mai, Antonello; Sbardella, Gianluca; Massa, Silvio; Musiu, Chiara; Lostia, Stefania; Demontis, Francesca; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.199937151 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Articolo in rivista | |
| Design, Synthesis and Biological Evaluation of Carboxy Analogues of Arginine Methyltransferase Inhibitor 1 (AMI-1) CHEMMEDCHEM. Vol. 5. Pag.398-414 ISSN:1860-7179. | |
| Castellano, Sabrina; Milite, Ciro; Ragno, R; Simeoni, S; Mai, A; Limongelli, V; Novellino, E; Bauer, I; Brosch, G; Spannhoff, A; Cheng, Dh; Bedford, Mt; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.200900459 Codice identificativo ISI: WOS:000275521200009 Codice identificativo SCOPUS: 2-s2.0-77249086700 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Articolo in rivista | |
| Synthesis of 3-Aryl/benzyl-4,5,6,6a-tetrahydro-3aH-pyrrolo[3,4-d]isoxazole Derivatives: A Comparison between Conventional, Microwave-Assisted and Flow-Based Methodologies. JOURNAL OF ORGANIC CHEMISTRY. Vol. 75. Pag.7439-7442 ISSN:0022-3263. | |
| Castellano, Sabrina; Lucia, Tamborini; Viviano, Monica; Andrea, Pinto; Sbardella, Gianluca; Paola, Conti | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jo1014323 Codice identificativo ISI: WOS:000283531100051 Codice identificativo SCOPUS: 2-s2.0-78049513527 | |
| Show it in Product Database (IRIS) |
| 2010 | |
| Articolo in rivista | |
| The identification of a novel natural activator of p300 Histone acetyltranferase provides new insights into the modulation mechanism of this enzyme CHEMBIOCHEM. Vol. 11. Pag.818-827 ISSN:1439-4227. | |
| DAL PIAZ, Fabrizio; Tosco, Alessandra; Eletto, Daniela; Piccinelli, ANNA LISA; Moltedo, Ornella; Franceschelli, Silvia; Sbardella, Gianluca; Remondelli, Paolo; Rastrelli, Luca; Loredana, Vesci; Claudio, Pisano; DE TOMMASI, Nunziatina | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cbic.200900721 Codice identificativo ISI: WOS:000277299800015 Codice identificativo SCOPUS: 2-s2.0-77950663978 | |
| Show it in Product Database (IRIS) |
| 2009 | |
| Articolo in rivista | |
| A regioselective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems TETRAHEDRON LETTERS. Vol. 50. Pag.6869-6871 ISSN:0040-4039. | |
| Castellano, Sabrina; Santoriello, Marisabella; Campiglia, Pietro; Cardillo, Giovanna; Bertamino, Alessia; Gomez Monterrey, Isabel; Novellino, Ettore; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.tetlet.2009.09.123 Codice identificativo ISI: WOS:000271603000037 Codice identificativo SCOPUS: 2-s2.0-70350038058 | |
| Show it in Product Database (IRIS) |
| 2009 | |
| Articolo in rivista | |
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 19. Pag.1132-1135 ISSN:0960-894X. | |
| Mai, A; Rotili, D; Tarantino, D; Nebbioso, A; Castellano, Sabrina; Sbardella, Gianluca; Tini, M; Altucci, L. | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2008.12.097 Codice identificativo ISI: WOS:000263295200021 Codice identificativo SCOPUS: 2-s2.0-59749103028 | |
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| 2008 | |
| Abstract in rivista | |
| ChemInform Abstract: A Practical, Green, and Selective Approach Toward the Synthesis of Pharmacologically Important Quinone-Containing Heterocyclic Systems Using Alumina-Catalyzed Michael Addition Reaction CHEM INFORM. Vol. 39. Pag.N/A-N/A ISSN:0931-7597. | |
| Castellano, Sabrina; Bertamino, Alessia; Gomez Monterrey, Isabel; Santoriello, Marisabella; Grieco, Paolo; Campiglia, Pietro; Sbardella, Gianluca; Novellino, Ettore | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/chin.200819096 | |
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20660Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1.
