Gianluca SBARDELLA | Publications
Gianluca SBARDELLA Publications
| 2022 | |
| Articolo in rivista | |
| Age-dependent attenuation of spatial memory deficits by the histone acetyltransferase p300/CBP-associated factor (PCAF) in 3xTG Alzheimer's disease mice LEARNING & MEMORY. Vol. 29. Pag.71-76 ISSN:1549-5485. | |
| Creighton, Samantha D.; Jardine, Kristen H.; Desimone, Alexa; Zmetana, Megan; Castellano, Sabrina; Milite, Ciro; Sbardella, Gianluca; Winters, Boyer D. | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1101/lm.053536.121 Codice identificativo ISI: WOS:000757289600001 Codice identificativo SCOPUS: 2-s2.0-85124680497 | |
| Show it in Product Database (IRIS) |
| 2022 | |
| Articolo in rivista | |
| Discovery of benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain CHEMMEDCHEM. Vol. 17. Pag.1-14 ISSN:1860-7179. | |
| Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1002/cmdc.202200343 Codice identificativo ISI: WOS:000853917200001 Codice identificativo SCOPUS: 2-s2.0-85138079605 | |
| Show it in Product Database (IRIS) |
| 2022 | |
| Articolo in rivista | |
| Lysine methyltransferase inhibitors: where we are now. RSC CHEMICAL BIOLOGY. Vol. 3. Pag.359-406 ISSN:2633-0679. | |
| Feoli, Alessandra; Viviano, Monica; Cipriano, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1039/D1CB00196E Codice identificativo ISI: WOS:000739939100001 Codice identificativo SCOPUS: 2-s2.0-85129384483 | |
| Show it in Product Database (IRIS) |
| 2022 | |
| Articolo in rivista | |
| Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction-Reconstruction and Fragment-Growing Approach JOURNAL OF MEDICINAL CHEMISTRY. Vol. 65. Pag.11574-11606 ISSN:0022-2623. | |
| Iannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1021/acs.jmedchem.2c00252 Codice identificativo ISI: WOS:000822512300001 Codice identificativo SCOPUS: 2-s2.0-85129915280 | |
| Show it in Product Database (IRIS) |
| 2022 | |
| Articolo in rivista | |
| Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. Vol. 237. Pag.114410-114440 ISSN:0223-5234. | |
| Menna, Martina; Fiorentino, Francesco; Marrocco, Biagina; Lucidi, Alessia; Tomassi, Stefano; Cilli, Domenica; Romanenghi, Mauro; Cassandri, Matteo; Pomella, Silvia; Pezzella, Michele; Del Bufalo, Donatella; Zeya Ansari, Mohammad Salik; Tomašević, Nevena; Mladenović, Milan; Viviano, Monica; Sbardella, Gianluca; Rota, Rossella; Trisciuoglio, Daniela; Minucci, Saverio; Mattevi, Andrea; Rotili, Dante; Mai, Antonello | |
| Versione online | |
| Digital Object Identifier (DOI): 10.1016/j.ejmech.2022.114410 Codice identificativo ISI: WOS:000804176200002 Codice identificativo SCOPUS: 2-s2.0-85129352278 | |
| Show it in Product Database (IRIS) |
