Publications

Gianluca SBARDELLA Publications


2001
Articolo in rivista
3-(4-Aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a New Class of Synthetic Histone Deacetylase Inhibitors
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 44. Pag.2069-2072
ISSN:0022-2623.
Silvio, Massa; Antonello, Mai; Sbardella, Gianluca; Monica, Esposito; Rino, Ragno; Peter, Loidl; Gerald, Brosch
Versione online
Digital Object Identifier (DOI): 10.1021/jm015515v
Codice identificativo ISI: WOS:000169367000004
Codice identificativo SCOPUS: 2-s2.0-0035927427
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2001
Articolo in rivista
A new facile and expeditious synthesis of N-hydroxy-N'-phenyloctanediamide, a potent inducer of terminal cytodifferentiation
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL. Vol. 33. Pag.391-394
ISSN:0030-4948.
Mai, A; Esposito, M; Sbardella, Gianluca; Massa, S.
Codice identificativo ISI: WOS:000169959200013
Codice identificativo SCOPUS: 2-s2.0-0035536590
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2001
Articolo in rivista
Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5- methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class.
CHIRALITY. Vol. 13. Pag.75-80
ISSN:0899-0042.
Quaglia, M. G.; Mai, A.; Sbardella, Gianluca; Artico, M.; Ragno, R.; Massa, S.; DEL PIANO, D.; Setzu, G.; Doratiotto, S.; Cotichini, V.
Versione online
Digital Object Identifier (DOI): 10.1002/1520-636X(2001)13:2<75::AID-CHIR1001>3.0.CO;2-W
Codice identificativo ISI: WOS:000166596300002
Codice identificativo SCOPUS: 2-s2.0-0035146092
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2001
Articolo in rivista
Structure-activity relationship studies of new DABOs: effect of substitutions at the pyrimidine C-5 and C-6 positions on anti-HIV-1 activity
ANTIVIRAL CHEMISTRY & CHEMOTHERAPY. Vol. 12. Pag.37-50
ISSN:0956-3202.
Sbardella, Gianluca; A., Mai; M., Artico; P., Chimenti; S., Massa; R., Loddo; M. E., Marongiu; P., LA COLLA; A., Pani
Codice identificativo SCOPUS: 2-s2.0-0034975054
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2001
Articolo in rivista
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase
JOURNAL OF MEDICINAL CHEMISTRY. Vol. 44. Pag.2544-2554
ISSN:0022-2623.
Mai, Antonello; Sbardella, Gianluca; Artico, Marino; Ragno, Rino; Massa, Silvio; Novellino, Ettore; Greco, Giovanni; Lavecchia, Aantonio; Musiu, Chiara; La Colla, Massimiliano; Murgioni, Chiara; La Colla, Paolo; Loddo, Roberta
Versione online
Digital Object Identifier (DOI): 10.1021/jm010853h
Codice identificativo ISI: WOS:000170167700007
Codice identificativo SCOPUS: 2-s2.0-0035797356
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2001
Contributo in volume (Capitolo o Saggio)
3,4-Dihydro-2-alkoxy-6-benzyl-oxopyrimidines [DABOs]: Development of a potent class of non-nucleoside reverse transcriptase inhibitors.
In Recent developments in antiviral research Pag.65-92 Trivandrum Transworld Research Network.
ISBN:817895012X
M., Elena Marongiu; Alessandra, Pani; Chiara, Musiu; Paolo La, Colla; Antonello, Mai; Sbardella, Gianluca; Silvio, Massa; Marino, Artico
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