| 2008 | |
| Articolo in rivista | |
| Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 51. Pag.2321-2325 ISSN:0022-2623. | |
| Castellano, Sabrina; Kuck, D; Sala, Marina; Novellino, E; Lyko, F; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm7015705 Codice identificativo ISI: WOS:000254709100040 Codice identificativo SCOPUS: 2-s2.0-41849128470 | |
| Show it in Product Database (IRIS) |
| 2008 | |
| Articolo in rivista | |
| Epigenetic Multiple Ligands: Mixed Histone/Protein Methyltransferase, Acetyltransferase, and Class III Deacetylase (Sirtuin) Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 51. Pag.2279-2290 ISSN:0022-2623. | |
| Mai, Antonello; Cheng, Donghang; Bedford, Mark T.; Valente, Sergio; Nebbioso, Angela; Perrone, Andrea; Brosch, Gerald; Sbardella, Gianluca; De Bellis, Floriana; Miceli, Marco; Altucci, Lucia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm701595q Codice identificativo ISI: WOS:000254709100033 Codice identificativo SCOPUS: 2-s2.0-41849146748 | |
| Show it in Product Database (IRIS) |
| 2008 | |
| Articolo in rivista | |
| A practical, green and selective approach toward the synthesis of pharmacologically important quinone-containing heterocyclic systems using alumina-catalyzed Michael addition reaction. TETRAHEDRON LETTERS. Vol. 49. Pag.583-585 ISSN:0040-4039. | |
| Castellano, Sabrina; Bertamino, Alessia; Gomez Monterrey, Isabel; Santoriello, Marisabella; Grieco, Paolo; Campiglia, Pietro; Sbardella, Gianluca; Novellino, Ettore | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.tetlet.2007.11.148 Codice identificativo ISI: WOS:000253279200001 Codice identificativo SCOPUS: 2-s2.0-37549035077 | |
| Show it in Product Database (IRIS) |
| 2008 | |
| Articolo in rivista | |
| Identification of Long Chain Alkylidenemalonates as Novel Small Molecule Modulators of Histone Acetyltransferases BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 18. Pag.2788-2792 ISSN:0960-894X. | |
| Sbardella, Gianluca; Castellano, Sabrina; Vicidomini, C; Rotili, D; Nebbioso, A; Miceli, M; Altucci, L; Mai, A. | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2008.04.017 Codice identificativo ISI: WOS:000255444300005 Codice identificativo SCOPUS: 2-s2.0-42949089945 | |
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| 2008 | |
| Articolo in rivista | |
| CYP19 (Aromatase): Exploring the Scaffold Flexibility for Novel Selective Inhibitors. BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 16. Pag.8349-8358 ISSN:0968-0896. | |
| Castellano, Sabrina; Stefancich, G; Ragno, R; Schewe, K; Santoriello, M; Caroli, A; Hartmann, R. W.; Sbardella, Gianluca | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2008.08.046 Codice identificativo ISI: WOS:000259173400004 Codice identificativo SCOPUS: 2-s2.0-51449099183 | |
| Show it in Product Database (IRIS) |
| 2007 | |
| Articolo in rivista | |
| Synthesis and Biological Properties of Novel 2-Aminopyrimidin-4(3H)-ones Highly Potent against HIV-1 Mutant Strains JOURNAL OF MEDICINAL CHEMISTRY. Vol. 50. Pag.5412-5424 ISSN:0022-2623. | |
| Mai, Antonello; Artico, Marino; Rotili, Dante; Tarantino, Domenico; Clotet Codina, Imma; Armand Ugón, Mercedes; Ragno, Rino; Simeoni, Silvia; Sbardella, Gianluca; Nawrozkij, Maxim B.; Samuele, Alberta; Maga, Giovanni; Esté, José A. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm070811e Codice identificativo ISI: WOS:000250557100019 Codice identificativo SCOPUS: 2-s2.0-35848949355 | |
| Show it in Product Database (IRIS) |
17718Synthesis and Biological Validation of Novel Synthetic Histone/Protein Methyltransferase Inhibitors
| 2007 | |
| Articolo in rivista | |
| Synthesis and Biological Validation of Novel Synthetic Histone/Protein Methyltransferase Inhibitors CHEMMEDCHEM. Vol. 2. Pag.987-991 ISSN:1860-7179. | |
| Mai, A; Valente, S; Cheng, D; Perrone, A; Ragno, R; Simeoni, S; Sbardella, Gianluca; Brosch, G; Nebbioso, A; Conte, M; Altucci, L; Bedford, M. T. | |
| Digital Object Identifier (DOI): 10.1002/cmdc.200700023 Codice identificativo ISI: WOS:000248065600003 Codice identificativo SCOPUS: 2-s2.0-41849112166 | |
| Show it in Product Database (IRIS) |
| 2007 | |
| Articolo in rivista | |
| Slow-, Tight-Binding HIV-1 Reverse Transcriptase Non-Nucleoside Inhibitors Highly Active against Drug-Resistant Mutants CHEMMEDCHEM. Vol. 2. Pag.445-448 ISSN:1860-7179. | |
| Cancio, R; Mai, A; Rotili, D; Artico, M; Sbardella, Gianluca; CLOTET CODINA, I; Est, J. A.; Crespan, E; Zanoli, S; Hbscher, U; Spadari, S; Maga, G. | |
| Digital Object Identifier (DOI): 10.1002/cmdc.200600310 Codice identificativo ISI: WOS:000246011500006 Codice identificativo SCOPUS: 2-s2.0-34547939030 | |
| Show it in Product Database (IRIS) |
| 2007 | |
| Articolo in rivista | |
| Small Molecule Inhibitors of Histone Arginine Methyltransferases: Homology Modeling, Molecular Docking, Binding Mode Analysis and Biological Evaluations JOURNAL OF MEDICINAL CHEMISTRY. Vol. 50. Pag.1241-1253 ISSN:0022-2623. | |
| Ragno, R; Simeoni, S; Castellano, Sabrina; Vicidomini, C; Mai, A; Caroli, A; Tramontano, A; Bonaccini, C; Trojer, P; Bauer, I; Brosch, G; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm061213n Codice identificativo ISI: WOS:000244895900016 Codice identificativo SCOPUS: 2-s2.0-33947685838 | |
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| 2007 | |
| Articolo in rivista | |
| Highly efficient synthesis and chemical separation of 5-amino- and 7-amino-4-hydroxy-2-naphthoic acids TETRAHEDRON LETTERS. Vol. 48. Pag.4653-4655 ISSN:0040-4039. | |
| Castellano, Sabrina; Milite, Ciro; Campiglia, Pietro; Sbardella, Gianluca | |
| Digital Object Identifier (DOI): 10.1016/j.tetlet.2007.05.040 Codice identificativo ISI: WOS:000247559500001 Codice identificativo SCOPUS: 2-s2.0-34249914804 | |
| Show it in Product Database (IRIS) |
| 2007 | |
| Brevetto | |
| SELECTIVE INHIBITORS FOR TRANSFERASES WO 2007149782 University of Medicine and Dentistry New Jersey | |
| Reinberg, D; Trojer, P; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 2006 | |
| Articolo in rivista | |
| Small-Molecule Inhibitors of Histone Acetyltransferase Activity: Identification and Biological Properties JOURNAL OF MEDICINAL CHEMISTRY. Vol. 49. Pag.6897-6907 ISSN:0022-2623. | |
| Mai, Antonello; Rotili, Dante; Tarantino, Domenico; Ornaghi, Prisca; Tosi, Federica; Vicidomini, Caterina; Sbardella, Gianluca; Nebbioso, Angela; Miceli, Marco; Altucci, Lucia; Filetici, Patrizia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm060601m Codice identificativo ISI: WOS:000241894000031 Codice identificativo SCOPUS: 2-s2.0-33750989910 | |
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| 2006 | |
| Articolo in rivista | |
| Identification of small molecules inhibitors of GCN5 histone acetyltransferase activity. ARKIVOC. Vol. VIII. Pag.24-37 ISSN:1551-7004. | |
| Mai, Antonello; Rotili, Dante; Ornaghi, Prisca; Tosi, Federica; Vicidomini, Caterina; Sbardella, Gianluca; Nebbioso, Angela; Altucci, Lucia; Filetici, Patrizia | |
| Versione online | |
| Codice identificativo ISI: WOS:000242574600004 Codice identificativo SCOPUS: 2-s2.0-33744470562 | |
| Show it in Product Database (IRIS) |
| 2006 | |
| Articolo in rivista | |
| 6-Alkylthio-4-[1-(2,6-difluorophenyl)alkyl]-1H-[1,3,5]triazin-2-ones (ADATs): Novel Regulators of Cell Differentiation and Proliferation CHEMMEDCHEM. Vol. 1. Pag.1073-1080 ISSN:1860-7179. | |
| Sbardella, Gianluca; Bartolini, S; Castellano, Sabrina; Artico, M; Paesano, N; Rotili, D; Spadafora, C; Mai, A. | |
| Digital Object Identifier (DOI): 10.1002/cmdc.200600139 Codice identificativo ISI: WOS:000202946300006 Codice identificativo SCOPUS: 2-s2.0-33750284393 | |
| Show it in Product Database (IRIS) |
| 2005 | |
| Articolo in rivista | |
| 3-(1H-Pyrrol-2-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors MEDICINAL CHEMISTRY. Vol. 1. Pag.117-124 ISSN:1573-4064. | |
| Mai, Antonello; Artico, Marino; Valente, Sergio; Sbardella, Gianluca; Turini, Paola; Befani, Olivia; Dalla Vedova, Laura; Agostinelli, Enzo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.2174/1573406053175247 Codice identificativo SCOPUS: 2-s2.0-33846116762 | |
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| 2005 | |
| Articolo in rivista | |
| 5-Alkyl-2-alkylamino-6-(2,6-difluorophenylalkyl)-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones, a New Series of Potent, Broad-Spectrum Non-Nucleoside Reverse Transcriptase Inhibitors Belonging to the DABO family BIOORGANIC & MEDICINAL CHEMISTRY. Vol. 13. Pag.2065-2077 ISSN:0968-0896. | |
| Mai, Antonello; Artico, Marino; Ragno, Rino; Sbardella, Gianluca; Massa, Silvio; Musiu, Claudia; Mura, Massimo; Marturana, Flavia; Cadeddu, Alessandra; Maga, Giovanni; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmc.2005.01.005 Codice identificativo ISI: WOS:000227576700017 Codice identificativo SCOPUS: 2-s2.0-13844316071 | |
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| 2005 | |
| Articolo in rivista | |
| Synthesis and biological evaluation of 3-benzyl-1-methyl- and 1-methyl-3-phenyl-isothioureas as potential inhibitors of iNOS BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 15. Pag.539-543 ISSN:0960-894X. | |
| Paesano, Nicola; Marzocco, Stefania; Vicidomini, Caterina; Saturnino, Carmela; Autore, Giuseppina; DE MARTINO, Giovanni; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2004.11.047 Codice identificativo ISI: WOS:000226935700010 Codice identificativo SCOPUS: 2-s2.0-12444284865 | |
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| 2005 | |
| Articolo in rivista | |
| A novel Gcn5p inhibitor represses cell growth, gene transcription and histone acetylation in budding yeast BIOCHEMICAL PHARMACOLOGY. Vol. 70. Pag.911-917 ISSN:0006-2952. | |
| Ornaghi, Prisca; Rotili, Dante; Sbardella, Gianluca; Mai, Antonello; Filetici, Patrizia | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bcp.2005.06.013 Codice identificativo ISI: WOS:000231663100011 Codice identificativo SCOPUS: 2-s2.0-23744453206 | |
| Show it in Product Database (IRIS) |
| 2005 | |
| Articolo in rivista | |
| 6-[1-(2,6-Difluorophenyl)ethyl]pyrimidinones Antagonize Cell Proliferation and Induce Cell Differentiation by Inhibiting (a Non Telomeric) Endogenous Reverse Transcriptase JOURNAL OF MEDICINAL CHEMISTRY. Vol. 48. Pag.6776-6778 ISSN:0022-2623. | |
| Bartolini, S; Mai, A; Artico, M; Paesano, N; Rotili, D; Spadafora, C; Sbardella, Gianluca | |
| Digital Object Identifier (DOI): 10.1021/jm0507330 Codice identificativo ISI: WOS:000233017300003 Codice identificativo SCOPUS: 2-s2.0-27444434731 | |
| Show it in Product Database (IRIS) |
| 2004 | |
| Articolo in rivista | |
| New 6-nitroquinolones: synthesis and antimicrobial activities IL FARMACO. Vol. 59. Pag.463-471 ISSN:0014-827X. | |
| Sbardella, Gianluca; Mai, Antonello; Artico, Marino; Setzu, Maria Giovanna; Poni, Graziella; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.farmac.2004.01.014 Codice identificativo SCOPUS: 2-s2.0-2642513828 | |
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| 2004 | |
| Articolo in rivista | |
| Synthesis and in vitro antimycobacterial activity of novel 3-(1H-pyrrol-1-yl)-2-oxazolidinone analogues of PNU-100480 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 14. Pag.1537-1541 ISSN:0960-894X. | |
| Sbardella, Gianluca; Mai, Antonello; Artico, Marino; Loddo, Roberta; Setzu, Maria Giovanna; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.bmcl.2004.01.010 Codice identificativo ISI: WOS:000220334000035 Codice identificativo SCOPUS: 2-s2.0-1542284725 | |
| Show it in Product Database (IRIS) |
| 2004 | |
| Articolo in rivista | |
| Computer-Aided Design, Synthesis, and Anti-HIV-1 Activity in Vitro of 2-Alkylamino-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)- ones as Novel Potent Non-Nucleoside Reverse Transcriptase Inhibitors, Also Active Against the Y181C Variant JOURNAL OF MEDICINAL CHEMISTRY. Vol. 47. Pag.928-934 ISSN:0022-2623. | |
| Ragno, Rino; Mai, Antonello; Sbardella, Gianluca; Artico, Marino; Massa, Silvio; Musiu, Chiara; Mura, Massimo; Marturana, Flavia; Cadeddu, Alessandra; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm0309856 Codice identificativo ISI: WOS:000188831300015 Codice identificativo SCOPUS: 2-s2.0-10744230514 | |
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| 2004 | |
| Brevetto | |
| Preparation of oxo-pyrimidine compounds for use in pharmaceutical compositions for the treatment of retroviral infection, particularly HIV infection WO 2004096147 Idenix Cayman Limited, Cayman I. | |
| Storer, Richard; Moussa, Adel; La Colla, Paolo; Mai, Antonello; Sbardella, Gianluca; Artico, Marino | |
| Show it in Product Database (IRIS) |
| 2003 | |
| Articolo in rivista | |
| Synthesis and biological evaluation of enantiomerically pure pyrrolyl-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors IL FARMACO. Vol. 58. Pag.231-241 ISSN:0014-827X. | |
| Mai, A; Artico, M; Esposito, M; Ragno, R; Sbardella, Gianluca; Massa, S. | |
| Digital Object Identifier (DOI): 10.1016/S0014-827X(03)00016-8 Codice identificativo SCOPUS: 2-s2.0-0037373722 | |
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| 2002 | |
| Articolo in rivista | |
| Binding Mode Analysis of 3-(4-Benzoyl-1-methyl-1H-2-pyrrolyl)-N-hydroxy-2-propenamide: A New Synthetic Histone Deacetylase Inhibitor Inducing Histone Hyperacetylation, Growth Inhibition, and Terminal Cell Differentiation JOURNAL OF MEDICINAL CHEMISTRY. Vol. 45. Pag.1778-1784 ISSN:0022-2623. | |
| Mai, Antonello; Massa, Silvio; Ragno, Rino; Esposito, Monica; Sbardella, Gianluca; Nocca, Giuseppina; Scatena, Roberto; Jesacher, Florian; Loidl, Peter; Brosch, Gerald | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm011088+ Codice identificativo ISI: WOS:000175168700006 Codice identificativo SCOPUS: 2-s2.0-0037171823 | |
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| 2002 | |
| Articolo in rivista | |
| 3-(1H-Pyrrol-2- and -3-yl)-2-oxazolidinones as Novel Monoamine Oxidase Type A Inhibitors DRUGS OF THE FUTURE. Vol. 27 suppl. A. Pag.438-438 ISSN:0377-8282. | |
| Sbardella, Gianluca; A., Mai; M., Esposito; M., Artico; S., Massa; O., Befani; V., Giovannini; B., Mondovì | |
| Show it in Product Database (IRIS) |
| 2002 | |
| Articolo in rivista | |
| A simplified synthesis of ethyl 5-chloro-6-fluoro-1H-indole-2-carboxylate and ethyl 5-chloro-4-fluoro-1H-indole-2-carboxylate ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL. Vol. 34. Pag.507-510 ISSN:0030-4948. | |
| Silvestri, Romano; De Martino, Gabriella; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1080/00304940209355772 Codice identificativo ISI: WOS:000178252000010 Codice identificativo SCOPUS: 2-s2.0-0036796527 | |
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| 2002 | |
| Articolo in rivista | |
| Computer-Aided Design of Novel Aroyl-pyrrolyl-hydroxy-alkylamide (APHA) Derivatives as New Synthetic Histone Deacetylase Inhibitors. DRUGS OF THE FUTURE. Vol. 27 suppl. A. Pag.441-441 ISSN:0377-8282. | |
| A., Mai; I., Cerbara; S., Massa; R., Ragno; Sbardella, Gianluca; F., Jesacher; G., Brosch; P., Loidl | |
| Show it in Product Database (IRIS) |
| 2002 | |
| Articolo in rivista | |
| Anti-HIV-1 Activity of Arylthiazolylcarboxyamides, a novel class of NNRTIs as Hybrid Congeners between PETT, UC781 and TDA DRUGS OF THE FUTURE. Vol. 27 suppl. A. Pag.440-440 ISSN:0377-8282. | |
| Sbardella, Gianluca; N., Paesano; R., Silvestri; G., DE MARTINO; M., Artico; R., Ragno; R., Loddo; M., LA COLLA; P., LA COLLA; M. E., Marongiu; A., Pani | |
| Show it in Product Database (IRIS) |
| 2002 | |
| Articolo in rivista | |
| Synthesis and biological evaluation of enantiomerically pure 3-(1H-Pyrrol-1-yl)-2-oxazolidinones as a new class of potent and selective monoamine oxidase type A inhibitors DRUGS OF THE FUTURE. Vol. 27 suppl. A. Pag.439-439 ISSN:0377-8282. | |
| Sbardella, Gianluca; A., Mai; M., Esposito; M., Artico; S., Massa; R., Ragno; O., Befani; V., Giovannini; B., Mondovì | |
| Show it in Product Database (IRIS) |
| 2002 | |
| Articolo in rivista | |
| 3-(1H-Pyrrol-1-yl)-2-oxazolidinones as Reversible, Highly Potent, and Selective Inhibitors of Monoamine Oxidase Type A JOURNAL OF MEDICINAL CHEMISTRY. Vol. 45. Pag.1180-1183 ISSN:0022-2623. | |
| Mai, Antonello; Artico, Marino; Esposito, Monica; Sbardella, Gianluca; Massa, Silvio; Befani, Olivia; Turini, Paola; Giovannini, Valentina; Mondovì, Bruno | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm015578d Codice identificativo ISI: WOS:000174506200003 Codice identificativo SCOPUS: 2-s2.0-0037075787 | |
| Show it in Product Database (IRIS) |
| 2002 | |
| Brevetto | |
| Methods for inhibiting the transmission of HIV using topically applied substituted 6-benzyl-4-oxopyrimidines WO 2002040021 Novirio Pharmaceuticals Limited, Cayman I.; Universita Degli Studi Di Cagliari | |
| Sommadossi, Jean Pierre; La Colla, Paolo; Artico, Marino; Mai, Antonello; Sbardella, Gianluca; Bryant, Martin L. | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Articolo in rivista | |
| Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class. CHIRALITY. Vol. 13. Pag.75-80 ISSN:0899-0042. | |
| Quaglia, M. G.; Mai, A.; Sbardella, Gianluca; Artico, M.; Ragno, R.; Massa, S.; DEL PIANO, D.; Setzu, G.; Doratiotto, S.; Cotichini, V. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/1520-636X(2001)13:2<75::AID-CHIR1001>3.0.CO;2-W Codice identificativo ISI: WOS:000166596300002 Codice identificativo SCOPUS: 2-s2.0-0035146092 | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Articolo in rivista | |
| A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL. Vol. 33. Pag.391-394 ISSN:0030-4948. | |
| Mai, A; Esposito, M; Sbardella, Gianluca; Massa, S. | |
| Codice identificativo ISI: WOS:000169959200013 Codice identificativo SCOPUS: 2-s2.0-0035536590 | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Articolo in rivista | |
| Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase JOURNAL OF MEDICINAL CHEMISTRY. Vol. 44. Pag.2544-2554 ISSN:0022-2623. | |
| Mai, Antonello; Sbardella, Gianluca; Artico, Marino; Ragno, Rino; Massa, Silvio; Novellino, Ettore; Greco, Giovanni; Lavecchia, Aantonio; Musiu, Chiara; La Colla, Massimiliano; Murgioni, Chiara; La Colla, Paolo; Loddo, Roberta | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm010853h Codice identificativo ISI: WOS:000170167700007 Codice identificativo SCOPUS: 2-s2.0-0035797356 | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Articolo in rivista | |
| Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity ANTIVIRAL CHEMISTRY & CHEMOTHERAPY. Vol. 12. Pag.37-50 ISSN:0956-3202. | |
| Sbardella, Gianluca; A., Mai; M., Artico; P., Chimenti; S., Massa; R., Loddo; M. E., Marongiu; P., LA COLLA; A., Pani | |
| Codice identificativo SCOPUS: 2-s2.0-0034975054 | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Articolo in rivista | |
| 3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors JOURNAL OF MEDICINAL CHEMISTRY. Vol. 44. Pag.2069-2072 ISSN:0022-2623. | |
| Silvio, Massa; Antonello, Mai; Sbardella, Gianluca; Monica, Esposito; Rino, Ragno; Peter, Loidl; Gerald, Brosch | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm015515v Codice identificativo ISI: WOS:000169367000004 Codice identificativo SCOPUS: 2-s2.0-0035927427 | |
| Show it in Product Database (IRIS) |
| 2001 | |
| Contributo in volume (Capitolo o Saggio) | |
| 3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors. In Recent developments in antiviral research Pag.65-92 Trivandrum Transworld Research Network. ISBN:817895012X | |
| M., Elena Marongiu; Alessandra, Pani; Chiara, Musiu; Paolo La, Colla; Antonello, Mai; Sbardella, Gianluca; Silvio, Massa; Marino, Artico | |
| Show it in Product Database (IRIS) |
| 2000 | |
| Articolo in rivista | |
| Does the 2-methylthiomethyl substituent really confer high anti-HIV-1 activity to S-DABOs ? MEDICINAL CHEMISTRY RESEARCH. Vol. 10. Pag.30-39 ISSN:1054-2523. | |
| Sbardella, Gianluca; Mai, A.; Artico, M.; Massa, S.; Marceddu, T.; Vargiu, L.; Marongiu, M. E.; LA COLLA, P. | |
| Codice identificativo SCOPUS: 2-s2.0-0033943608 | |
| Show it in Product Database (IRIS) |
| 2000 | |
| Brevetto | |
| Preparation of substituted 6-benzyl-4-oxopyrimidines for prevention and treatment of HIV infection WO 2000003998 Novirio Pharmaceuticals Limited, Cayman I. | |
| La Colla, Paolo; Mai, Antonello; Sbardella, Gianluca; Artico, Marino | |
| Show it in Product Database (IRIS) |
| 1999 | |
| Articolo in rivista | |
| N-[4-(1,1'-biphenylyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines, a new class of synthetic antituberculosis agents active against Mycobacterium avium. MEDICINAL CHEMISTRY RESEARCH. Vol. 9. Pag.149-161 ISSN:1054-2523. | |
| Mai, A.; Sbardella, Gianluca; Artico, M.; Massa, S.; Lampis, G.; Deidda, D.; Pompei, R. | |
| Codice identificativo ISI: WOS:000080663900001 Codice identificativo SCOPUS: 2-s2.0-0032996022 | |
| Show it in Product Database (IRIS) |
| 1999 | |
| Articolo in rivista | |
| 5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4( 3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 42. Pag.619-627 ISSN:0022-2623. | |
| Mai, Antonello; Artico, Marino; Sbardella, Gianluca; Massa, Silvio; Novellino, Ettore; Greco, Giovanni; Loi, Anna Giulia; Tramontano, Enzo; Marongiu, Maria Elena; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm980260f Codice identificativo ISI: WOS:000078826300011 Codice identificativo SCOPUS: 2-s2.0-0033602141 | |
| Show it in Product Database (IRIS) |
| 1999 | |
| Articolo in rivista | |
| Nitroquinolones with broad-spectrum antimycobacterial activity in vitro. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 9. Pag.1651-1656 ISSN:0960-894X. | |
| Artico, Marino; Mai, Antonello; Sbardella, Gianluca; Massa, Silvio; Musiu, Chiara; Lostia, Stefania; Demontis, Francesca; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/S0960-894X(99)00251-6 Codice identificativo ISI: WOS:000080896500005 Codice identificativo SCOPUS: 2-s2.0-0033591758 | |
| Show it in Product Database (IRIS) |
| 1998 | |
| Articolo in rivista | |
| Crystal structure of 3,4-dihydro-6-(3¢-methylbenzyl)-2-[(1-methyl-propyl)thio]-4-oxopyrimidine (S-DABO 618), C16H20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors ZEITSCHRIFT FUR KRISTALLOGRAPHIE. NEW CRYSTAL STRUCTURES. Vol. 213. Pag.593-595 ISSN:1433-7266. | |
| A., Ettorre; A., Mai; Sbardella, Gianluca; M., Artico; P., LA COLLA; S., Massa | |
| Codice identificativo ISI: WOS:000074680700076 Codice identificativo SCOPUS: 2-s2.0-22044439538 | |
| Show it in Product Database (IRIS) |
| 1998 | |
| Articolo in rivista | |
| Crystal structure of 3,4-dihydro-6-(3′-methylbenzyl)-2-[(1-methylpropyl)thio]-4-oxopyrimidine (S-DABO 618), C16H2O20N2OS and of 3,4-dihydro-2-[(1-methylpropyl)thio]-6-(2-naphthylmethyl)-4-oxopyrimidine (DATNO 774), C19H20N2OS, two HIV-1 reverse transcriptase inhibitors ZEITSCHRIFT FUR KRISTALLOGRAPHIE. NEW CRYSTAL STRUCTURES. Vol. 213. Pag.621-623 ISSN:1433-7266. | |
| Ettorre, A.; Mai, A.; Sbardella, G.; Artico, M.; La Colla, P.; Massa, S. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1524/ncrs.1998.213.14.621 Codice identificativo SCOPUS: 2-s2.0-85025246639 | |
| Show it in Product Database (IRIS) |
| 1998 | |
| Articolo in rivista | |
| N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmetyl)benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480 BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. Vol. 8. Pag.1493-1498 ISSN:0960-894X. | |
| M., Artico; A., Mai; Sbardella, Gianluca; S., Massa; G., Lampis; D., Deidda; R., Pompei | |
| Digital Object Identifier (DOI): 10.1016/S0960-894X(98)00248-0 Codice identificativo ISI: WOS:000074291800010 Codice identificativo SCOPUS: 2-s2.0-0032537533 | |
| Show it in Product Database (IRIS) |
| 1997 | |
| Articolo in rivista | |
| Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: novel non-nucleoside reverse transcriptase inhibitors of the S-DABO series. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 40. Pag.1447-1454 ISSN:0022-2623. | |
| Mai, Antonello; Artico, Marino; Sbardella, Gianluca; Quartarone, Silvana; Massa, Silvio; Loi, Anna Giulia; De Montis, Antonella; Scintu, Franca; Putzolu, Monica; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm960802y Codice identificativo ISI: WOS:A1997WY39500005 Codice identificativo SCOPUS: 2-s2.0-15444340492 | |
| Show it in Product Database (IRIS) |
| 1997 | |
| Articolo in rivista | |
| Arylketotetramethylene analogs of disoxaril with anti-human rhinovirus 14 activity. ANTIVIRAL CHEMISTRY & CHEMOTHERAPY. Vol. 8. Pag.235-242 ISSN:0956-3202. | |
| Antonello, Mai; Marino, Artico; Sbardella, Gianluca; Silvio, Massa; Alessandra De, Montis; Ilaria, Puddu; Claudia, Musiu; Paolo La, Colla | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1177/095632029700800307 Codice identificativo ISI: WOS:A1997WY39600007 Codice identificativo SCOPUS: 2-s2.0-0031009277 | |
| Show it in Product Database (IRIS) |
| 1996 | |
| Brevetto | |
| Preparation of 6-benzyl-4-oxopyrimidines as antiviral agents WO 9610565 (A1) Istituto Superiore Di Sanita', Italy; Universita' Degli Studi Di Cagliari | |
| Artico, Marino; Massa, Silvio; Mai, Antonello; Sbardella, Gianluca; La Colla, Paolo; Marongiu, Maria Elena; Tramontano, Enzo | |
| Show it in Product Database (IRIS) |
| 1995 | |
| Articolo in rivista | |
| Synthesis and antiviral activity of new 3,4-dihydro-2-alkoxy-6-benzyl-4-oxopyrimidines (DABOs), specific inhibitors of human immunodeficiency virus type 1. ANTIVIRAL CHEMISTRY & CHEMOTHERAPY. Vol. 6. Pag.1-8 ISSN:0956-3202. | |
| Silvio, Massa; Antonello, Mai; Marino, Artico; Sbardella, Gianluca; Enzo, Tramontano; Anna Giulia, Loi; Patrizia, Scano; Paolo La, Colla | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1177/095632029500600101 Codice identificativo ISI: WOS:A1995QA06000001 Codice identificativo SCOPUS: 2-s2.0-0028869436 | |
| Show it in Product Database (IRIS) |
| 1995 | |
| Articolo in rivista | |
| Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines. JOURNAL OF MEDICINAL CHEMISTRY. Vol. 38. Pag.3258-3263 ISSN:0022-2623. | |
| Mai, Antonello; Artico, Marino; Sbardella, Gianluca; Massa, Silvio; Loi, Anna Giulia; Tramontano, Enzo; Scano, Patrizia; La Colla, Paolo | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/jm00017a010 Codice identificativo ISI: WOS:A1995RQ57600010 Codice identificativo SCOPUS: 2-s2.0-0029095334 | |
| Show it in Product Database (IRIS) |
| 1994 | |
| Contributo in Atti di convegno | |
| Synthesis and Antiviral Activity of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs), New Potent and Selective HIV-1 Inhibitors.. In: XI Convegno Nazionale. Divisione di Chimica Farmaceutica. Società Chimica Italiana. Atti del Congresso Pag.122-122 | |
| XI Convegno Nazionale. Divisione di Chimica Farmaceutica. Società Chimica Italiana Bari 2-5 Ottobre | |
| Mai, Antonello; Massa, Silvio; Sbardella, Gianluca; Quartarone, Silvana; Artico, Marino; Musu, Daniela; Doa, Manuela; Scano, Patrizia; La Colla, Paolo | |
| Show it in Product Database (IRIS) |
| 1994 | |
| Contributo in Atti di convegno | |
| DABOs: A New Class of Non-Nucleoside Reverse Transcriptase Inhibitors. In: Seventh Research Project on AIDS (1994). Operation plan Settimo progetto di ricerche sull'AIDS (1994). Piano esecutivo Istituto Superiore di Sanita', Rome (Italy) Pag.84-84 | |
| Seventh Research Project on AIDS Roma 4-8 luglio | |
| Tramontano, Enzo; Loi, Anna Giulia; De Montis, Antonella; Marongiu, Maria Elena; Scano, Patrizia; La Colla, Paolo; Artico, Marino; Massa, Silvio; Mai, Antonello; Sbardella, Gianluca | |
| Show it in Product Database (IRIS) |
| 1994 | |
| Contributo in Atti di convegno | |
| Synthesis of 2-Alkylthio-6-benzyl-3,4-dihydro-4-oxopyrimidines (DABOs) as Potent and Selective HIV-1 Inhibitors. In: Proceedings of the XIIIth International Symposium on Medicinal Chemistry, Paris, 1994 Paris Elsevier Vol.30, Pag.214-214 | |
| XIIIth International Symposium on Medicinal Chemistry Paris 19-23 September | |
| Mai, Antonello; Massa, Silvio; Sbardella, Gianluca; Artico, Marino; Musu, Daniela; Doa, Manuela; Scano, Patrizia; La Colla, Paolo | |
| Show it in Product Database (IRIS) |
